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3-({4-[(4-fluorophenyl)methyl]piperidin-1-yl}methyl)pyridine
1-{1-[(5-cyclopentylthiophen-2-yl)methyl]piperidin-4-yl}-N-cyclopropylpiperidine-4-carboxamide
5-[2-(5-methyl-1,2-oxazol-3-yl)pyrrolidine-1-carbonyl]-2-(phenoxymethyl)pyrimidin-4-ol
dimethyl[(5-{[(1S,5R)-3-[(4-methyl-1H-imidazol-5-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}thiophen-3-yl)methyl]amine
1-(3-cyanophenyl)-3-(1,4-dioxan-2-ylmethyl)urea
6-[(1E)-pent-1-en-1-yl]-N-(propan-2-yl)pyrimidin-4-amine
1-(2-methyl-1,2,3,4-tetrahydroisoquinoline-3-carbonyl)-4-(5-methylpyridin-2-yl)piperidin-4-ol
3-{2-oxo-2-[2-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-4-yl]ethyl}-3,4-dihydroquinazolin-4-one
N-({6-ethyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyridine-3-carboxamide
(2S)-2-{[6-(2,5-dimethylphenyl)imidazo[2,1-b][1,3]thiazol-3-yl]formamido}-4-methylpentanamide
1-(3-hydroxypiperidin-1-yl)-4-[5-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]butan-1-one
[(4-methoxy-3-methylphenyl)methyl][2-(4-methoxyphenyl)ethyl][(1-methylpiperidin-4-yl)methyl]amine
1-[4-(2-fluorophenyl)piperazin-1-yl]-2-{5-[(4-methylpiperidin-1-yl)methyl]-1H-1,2,3,4-tetrazol-1-yl}ethan-1-one
2-{4-[2-(4-acetyl-3,5-dimethyl-1H-pyrazol-1-yl)acetyl]-2-oxopiperazin-1-yl}benzonitrile
N-{5H,6H,7H-cyclopenta[d]pyrimidin-2-ylmethyl}-2-(phenylamino)pyrimidine-5-carboxamide
9-[5-(hydroxymethyl)furan-2-carbonyl]-2-(2-hydroxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
1-[4-(1-{[4-(hydroxymethyl)phenyl]methyl}-1H-1,2,3-triazol-4-yl)thiophen-2-yl]ethan-1-one
5-[(5-cyclopentylthiophen-2-yl)methyl]-N,N-dimethyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
8-chloro-N-[2-(methylsulfanyl)ethyl]quinoline-2-carboxamide
2-(5-cyclopropyl-1,3-oxazole-4-carbonyl)-6,7-dimethoxy-1,2,3,4-tetrahydroisoquinoline
N-[(2R,3R)-1'-[2-(3-methyl-1H-pyrazol-1-yl)acetyl]-2-(pyridin-3-ylmethoxy)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]propanamide
dimethyl({[4-methyl-5-(1-{[1-(3-methylphenyl)-1H-pyrazol-4-yl]methyl}piperidin-4-yl)-4H-1,2,4-triazol-3-yl]methyl})amine
N-({5-cyclohexyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)-4,6-dimethylpyridine-3-carboxamide
1-(4-methoxyphenyl)-N-methyl-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}cyclopropane-1-carboxamide
(3S,9aR)-8-(3-methylbutyl)-3-(propan-2-yl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-[3-(methylsulfanyl)propyl]-2,3,4,5-tetrahydro-1-benzoxepine-4-carboxamide
(3S,4R)-1-{5-[(diethylamino)methyl]-2-methylfuran-3-carbonyl}-N,N-dimethyl-4-propylpyrrolidin-3-amine
ethyl 4-[3-(5-fluoro-2-methoxybenzoyl)piperidin-1-yl]piperidine-1-carboxylate
[(3R,4R)-1-(2,5-dimethylfuran-3-carbonyl)-4-{[(2-methoxyethyl)(methyl)amino]methyl}pyrrolidin-3-yl]methanol
ethyl 2-[4-(6-methoxy-1-methyl-1H-indole-2-carbonyl)morpholin-3-yl]acetate
1-(1-{6-[(2,2-dimethylpropyl)amino]pyridine-3-carbonyl}piperidin-3-yl)-3-methylbutan-1-one
N-{2-[(8-methoxy-2-oxo-1,2,3,4-tetrahydroquinolin-4-yl)formamido]ethyl}pyridine-3-carboxamide
2-(4-fluorophenyl)-N-(2-{7-[(5-methylthiophen-2-yl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)acetamide
methyl 5-{2-methyl-3-oxo-4-phenyl-2,9-diazaspiro[5.5]undecan-9-yl}pentanoate
(4aR,7aS)-1-(cyclopropylmethyl)-4-[3-(4,5-dimethyl-1H-pyrazol-3-yl)propanoyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-methyl-9-(prop-2-en-1-yl)-4-[2-(1H-1,2,3-triazol-1-yl)acetyl]-1,4,9-triazaspiro[5.6]dodecan-10-one
3-[(4-fluorophenyl)methyl]-5-methyl-5-{1-[3-(3-methyl-1H-pyrazol-1-yl)propanoyl]piperidin-4-yl}imidazolidine-2,4-dione
N-[(3-ethyl-1,2-oxazol-5-yl)methyl]-N-methyl-5-phenyl-1H-pyrazole-3-carboxamide
1-[(4-methoxy-2,3-dimethylphenyl)methyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
9-[(dimethyl-1H-1,2,4-triazol-5-yl)methyl]-1-oxa-9-azaspiro[5.5]undecan-5-ol
5-(2,5-dimethylphenoxymethyl)-N-ethyl-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-1,2-oxazole-3-carboxamide
3-{[3-oxo-2-(prop-2-en-1-yl)-2,9-diazaspiro[5.5]undecan-9-yl]methyl}benzonitrile
4-benzyl-3-ethyl-1-(5-ethyl-2-methylpyrimidin-4-yl)-1,4-diazepan-5-one
N-(4-chloro-3-methoxyphenyl)-2-[4-(pyrimidin-2-yl)-1,4-diazepan-1-yl]acetamide
4-[(3-fluorophenyl)methyl]-3-{2-oxo-2-[4-(pyridin-3-ylmethyl)piperazin-1-yl]ethyl}piperazin-2-one
[(5-tert-butyl-1H-pyrazol-3-yl)methyl][(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl](2-methoxyethyl)amine
2-{4-[(4-methylpiperazin-1-yl)methyl]phenyl}-6-(pyridin-3-yl)-3,4-dihydropyrimidin-4-one
methyl 2-[2,4-dioxo-1-(2-phenylethyl)-8-(thiolan-3-yl)-1,3,8-triazaspiro[4.5]decan-3-yl]acetate
2-(4-benzyl-2-oxopyrrolidin-1-yl)-N-methyl-N-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}acetamide
5-methyl-1-propyl-N-[2-(thiophen-2-yl)ethyl]-1H-pyrazole-4-carboxamide