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9-methoxy-N-methyl-7-oxo-N-(1,3-thiazol-2-ylmethyl)-3-[(2,3,6-trifluorophenyl)methyl]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
2-[1-(2,2-dimethylpropyl)-4-(quinolin-8-ylmethyl)piperazin-2-yl]ethan-1-ol
N-[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl]-2-(pyridin-3-yl)-5,6,7,8-tetrahydroquinazolin-5-amine
1-(1-cyclopropyl-5-oxopyrrolidine-3-carbonyl)-4-(1H-imidazol-1-yl)piperidine-4-carboxylic acid
2-({[(3R,4R)-4-(hydroxymethyl)-1-[4-(trifluoromethyl)pyrimidin-2-yl]pyrrolidin-3-yl]methyl}(methyl)amino)ethan-1-ol
1-[(4-chlorophenyl)methyl]-N-[(3,4,5-trimethoxyphenyl)methyl]-1H-1,2,3-triazole-4-carboxamide
3-{[1-(4-fluorophenyl)cyclopropyl]formamido}-3-(furan-2-yl)propanoic acid
6-methyl-2-({[3-(oxolan-3-yl)propyl]amino}methyl)quinolin-4-ol
2-(azepan-1-yl)-1-{5-cyclopropanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}ethan-1-one
5-{1-[(2E)-3-(4-fluorophenyl)prop-2-enoyl]piperidin-4-yl}-3-(oxolan-2-ylmethyl)-5-(pyridin-2-yl)imidazolidine-2,4-dione
1'-[5-(1H-pyrazol-1-ylmethyl)furan-2-carbonyl]-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
5-{3-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyrazin-2-ol
1-(3,5-dimethylphenyl)-4-[2-(oxan-2-ylmethoxy)acetyl]piperazin-2-one
[(1S,3S,3aS,6aR)-5-methyl-1-phenyl-3-[4-(1H-pyrazol-1-yl)phenyl]-octahydropyrrolo[3,4-c]pyrrol-1-yl]methanol
diethyl({[1-(3-phenylpropyl)piperidin-3-yl]sulfamoyl})amine
1-(2-aminoethyl)-N-[(2-methyl-2,3-dihydro-1-benzofuran-5-yl)methyl]-1H-1,2,3-triazole-4-carboxamide
2-amino-4-[3,5-dimethyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]-6-(3,5-dimethyl-1H-pyrazol-4-yl)pyridine-3-carbonitrile
N-[1-(hydroxymethyl)cyclopentyl]-2-{1-[(2-methylphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
N-cyclopropyl-N-{[7-fluoro-2-(4-methoxyphenyl)quinolin-3-yl]methyl}-3-(3-methyl-1H-pyrazol-1-yl)propanamide
N-[2-(dimethylamino)-2-(thiophen-2-yl)ethyl]-2,3,5,6-tetramethylbenzamide
ethyl 4-(cyclopropylmethyl)-1-(3-phenyl-1H-pyrazole-5-carbonyl)piperidine-4-carboxylate
(2R,3R,6R)-3-(2,3-difluorophenyl)-5-(pyridin-3-ylmethyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
5-methoxy-2-{[3-(2-{[2-(pyrrolidin-1-yl)ethyl]sulfanyl}pyrimidin-4-yl)piperidin-1-yl]methyl}phenol
1-(2-fluorobenzenesulfonyl)-3-{[4-(pyrrolidine-1-carbonyl)-1H-1,2,3-triazol-1-yl]methyl}piperidine
(3aS,6aS)-2-[(3,5-dimethyl-4-oxo-1,4-dihydropyridin-2-yl)methyl]-5-(oxan-4-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-methyl-9-[(1-propyl-1H-pyrazol-4-yl)sulfonyl]-2,9-diazaspiro[5.5]undecan-3-one
4-[(2-fluoro-4,5-dimethoxyphenyl)methyl]-1-methyl-2,3,4,5-tetrahydro-1H-1,4-benzodiazepine-2,5-dione
1-(2-methoxyethyl)-5-(thiomorpholine-4-carbonyl)piperidin-2-one
N-[1-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)benzamide
(2S,4S)-4-(4-{[(tert-butylcarbamoyl)(methyl)amino]methyl}-1H-1,2,3-triazol-1-yl)-N-methylpyrrolidine-2-carboxamide
1-(5-methyl-4,5,6,7-tetrahydro-2H-indazole-3-carbonyl)-4-(pyridin-3-yl)piperidin-4-ol
3-(carbamoylmethoxy)-N-[(2E)-3-phenylprop-2-en-1-yl]-N-propylbenzamide
4-(3-ethyl-4-methylpiperazine-1-carbonyl)-8-methyl-2-(1-methyl-1H-pyrazol-4-yl)quinoline
6-methyl-2-[1-(5-methyl-1-propyl-1H-pyrazole-4-carbonyl)pyrrolidin-2-yl]-1H-1,3-benzodiazole
1-[(1-{[1-(2-fluorophenyl)-1H-pyrazol-4-yl]methyl}piperidin-3-yl)methyl]-1H-1,2,3-triazole-4-carboxylic acid
N-({8-[2-(3-fluorophenyl)acetyl]-1-oxa-8-azaspiro[4.5]decan-2-yl}methyl)pyridine-2-carboxamide
N-[(1-ethyl-1H-indazol-3-yl)methyl]-2-[2-(propan-2-yl)-1H-imidazol-1-yl]propanamide
1-[3-(3-methoxyphenyl)-1H-pyrazole-4-carbonyl]-3-(1H-pyrazol-5-yl)piperidine
N-[1-(2-fluorophenyl)piperidin-4-yl]-2-(1H-imidazol-2-yl)benzamide
1-[2-(furan-2-yl)-2-(pyrrolidin-1-yl)ethyl]-2-(4-methyl-1H-imidazol-5-yl)-1H-imidazole
5-(oxan-4-yl)-3-(thiophen-3-ylmethyl)-1,2,4-oxadiazole
N-{2-[2-(hydroxymethyl)piperidin-1-yl]ethyl}-2-[(2-methylprop-2-en-1-yl)oxy]benzamide
1-(azepan-1-yl)-3-[3-({[(3-chlorophenyl)methyl]amino}methyl)phenoxy]propan-2-ol
[1-({4-[methyl(phenyl)amino]phenyl}methyl)-4-(oxan-2-ylmethyl)piperidin-4-yl]methanol
2-(4-benzyl-3-methyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-1-yl)-N-[2-(pyridin-4-yl)ethyl]acetamide
4-({1-[(2,3,4-trifluorophenyl)methyl]piperidin-2-yl}methyl)morpholine
2-{2-cyano-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl}-N-[2-(4-methoxyphenyl)ethyl]acetamide
(3R)-3,4,4-trimethyl-1-[1-methyl-3-(trifluoromethyl)-1H-pyrazole-5-carbonyl]pyrrolidin-3-ol
1-methyl-4-[2-(2-{[3-(propan-2-yl)piperidin-1-yl]methyl}phenoxy)ethyl]piperazine
3-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]-N-(2-methoxyphenyl)piperidine-1-carboxamide