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(2-methoxyethyl)({[1-(2-methoxyethyl)-1H-imidazol-2-yl]methyl})[(3-methylthiophen-2-yl)methyl]amine
N-{4-[2-(2-methyl-5-oxo-1,4-diazepan-1-yl)-2-oxoethoxy]phenyl}propanamide
4-{2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidine-1-carbonyl}morpholine
3-hexyl-8-(pyrazine-2-carbonyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
(2S,4R)-N-(1,3-dihydro-2-benzofuran-5-yl)-1-[(2E)-3-phenylprop-2-en-1-yl]-4-(1H-1,2,3,4-tetrazol-1-yl)pyrrolidine-2-carboxamide
5-ethyl-5-{1-[2-(2-methoxyphenoxy)acetyl]piperidin-4-yl}-3-(pyridin-2-ylmethyl)imidazolidine-2,4-dione
N-ethyl-N-(oxan-4-yl)-2-[(quinolin-8-yloxy)methyl]-1,3-oxazole-4-carboxamide
5-[(dimethylamino)methyl]-N-methyl-N-[2-(pyridin-2-yl)ethyl]-1,3,4-oxadiazole-2-carboxamide
ethyl 3-({4-[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]piperidine-1-carbonyl}amino)propanoate
4-methoxy-4-(prop-2-en-1-yl)-N-[2-(trifluoromethoxy)phenyl]piperidine-1-carboxamide
N-(2,1,3-benzoxadiazol-5-ylmethyl)-N-methyl-2-(morpholin-4-yl)pyrimidine-5-carboxamide
6-(aminomethyl)-2-methyl-N-{[2-(2-methyl-1H-imidazol-1-yl)phenyl]methyl}pyrimidin-4-amine
N-methyl-N-[2-(methylsulfanyl)ethyl]-3-{[(1r,4r)-4-hydroxycyclohexyl]sulfamoyl}benzamide
2-(1-methylpyrrolidin-3-yl)-3-oxo-N-phenyl-2,9-diazaspiro[5.5]undecane-9-carboxamide
N-[(2,3-dimethoxyphenyl)methyl]-5-ethylpyrazolo[1,5-a]pyrimidin-7-amine
N-(2-{7-[3-(3-methylphenyl)benzoyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)cyclohexanecarboxamide
N-methyl-N-[1-(4-methylpyridin-2-yl)propan-2-yl]cyclohexanecarboxamide
2-ethyl-7-[(4-hydroxy-1,2,3,4-tetrahydroisoquinolin-2-yl)methyl]-5H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-5-one
3-(4-{[3-(piperidin-1-yl)azetidin-1-yl]methyl}-1H-pyrazol-1-yl)propanoic acid
N-[4-(4-benzyl-3-ethyl-5-oxo-1,4-diazepan-1-yl)-4-oxobutyl]acetamide
7-methyl-2-[3-(4-oxo-3,4-dihydroquinazolin-3-yl)propanoyl]-2,7-diazaspiro[4.5]decan-6-one
1-[3-({[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]amino}methyl)-5,6,7-trimethoxyquinolin-2-yl]piperidin-3-ol
(3S,4R)-4-(2,3-dimethoxyphenyl)-1-(3-fluoropyridin-4-yl)pyrrolidine-3-carboxylic acid
3,3-dimethyl-4-({3-[4-(trifluoromethyl)phenyl]-1,2,4-oxadiazol-5-yl}methyl)piperazin-2-one
N-methyl-N-{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}pyridine-3-carboxamide
8-{4-[1-(pyrrolidin-1-yl)ethyl]phenyl}quinolin-4-amine
2-methyl-8-{[4-(1H-1,2,4-triazol-1-yl)phenyl]methyl}-2,8-diazaspiro[4.5]decane
7-(2-hydroxyethyl)-2-{[3-(trifluoromethyl)phenyl]methyl}-2,7-diazaspiro[4.5]decan-6-one
N-methyl-N-[(3-methylpyridin-4-yl)methyl]-2-(phenylamino)pyrimidine-5-carboxamide
(2R,3R)-3-(pyrrolidin-1-yl)-1'-(thiophen-2-ylmethyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
1-{1-[1-(pyridin-4-ylmethyl)piperidin-4-yl]piperidine-3-carbonyl}-1,4-diazepane
N-methyl-2-(2-oxopyrrolidin-1-yl)-N-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]acetamide
3-benzoyl-1-(1-methyl-1H-pyrrole-2-carbonyl)piperidine
N-[(dimethyl-1,2-oxazol-4-yl)methyl]-2-oxo-1,2,5,6,7,8-hexahydroquinoline-3-carboxamide
5-[2-(2-phenyl-1H-imidazol-1-yl)acetyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carbonitrile
3-cyclopentyl-5-[(4-fluorophenyl)methyl]-5-{1-[(2E)-3-(furan-2-yl)-2-methylprop-2-en-1-yl]piperidin-4-yl}imidazolidine-2,4-dione
3-{[1-(2-methylfuran-3-carbonyl)piperidin-4-yl]oxy}-N-(pyridin-2-ylmethyl)benzamide
9-[4-(trifluoromethyl)pyrimidin-2-yl]-1-oxa-9-azaspiro[5.5]undecan-5-ol
N-phenyl-5-[3-(1H-pyrazol-3-yl)phenyl]furan-2-carboxamide
5-(4-methyl-5-phenylthiophene-2-carbonyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-6-carboxylic acid
N-[(3-methoxyphenyl)methyl]-6-oxo-1-[3-(2-oxopyrrolidin-1-yl)propyl]piperidine-3-carboxamide
2-[1-(cyclohexylmethyl)-4-{[3,5-dimethyl-1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}piperazin-2-yl]ethan-1-ol
2-[4-({3-[(3-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)piperazin-1-yl]ethan-1-ol
(4aR,7aS)-1-methyl-4-[2-(thiophen-2-yl)-1,3-thiazole-4-carbonyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-({2-[4-(pyridin-2-yl)piperazin-1-yl]pyridin-3-yl}methyl)cyclopentanamine
8-[6-ethyl-2-(piperidin-1-yl)pyrimidin-4-yl]-1,3-dioxa-8-azaspiro[4.5]decan-2-one
5-[(4-fluorophenyl)methyl]-3-(oxolan-3-yl)-5-[1-(3-phenylprop-2-ynoyl)piperidin-4-yl]imidazolidine-2,4-dione
4-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}-N-[1-(pyridin-3-yl)propan-2-yl]benzamide
1-({4-[3-(3-ethylphenoxy)azetidine-1-carbonyl]phenyl}methyl)pyrrolidine
7-(2-methoxyethyl)-2-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]-2,7-diazaspiro[4.5]decan-6-one