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2-butyl-8-[3-(2-methyl-1H-imidazol-1-yl)propanoyl]-2,8-diazaspiro[5.5]undecan-3-one
N-(2-ethoxyphenyl)-8-methyl-6,9-dioxo-octahydro-1H-pyrazino[1,2-a]piperazine-2-carboxamide
4-methoxy-N-(2-{7-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)benzamide
2-methoxy-1-[4-(6-methoxy-3-methyl-1-benzofuran-2-carbonyl)-1,4-diazepan-1-yl]ethan-1-one
(1S,5R)-N-(2,3-dimethylphenyl)-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane-6-carboxamide
N-(3-{[2-(trifluoromethyl)morpholin-4-yl]sulfonyl}phenyl)acetamide
[7-(6-methylpyridin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methanamine
(1-methyl-5-{2-methyl-2,8-diazaspiro[4.5]decane-3-carbonyl}-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-3-yl)methanol
2-[4-(quinolin-3-yl)-1H-pyrazol-1-yl]propanamide
N-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}-N-(pyridin-4-ylmethyl)cyclobutanamine
2-(1-{5-ethyl-6-methylthieno[2,3-d]pyrimidin-4-yl}azetidin-3-yl)pyridine
N-[3-(dimethylamino)propyl]-N-methylpiperidin-3-amine
6-(4-methoxy-2,3-dimethylphenyl)-1,3,8-triazatricyclo[7.4.0.02,7]trideca-2(7),8-dien-4-one
2-(1-{[2-(ethanesulfonyl)-1-(2-phenylethyl)-1H-imidazol-5-yl]methyl}piperidin-2-yl)ethan-1-ol
1-[(3R,4R)-4-hydroxy-4-(2-methoxyethyl)-3-methylpiperidin-1-yl]-3-(1-methyl-1H-pyrazol-4-yl)propan-1-one
5-[4-(propan-2-yloxy)phenyl]pyrimidin-2-amine
2-(2-{[1-(3-methylphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}-1H-pyrrol-1-yl)pyrimidine
N-methyl-N-{[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]methyl}-1-benzothiophene-2-carboxamide
(1S,5R)-6-{[4-(methylsulfanyl)phenyl]methyl}-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
N-[(2-chloropyridin-3-yl)methyl]-6-methoxy-N,3-dimethyl-1-benzofuran-2-carboxamide
[(2S,4R)-1-(2-chloro-4-fluorobenzenesulfonyl)-4-(dimethylamino)pyrrolidin-2-yl]methanol
ethyl 3-(2-methoxyethyl)-1-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)piperidine-3-carboxylate
5-{[(1R,5R)-3-(dimethylsulfamoyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}-N,N-dimethylfuran-2-carboxamide
1-[2-(2,6,6-trimethyl-4-oxo-1-propyl-4,5,6,7-tetrahydro-1H-indol-3-yl)acetyl]piperidine-3-carboxamide
2-{3-[2-(2-fluorophenyl)ethyl]piperidin-1-yl}propane-1,3-diol
(1R,2S,6R,7S)-4-[2-(pyridin-2-yl)pyrimidine-5-carbonyl]-4-azatricyclo[5.2.2.02,6]undecane
4-(cyclohexylmethyl)-3-(1-methyl-1H-pyrazol-3-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
1-cyclopentyl-N-[2-(2-fluorophenyl)ethyl]-6-oxopiperidine-3-carboxamide
1-phenyl-N-{[1-(pyridin-3-ylmethyl)piperidin-3-yl]methyl}methanesulfonamide
2-methyl-N-{1-[5-(trifluoromethyl)pyridin-2-yl]piperidin-3-yl}-1-benzofuran-7-carboxamide
1-(cyclopropylmethyl)-4'-(2,2-dimethylpropyl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
2-(3-{5-hydroxy-1-oxa-9-azaspiro[5.5]undecan-9-yl}-3-oxopropyl)-2,3-dihydro-1H-isoindol-1-one
(3R,5S)-N3-(2,3-dihydro-1H-inden-5-yl)-N5-[(3-fluorophenyl)methyl]-1-(pyridin-4-ylmethyl)piperidine-3,5-dicarboxamide
(3aR,6aS)-5-{[2-(2-hydroxyethoxy)phenyl]methyl}-1-oxo-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-{3-[4-(4-methylphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}pyrimidine
2-[(1R,5R)-6-(cyclopropylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
5-{7-cyclopentyl-6-oxo-2,7-diazaspiro[4.5]decane-2-carbonyl}-1-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
8-[(2S)-2-(methylamino)propanoyl]-2-[(2E)-3-phenylprop-2-en-1-yl]-2,8-diazaspiro[4.5]decan-3-one
2-(2-{[4-(4-methylphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}-1H-pyrrol-1-yl)pyrimidine
N-(2-{1-[3-(1H-pyrrol-1-yl)propyl]-1,2,5,6-tetrahydropyridin-3-yl}ethyl)furan-2-carboxamide
N-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-N-methyl-3-(2-methyl-1H-indol-1-yl)propanamide
1-[(3-methoxyphenyl)methyl]-N-methyl-6-oxo-N-(2-phenylethyl)piperidine-3-carboxamide
N-[(2,4-dimethoxyphenyl)methyl]-3-[1-(pyridin-4-ylmethyl)piperidin-3-yl]propanamide
{1-[4-methyl-2-(pyridin-4-yl)pyrimidin-5-yl]ethyl}[(2,4,5-trimethylphenyl)methyl]amine
1-[1-(2-chlorophenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]-3-(thiophen-2-yl)propan-1-one
1-[(4-fluorophenyl)methyl]-3-hydroxy-3-({[(5-methylfuran-2-yl)methyl]amino}methyl)piperidin-2-one
(3aR,7aS)-N-(4-methanesulfonylphenyl)-2,3,3a,4,7,7a-hexahydro-1H-isoindole-2-carboxamide
4-{[1-(dimethylsulfamoyl)piperidin-4-yl]oxy}-N,N-bis(prop-2-en-1-yl)benzamide
3-(4-acetylphenyl)-1-(1-methylpiperidin-4-yl)-1-(pyridin-4-ylmethyl)urea
5-(2-methoxyphenoxymethyl)-N-methyl-N-[1-(thiophen-2-yl)ethyl]-1,2-oxazole-3-carboxamide