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2-(3,5-dimethyl-1H-pyrazol-1-yl)-1-[9-methoxy-7-(4-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]ethan-1-one
N-[2-(3-methylthiophen-2-yl)ethyl]-2-(1H-pyrazol-1-yl)butanamide
1-{[2-(2,4-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-(2-methylphenyl)piperazine
N-(2-methoxyethyl)-N-[(3-methylthiophen-2-yl)methyl]-2H,3H-thieno[3,4-b][1,4]dioxine-5-carboxamide
2-{1-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]-3-oxopiperazin-2-yl}-N-methyl-N-(propan-2-yl)acetamide
2-fluoro-N-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-5-sulfamoylbenzamide
2-(oxolan-2-yl)-1-{[3-(thiophen-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-1H-1,3-benzodiazole
3-methyl-5-(6-methyl-2H-1,3-benzodioxol-5-yl)-1-(2-methylpropyl)-1H,4H-pyrazolo[3,4-d]imidazole
methyl({[5-(1-methyl-1H-1,3-benzodiazol-2-yl)furan-2-yl]methyl})(oxan-4-ylmethyl)amine
2-{1-[(3-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-methyl-N-(oxan-4-yl)acetamide
6-(6-aminopyridin-3-yl)-N-[2-(2,3-dihydro-1,4-benzodioxin-2-yl)ethyl]pyridine-3-carboxamide
(3R,5R)-N-[(2-ethyl-4-methyl-1,3-thiazol-5-yl)methyl]-5-(morpholine-4-carbonyl)piperidine-3-carboxamide
3-(3-{1-[(5-cyclopropyl-1,2,4-oxadiazol-3-yl)methyl]-1H-pyrazol-3-yl}phenyl)-6-methylpyridazine
5-methyl-3-[5-(4,5,6,7-tetrahydro-2-benzothiophene-1-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-3-yl]-1,2-oxazole
5-fluoro-2-{1-[3-(1H-1,2,3,4-tetrazol-1-yl)-1H-pyrazole-4-carbonyl]pyrrolidin-2-yl}-1H-1,3-benzodiazole
1-(4-benzylpiperidin-1-yl)-3-[1-(pyridine-2-carbonyl)piperidin-4-yl]propan-1-one
1-({1-[2-(4-fluorophenyl)ethyl]piperidin-3-yl}methyl)-3-(4-methoxy-2-methylphenyl)-1-methylurea
(4aR,8aR)-2-cyclopentanecarbonyl-7-(1H-indol-4-ylmethyl)-decahydro-2,7-naphthyridin-4a-ol
methyl 6-({[(5-methylpyrazin-2-yl)methyl]carbamoyl}amino)-1,2,3,4-tetrahydroquinoline-1-carboxylate
3-ethyl-1-(4-ethyl-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-7-yl)-3-(2-methoxyethyl)urea
1-{1-[(2-ethoxyphenyl)methyl]piperidin-3-yl}-N-(3-hydroxypropyl)-1H-1,2,3-triazole-4-carboxamide
2-{2-[3-(furan-2-yl)phenyl]-1H-imidazol-1-yl}ethan-1-ol
4-{[2-(2-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-1λ6-thiomorpholine-1,1-dione
(2R,3R)-3-(1H-imidazol-1-yl)-1'-(pyrazine-2-carbonyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
1-(2-methylpropyl)-4-[3-(pyrazin-2-yl)propanoyl]-6-(pyridin-3-ylmethoxy)-1,4-diazepan-2-one
N-[1-(2,5-dimethoxyphenyl)ethyl]-4-propylpyrimidine-5-carboxamide
4-(5-methylpyridin-2-yl)-1-{[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}piperidin-4-ol
methyl 9-[(4-fluorophenyl)methoxy]-7-oxo-3-(thiophen-2-ylmethyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
2-(5-{5H,6H,7H-[1,3]thiazolo[3,2-a]pyrimidin-3-ylmethyl}-1,2,4-oxadiazol-3-yl)pyridine
4-fluoro-3-hydroxy-N-[1-(pyrazin-2-yl)propan-2-yl]benzamide
7-{2,7-dimethylpyrazolo[1,5-a]pyrimidine-5-carbonyl}-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-3-carboxamide
4-[(diethylamino)methyl]-5-ethyl-N-(prop-2-en-1-yl)-N-(pyridin-3-ylmethyl)furan-2-carboxamide
3-{[4-(2-methoxyphenyl)-3-oxopiperazin-1-yl]methyl}-N-methyl-1,2,4-oxadiazole-5-carboxamide
9-oxo-N-[3-(pyridin-3-yloxy)propyl]-1-azatricyclo[6.3.1.04,12]dodeca-4(12),5,7,10-tetraene-10-carboxamide
N-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-3-(4-methoxyphenyl)-N-methyl-3-phenylpropanamide
1'-(furan-2-ylmethyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
1-(cyclopropylmethyl)-5-[4-(methylsulfanyl)benzoyl]-N-(pyridin-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
2-[5-(2,3-dihydro-1H-inden-1-ylmethyl)-3-(5-methylfuran-2-yl)-1H-1,2,4-triazol-1-yl]ethan-1-ol
(4S)-3-[(2,4-difluorophenyl)methyl]-4-(propan-2-yl)-1,3-oxazolidin-2-one
1,3-dimethyl-N-{[2-(4-methylpiperazin-1-yl)pyridin-3-yl]methyl}-1H-indole-2-carboxamide
{[3-(3-fluorophenyl)-1-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}[2-(pyridin-3-yloxy)ethyl]amine
ethyl 4-[(2-chlorophenyl)methyl]-1-(3-phenoxypropanoyl)piperidine-4-carboxylate
2-{3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-1H-indole
1-{[3-(2-methoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl}-1H-indazole
N-[1-(pyrimidin-4-yl)ethyl]-4-(3,3,3-trifluoropropyl)pyrimidin-2-amine
2-(2-{[2-(pyridin-3-yloxy)propyl]amino}pyrimidin-4-yl)pyridine-4-carboxylic acid
2-[9-(3-fluoro-4-methoxybenzoyl)-3-oxo-2,9-diazaspiro[5.5]undecan-2-yl]acetic acid
4,6-dimethyl-2-[3-(morpholin-4-yl)piperidin-1-yl]pyridine-3-carbonitrile
N-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-5-oxo-1-(pyridin-3-ylmethyl)pyrrolidine-3-carboxamide
5-(2,6-dimethoxyphenyl)-1-(1,4-dioxan-2-ylmethyl)-4-phenyl-1H-imidazole