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2-methyl-8-(5,6,7,8-tetrahydroquinoline-3-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
1-(5-ethyl-1,2,4-oxadiazol-3-yl)-4-(2-methoxyphenoxy)piperidine
2-{4-[3-(2-phenylpropyl)-1,2-oxazole-5-carbonyl]piperazin-1-yl}pyrazine
2-({4-[2-(dimethyl-1,3-thiazol-5-yl)acetyl]-2-oxo-1-(2-phenylethyl)-1,4-diazepan-6-yl}oxy)-N,N-diethylacetamide
2-cyclopentyl-N-{[(2S,4S)-1-{3,6-dimethyl-[1,2]oxazolo[5,4-b]pyridine-4-carbonyl}-4-fluoropyrrolidin-2-yl]methyl}acetamide
3-(4-chloro-2,6-dimethylphenyl)-1-[3-(3-oxopiperazin-1-yl)propyl]urea
7-(2-cyclohexylethyl)-2-(pyridin-4-ylmethyl)-2,7-diazaspiro[4.5]decan-6-one
(2S,4R)-4-amino-1-[2-(5-amino-1H-1,2,3,4-tetrazol-1-yl)acetyl]-N,N-diethylpyrrolidine-2-carboxamide
5-ethyl-1'-[(1-ethyl-1H-indol-5-yl)methyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
2-(3-methoxyphenyl)-N-{[3-(pyrrolidin-1-yl)phenyl]methyl}acetamide
6-[4-(4-methoxyphenyl)-4-oxobutanoyl]-N-[4-(methylsulfanyl)phenyl]-6-azaspiro[2.5]octane-1-carboxamide
N-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]methyl}-3-methyl-N-(oxolan-2-ylmethyl)thiophene-2-carboxamide
5-[(2-fluorophenyl)methyl]-3-phenyl-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine
5-ethyl-5-{1-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]piperidin-4-yl}-3-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]imidazolidine-2,4-dione
5-methyl-1-{2-[3-(3-methylphenyl)piperidin-1-yl]-2-oxoethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-(2,3-dihydro-1H-inden-2-yl)-3-(4-hydroxyphenyl)-1H-pyrazole-5-carboxamide
1-(2-methoxyethyl)-N-({6-methylimidazo[1,2-a]pyridin-2-yl}methyl)-6-oxopiperidine-3-carboxamide
4-(1-methyl-2-oxo-1,2-dihydroquinoline-4-carbonyl)piperazine-2-carboxylic acid
6-fluoro-2-oxo-N-(pyrimidin-4-ylmethyl)-1,2-dihydroquinoline-4-carboxamide
5-(2-fluorophenyl)-N-[(1R,2S)-2-phenylcyclopropyl]-1,2,4-triazin-3-amine
methyl 6-{[(2-methoxy-2-oxoethyl)(methyl)amino]methyl}-3-(2-methylbutanamido)thieno[2,3-b]pyridine-2-carboxylate
[(1S,9aR)-octahydro-1H-quinolizin-1-ylmethyl](methyl){[2-(1H-pyrazol-1-yl)phenyl]methyl}amine
2-[3-(4-ethoxyphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-4-methoxypyrimidine
N-cyclopropyl-2-(dimethylamino)-2-(2-methylphenyl)-N-[(trimethyl-1H-pyrazol-4-yl)methyl]acetamide
5-{[4-(3-methylphenoxy)piperidin-1-yl]methyl}-2-propylpyrimidine
N,N-diethyl-1-{1-[(2-hydroxy-3-methoxyphenyl)methyl]piperidin-4-yl}-1H-1,2,3-triazole-4-carboxamide
3,3-dimethyl-1-{[5-(naphthalen-2-ylmethyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}urea
1-{[2-(4-chlorophenyl)-7-(methylsulfanyl)quinolin-3-yl]methyl}piperidin-4-ol
1-methyl-6-(propan-2-yl)-N-[3-(pyridin-4-yl)propyl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
2-[2-(2-methyl-1H-imidazol-1-yl)ethyl]-1-{[3-(3,4,5-trimethoxyphenyl)-1H-pyrazol-4-yl]methyl}piperidine
2-{[2-(dimethylamino)ethyl](thiophen-3-ylmethyl)amino}-2-(2-methoxy-5-methylphenyl)acetic acid
8-[(1-ethyl-1H-indol-6-yl)methyl]-2-(2-hydroxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
2-[1-(5-chloro-3-phenyl-1H-indole-2-carbonyl)pyrrolidin-2-yl]ethan-1-ol
5-chloro-N-({1-[2-(3-fluorophenyl)ethyl]piperidin-4-yl}methyl)-N-methylpyridine-3-carboxamide
methyl (2S,3S)-2-{[5-(2-fluorophenyl)-1,2,4-triazin-3-yl]amino}-3-methylpentanoate
N-(2,4-dimethoxyphenyl)-3-[1-(1H-imidazole-4-carbonyl)piperidin-4-yl]propanamide
1-[(1-cyclopropanecarbonylpiperidin-4-yl)methyl]-3-[5-(thiophen-2-yl)-1,3,4-thiadiazol-2-yl]urea
3-{2-[5-(morpholine-4-carbonyl)thiophen-2-yl]pyrrolidine-1-carbonyl}benzonitrile
2-(dimethyl-1,2-oxazol-4-yl)-N-[(4-hydroxyazepan-4-yl)methyl]acetamide
{[3-(2,5-dimethylthiophen-3-yl)-1-(2-fluorophenyl)-1H-pyrazol-4-yl]methyl}(methyl)[(1-methyl-1H-pyrazol-4-yl)methyl]amine
5-tert-butyl-4-{[(1R,5R)-3-methanesulfonyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}furan-2-carboxamide
3-[5-(3-methyl-1H-pyrazol-4-yl)-1,2,4-oxadiazol-3-yl]-2-phenoxypyridine
(2S,3R)-2-[(5-{[benzyl(methyl)amino]methyl}-1,2-oxazol-3-yl)formamido]-3-hydroxybutanamide
N-{2-[3-(ethylsulfanyl)-5-oxo-4,5-dihydro-1,2,4-triazin-6-yl]phenyl}-2-(pyridin-3-yloxy)acetamide
N-{2-[5-methyl-3-(trifluoromethyl)-1H-pyrazol-1-yl]ethyl}-2,3,4,5-tetrahydro-1-benzoxepine-4-carboxamide
4-[4-(3-fluorophenyl)-1H-pyrazol-5-yl]-1-(thiophen-2-ylmethyl)piperidine
2-[3-(6-hydroxy-2-methylpyrimidin-4-yl)piperidin-1-yl]-N,N-bis(prop-2-en-1-yl)acetamide
4-methoxy-N-({1-[3-(2-methyl-1H-imidazol-1-yl)propanoyl]piperidin-3-yl}methyl)benzene-1-sulfonamide
2-{1-benzyl-4-[(5-methylthiophen-2-yl)methyl]piperazin-2-yl}ethan-1-ol
(4S)-4-phenyl-3-{[1-(propan-2-yl)-1H-imidazol-2-yl]methyl}-1,3-oxazolidin-2-one