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4-(2,5-dimethoxyphenyl)thieno[2,3-d]pyrimidine
3-(2-chloro-4-fluorophenyl)-4-methyl-1,2-dihydroquinolin-2-one
2-hydroxy-1-[3-(4-methoxyphenoxymethyl)piperidin-1-yl]ethan-1-one
1-[(3R,4R)-4-hydroxy-3-methyl-4-(oxan-4-yl)piperidin-1-yl]-2-{8-methylimidazo[1,2-a]pyridin-3-yl}ethan-1-one
1-[5-(5-ethyl-1,3,4-oxadiazol-2-yl)-2-methoxyphenyl]-3-{[5-(methoxymethyl)-1,2,4-oxadiazol-3-yl]methyl}urea
1-{[1-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}-2-(5-methyl-1,2-oxazol-3-yl)piperidine
4-[4-(oxan-4-yl)piperazine-1-carbonyl]-1-(pyridin-4-ylmethyl)pyrrolidin-2-one
2-[4-(4-methoxyphenyl)-4H-1,2,4-triazol-3-yl]ethan-1-amine
3-[(2-oxopyrrolidin-1-yl)methyl]-N-(3-phenyl-1,2,4-thiadiazol-5-yl)piperidine-1-carboxamide
6-{1-[(2,2-dimethyl-2,3-dihydro-1-benzofuran-5-yl)methyl]piperidin-3-yl}-2-methylpyrimidin-4-ol
2-(1H-1,3-benzodiazol-1-yl)-N-[1-(5-methyl-1-phenyl-1H-pyrazol-4-yl)ethyl]acetamide
2-({2-[2-(1H-pyrazol-1-yl)ethyl]piperidin-1-yl}methyl)benzoic acid
1-(dimethylsulfamoyl)-4-(2-fluorophenoxy)piperidine-4-carboxylic acid
3-methoxy-N-[1-(7-{[4-(pyrrolidin-1-yl)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)ethyl]propanamide
2-butyl-8-(1-ethyl-1H-pyrazole-5-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
5-[4-(piperidine-1-sulfonyl)phenyl]-2-(4H-1,2,4-triazol-4-yl)pyridine
3-(3-benzyl-1-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-N-butyl-N-methylpropanamide
N-{2-[4-(4-fluorophenyl)-5-{[(2-methylphenyl)methyl]sulfanyl}-4H-1,2,4-triazol-3-yl]ethyl}-3-(2-methoxyphenyl)propanamide
7-(4-fluoro-2-methylbenzoyl)-2-(pyridin-4-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
N-(2-phenoxyethyl)-1-(propan-2-yl)piperidine-4-carboxamide
3-[1-({3-[4-(trifluoromethyl)phenyl]-1,2,4-oxadiazol-5-yl}methyl)piperidine-3-carbonyl]pyridine
N-methyl-N-[2-(pyridin-2-yl)ethyl]-2-(1H-1,2,4-triazol-5-yl)benzamide
S-(2-cyclohexanecarbonyl-1,2,3,4-tetrahydroisoquinolin-7-yl)-3-hydroxybutane-1-sulfonamido
4-{1-[3-(5-methylfuran-2-yl)butyl]piperidin-3-yl}-2-{[2-(pyrrolidin-1-yl)ethyl]sulfanyl}pyrimidine
1-{1-[4-(1-methyl-1H-pyrazol-4-yl)pyrimidin-2-yl]piperidin-4-yl}-2-phenylethan-1-ol
N-(2-{1-[(4-methoxy-3,5-dimethylpyridin-2-yl)methyl]piperidin-2-yl}ethyl)acetamide
5,6-dimethyl-N-[1-(5-methyl-1H-1,3-benzodiazol-2-yl)ethyl]-2-oxo-1,2-dihydropyridine-3-carboxamide
5-(furan-2-ylmethyl)-3-(3-methoxyphenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine
2-{methyl[(3-methyl-1,2-oxazol-5-yl)methyl]amino}-2-[3-(trifluoromethyl)phenyl]acetic acid
5-{5-amino-4-cyano-1,6-diazatricyclo[6.2.2.02,7]dodeca-2,4,6-trien-3-yl}-2-hydroxybenzoic acid
5-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-N,N-dimethylpyridin-2-amine
6-(2H-1,3-benzodioxol-5-yl)-N-[3-(dimethyl-1,2-oxazol-4-yl)propyl]pyridine-3-carboxamide
3-{4-[(4-fluorophenyl)methyl]-5-oxo-3-(propan-2-yl)-1,4-diazepan-1-yl}-N,N-dimethylpropanamide
5-(2H-1,3-benzodioxole-5-carbonyl)-3-(1-phenoxyethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
3-(1-cyclopentyl-1H-pyrazol-5-yl)-1-[2-(5-methylfuran-2-yl)ethyl]urea
2-methyl-5-(4-{[5-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}piperazin-1-yl)-2,3-dihydropyridazin-3-one
(3S,4R)-1-cyclopentanecarbonyl-4-(3-methoxyphenyl)pyrrolidine-3-carboxylic acid
N-(3,4-dimethoxyphenyl)-1-(1-methylcyclohexanecarbonyl)piperidin-3-amine
N-cyclopropyl-N-{[1-(2,3-dihydroxypropyl)-1,2,5,6-tetrahydropyridin-3-yl]methyl}cyclobutanecarboxamide
1-ethyl-5-(3-{imidazo[1,2-a]pyridin-2-yl}-1,2,4-oxadiazol-5-yl)piperidin-2-one
N-(2-methoxyethyl)-3-(1-{[4-(methylsulfanyl)phenyl]methyl}piperidin-4-yl)propanamide
1-(4-{[(1H-1,3-benzodiazol-2-ylmethyl)(methyl)amino]methyl}-2-methoxyphenoxy)-3-[methyl(propan-2-yl)amino]propan-2-ol
(3R,5S)-5-[(2,3-dihydro-1H-inden-5-yloxy)methyl]-N-[2-(2-oxoimidazolidin-1-yl)ethyl]piperidine-3-carboxamide
N-[(3S,4R)-1-[(2-cyanophenyl)methyl]-4-(4-methylphenyl)pyrrolidin-3-yl]cyclopropanecarboxamide
7-[3-(2-oxooxolan-3-yl)propanoyl]-2-phenyl-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
N-[2-(2-fluorophenyl)-1-[1-(pyridin-2-ylmethyl)piperidin-4-yl]ethyl]-N-methylthiophene-2-carboxamide
6-tert-butyl-N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-2-oxo-2,3-dihydropyrimidine-4-carboxamide
1-(2-{2-methyl-4-phenyl-2,9-diazaspiro[5.5]undecan-9-yl}-2-oxoethyl)piperidin-2-one
3-hexyl-8-(4-hydroxy-3-methylbenzoyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-(1-{7-[(2E)-3-phenylprop-2-en-1-yl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)cyclopropanecarboxamide