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3-(4-methanesulfonylphenyl)pyrazolo[1,5-a]pyrimidine
2-{[1-(3-methoxyphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}-4-methyl-1H-imidazole
1-[4-(2-methyl-1H-imidazol-1-yl)phenyl]-N-[(2S)-3-methylbutan-2-yl]piperidin-4-amine
(3aS,6aS)-2-[(4-phenylphenyl)carbamoyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-(2,3-dihydro-1H-inden-5-yl)-5-(methoxymethyl)-3-(oxolan-3-yl)-1H-1,2,4-triazole
N-[(3-tert-butyl-1H-pyrazol-5-yl)methyl]-N-methyl-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
(2R,3R)-1'-(6-aminopyridine-3-carbonyl)-3-(pyrrolidin-1-yl)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
1-benzyl-N-{2-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}piperidine-2-carboxamide
2-(1-methylcyclopropanecarbonyl)-7-{[4-(propan-2-yl)phenyl]methyl}-2,7-diazaspiro[4.5]decane
N-[(5-fluoro-1H-indol-2-yl)methyl]-8-methoxy-3,4-dihydro-2H-1-benzopyran-3-carboxamide
[1-(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)-3-(3-phenylpropyl)piperidin-3-yl]methanol
1-[2-(3-methoxypropyl)piperidin-1-yl]-2-(4-methyl-1H-pyrazol-1-yl)ethan-1-one
3-[(3R,4S)-1-{5-[(methylsulfanyl)methyl]furan-2-carbonyl}-4-(morpholin-4-yl)piperidin-3-yl]propan-1-ol
N-(2H-1,3-benzodioxol-5-ylmethyl)-6-[(1R,5S)-3,8-diazabicyclo[3.2.1]octan-8-ylmethyl]-2-oxo-1,2-dihydropyridine-3-carboxamide
[2,4,6-trimethyl-3-({[2-methyl-1-(1-methyl-1H-imidazol-2-yl)propyl]amino}methyl)phenyl]methyl acetate
1-(1H-imidazol-4-ylmethyl)-3-(4-phenylbenzoyl)piperidine
5-[(1S,5R)-3-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]pyridine-2-carbonitrile
N-cycloheptyl-3-[(3S,4R)-4-(dimethylamino)-1-(pyridin-3-ylmethyl)piperidin-3-yl]propanamide
3-(1-{2-[(4-methyl-1,3-thiazol-2-yl)sulfanyl]acetyl}piperidin-4-yl)-1-(morpholin-4-yl)propan-1-one
1-(furan-2-ylmethyl)-N-[2-(6-hydroxy-2-methylpyrimidin-4-yl)ethyl]piperidine-3-carboxamide
5-(3-cyclopropyl-1,2,4-oxadiazol-5-yl)-N-[3-(1H-pyrazol-1-yl)propyl]pyridin-2-amine
3-{4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperazine-1-carbonyl}-2,8-diazaspiro[4.5]decane
4-phenyl-1-[(2R)-pyrrolidin-2-ylmethyl]-5-(2,4,5-trifluorophenyl)-1H-imidazole
5-[2-(3-chlorophenyl)ethyl]-3-(oxolan-3-yl)-1,2,4-oxadiazole
3-[3-fluoro-5-(propan-2-yloxy)phenyl]-N,N,1-trimethyl-1H-1,2,4-triazol-5-amine
N-{[2-(morpholin-4-yl)-1,3-thiazol-4-yl]methyl}pyrazolo[1,5-a]pyridine-7-carboxamide
2-(2-methyl-1,3-thiazol-4-yl)-1-[2-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidin-1-yl]ethan-1-one
2-ethyl-9-(5-ethyl-1,3,4-thiadiazol-2-yl)-4-phenyl-2,9-diazaspiro[5.5]undecan-3-one
2-{1-[(2,3,4-trimethoxyphenyl)methyl]-1,4-diazepan-6-yl}acetic acid
(4aR,7aS)-1-acetyl-4-[(2-methoxy-4-methylphenyl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-(2-{2-amino-4H,5H,6H,7H-[1,3]thiazolo[5,4-c]pyridin-5-yl}pyrimidin-4-yl)pyridine-4-carboxylic acid
N-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]-N,5-dimethyl-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide
methyl 4-{[(1-methylpiperidin-2-yl)formamido]methyl}benzoate
(1R,3S)-N3-ethyl-1,2,2-trimethyl-N1-[3-(morpholin-4-yl)propyl]cyclopentane-1,3-dicarboxamide
(4aS,7aR)-1-ethyl-4-[(4-methyl-1H-imidazol-5-yl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-ethyl-8-[1-(methylsulfanyl)propan-2-yl]-3-[3-(pyridin-3-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
methyl 4-{5-[(4-phenyl-1,4-diazepan-1-yl)methyl]-1,2,4-oxadiazol-3-yl}benzoate
methyl 2-({2-[(1-acetylpiperidin-4-yl)oxy]-5-chlorophenyl}formamido)-4-(methylsulfanyl)butanoate
methyl 4-({4-[2,5-dioxo-1-(oxolan-2-ylmethyl)-4-(pyridin-2-yl)imidazolidin-4-yl]piperidin-1-yl}methyl)benzoate
4-(2-ethoxyacetyl)-5-methyl-1-(3-methylphenyl)piperazin-2-one
(3R,4S)-4-cyclopropyl-1-(4-phenylbenzenesulfonyl)pyrrolidin-3-amine
2-({[(1,3-dimethylpyrrolidin-3-yl)methyl](methyl)amino}methyl)-3,5-dimethoxybenzoic acid
2-(2-methoxyethyl)-1-(3-phenyl-1H-pyrazole-4-carbonyl)piperidine
N-[(5-methylfuran-2-yl)methyl]-2-[1-(3-methylphenyl)-5-oxo-3-propyl-4,5-dihydro-1H-1,2,4-triazol-4-yl]acetamide
1-[2-(2-chlorophenyl)-3-methyl-3H-imidazo[4,5-b]pyridine-6-carbonyl]-4-ethoxypiperidine
1-{4-[(3S,4S)-4-(4-fluorophenyl)-3-hydroxypiperidine-1-carbonyl]phenyl}pyrrolidin-2-one
(1R,5R)-6-[(3-cyanophenyl)methyl]-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-sulfonamide
(2S,4S)-N-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-1-[(3-chlorophenyl)methyl]-4-{[(2,5-difluorophenyl)methyl]amino}pyrrolidine-2-carboxamide
(1R,3S)-3-(2-hydroxyethoxy)-7-{[5-(2-methylpropyl)thiophen-2-yl]methyl}-7-azaspiro[3.5]nonan-1-ol
5-[1-(2H-1,3-benzodioxol-5-ylmethyl)piperidin-4-yl]-5-ethyl-3-(2-methylprop-2-en-1-yl)imidazolidine-2,4-dione