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N-methyl-2-(2-oxo-1,3-oxazolidin-3-yl)-N-[(1-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidin-4-yl)methyl]acetamide
2-({4-[4-(3,3,3-trifluoropropyl)pyrimidin-2-yl]piperazin-1-yl}methyl)benzonitrile
1-{4-[(4-{[4-methyl-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}piperidin-1-yl)methyl]thiophen-2-yl}ethan-1-one
1-[6-methyl-2-(pyridin-3-yl)pyrimidin-4-yl]-4-(2-methylpropyl)-1,4-diazepane
2-(3-fluorophenoxymethyl)-N-methyl-N-{[1-(propan-2-yl)pyrrolidin-3-yl]methyl}-1,3-oxazole-4-carboxamide
3-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]-N-[2-(3-phenylpyrrolidin-1-yl)ethyl]propanamide
1-(10-methoxy-3,4,5,6-tetrahydro-2H-1,5-benzoxazocin-5-yl)-2-(1-methyl-1H-pyrrol-2-yl)ethane-1,2-dione
N-[(5,6-dimethyl-1H-1,3-benzodiazol-2-yl)methyl]-2-[3-(2-fluorophenyl)-1-(2-methoxyethyl)-2,5-dioxopyrrolidin-3-yl]-N-methylacetamide
N-[(3-cyclohexyl-1,2,4-oxadiazol-5-yl)methyl]-5-fluoro-4-(morpholin-4-yl)pyrimidin-2-amine
3-chloro-N-{[2-(dimethylamino)-5,8-dimethoxyquinolin-3-yl]methyl}-N-[3-(2-oxopyrrolidin-1-yl)propyl]benzamide
2-(1-{[1-(1,3-benzothiazol-2-ylmethyl)piperidin-3-yl]methyl}-1H-1,2,3-triazol-4-yl)ethan-1-ol
(3S,4S)-1-{5-methyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carbonyl}-4-(pyrrolidin-1-yl)pyrrolidin-3-ol
2-(2,5-dioxoimidazolidin-1-yl)-N-[(3R,4S)-4-propyl-1-(pyridin-4-ylmethyl)pyrrolidin-3-yl]acetamide
3-[3,5-dimethyl-1-(propan-2-yl)-1H-pyrazol-4-yl]-1-methyl-1-{[3-(thiophen-2-yl)-1H-pyrazol-5-yl]methyl}urea
{[1-(2,5-dimethylphenyl)-3-phenyl-1H-pyrazol-4-yl]methyl}(methyl)(pyrimidin-4-ylmethyl)amine
methyl({[3-(propan-2-yl)-1,2-oxazol-5-yl]methyl}){[3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}amine
N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-2-hydroxyacetamide
N-{1-[7-(1-benzothiophen-2-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]-2-methylpropyl}-2-methoxyacetamide
3-{[1-(3,4-dihydro-2H-1-benzopyran-3-carbonyl)piperidin-4-yl]oxy}pyridine
N-ethyl-5-methyl-N-(2-methylprop-2-en-1-yl)-4-[(pyridin-2-ylmethyl)amino]thieno[2,3-d]pyrimidine-6-carboxamide
[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]({[3-(3-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl})methylamine
6-(4-methylpiperidin-1-yl)-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}pyridine-3-carboxamide
4-[(4-methoxy-3,5-dimethylpyridin-2-yl)methyl]-3-methyl-1-(2-methylpropyl)piperazin-2-one
N-[(2S)-1-hydroxy-4-(methylsulfanyl)butan-2-yl]-5-[(isoquinolin-5-yloxy)methyl]-1,2-oxazole-3-carboxamide
(3aR,7aS)-5-methyl-2-[4-methyl-2-(propan-2-yl)-1,3-thiazole-5-carbonyl]-2,3,3a,4,7,7a-hexahydro-1H-isoindole
1-cyclohexyl-N-[1-(4-methylphenyl)propyl]-1H-1,2,3-triazole-4-carboxamide
2-[4-(dimethylamino)-6-oxo-1,6-dihydropyridazin-1-yl]-N-(furan-3-ylmethyl)-N-methylacetamide
1-(3-methoxypiperidin-1-yl)-3-[5-(2-phenylethyl)-1,3,4-oxadiazol-2-yl]propan-1-one
N-methyl-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-2,3,4,9-tetrahydro-1H-carbazole-6-carboxamide
(1S,5R)-6-(2,6-dimethylpyrimidine-4-carbonyl)-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
N-[(3S,4R)-1-[(1-methyl-1H-indol-2-yl)methyl]-4-(propan-2-yl)pyrrolidin-3-yl]acetamide
N-({3-[2-(dimethylamino)ethoxy]phenyl}methyl)-N-(pyridin-2-ylmethyl)-1,3-thiazole-5-carboxamide
N-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-N,2,4-trimethylpyrimidine-5-carboxamide
1-({1-butyl-3-[(1-methylpiperidin-4-yl)methyl]-1H-1,2,4-triazol-5-yl}methyl)-5-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
(2S)-1-{[2-(3,4-dimethoxyphenyl)-7-methylquinolin-3-yl]methyl}pyrrolidine-2-carboxamide
2-[2,4-dioxo-1-(2-phenylethyl)-8-{[(4S)-4-(prop-1-en-2-yl)cyclohex-1-en-1-yl]methyl}-1,3,8-triazaspiro[4.5]decan-3-yl]acetamide
2-[2-(pyridin-3-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl]-2,3-dihydro-1H-isoindole
8-[2-(ethylamino)pyrimidine-5-carbonyl]-2-(2-hydroxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
6-butyl-2-{4-[(4-methylpiperazin-1-yl)methyl]phenyl}-3,4-dihydropyrimidin-4-one
methyl 1-(2-methylpropyl)-3-(2-phenylacetamido)-5-(propylamino)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
3-(3-methoxyphenyl)-N-{[3-(2-methylpropyl)-1,2-oxazol-5-yl]methyl}-1H-pyrazole-4-carboxamide
N-({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)-N-(2-methoxyethyl)-4-methyl-1,3-oxazole-5-carboxamide
1-(2-methoxyethyl)-3-[(3-methoxyphenyl)methyl]-8-(2-methylpropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-(2-cyclohexylethyl)-N-[2-(pyridin-4-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
3-(1-{[2-(2-methoxyphenyl)-1,3-thiazol-5-yl]methyl}-1H-1,2,3-triazol-4-yl)benzonitrile
1-cyclopropyl-4-[4-(4-methylphenoxy)piperidine-1-carbonyl]pyrrolidin-2-one
1-[4-(2,4-dioxoimidazolidin-1-yl)benzoyl]-3-propylpiperidine-3-carboxylic acid
N-benzyl-2-[1-cyclopropyl-2,5-dioxo-3-(4-phenylphenyl)pyrrolidin-3-yl]-N-(2-hydroxyethyl)acetamide
8-{[4-(2-fluorophenyl)phenyl]methyl}-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
4-[(4-chlorophenyl)methyl]-9-methoxy-7-(3-methoxyphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine