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N-cyclopropyl-2-methyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]furan-3-carboxamide
N-{1-[1-(2,1,3-benzoxadiazol-4-ylmethyl)piperidin-4-yl]-1H-pyrazol-5-yl}-3-phenylpropanamide
7-[2-(2-ethyl-1H-imidazol-1-yl)ethyl]-2-oxa-7-azaspiro[4.5]decan-8-one
2-(2-hydroxyethyl)-9-(2-methoxy-3-methylbenzoyl)-2,9-diazaspiro[5.5]undecan-3-one
N-[2-(1H-1,2,4-triazol-1-yl)propyl]-N'-(2,4,6-trimethylphenyl)butanediamide
N-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-1-(7-methanesulfonyl-4-methylquinazolin-2-yl)piperidine-3-carboxamide
3-(2,3-dihydro-1H-inden-2-yl)-1-(2-methylpropyl)-8-[(3-methylquinoxalin-2-yl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-[(3S)-1-benzylpyrrolidin-3-yl]-1-methyl-3-(3-methyl-2-oxo-2,3-dihydro-1,3-benzoxazol-5-yl)urea
3-(2-methoxyphenyl)-1-(3-methoxypropyl)-3-{2-[3-(3-methylbutanoyl)piperidin-1-yl]-2-oxoethyl}pyrrolidine-2,5-dione
1-methyl-4-{[5-(oxan-3-ylmethyl)-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazol-3-yl]methyl}piperidine
2,5-dimethyl-N-[2-(pyridin-3-yl)-5,6,7,8-tetrahydroquinazolin-5-yl]furan-3-carboxamide
(1-{[1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}-4-{[3-(trifluoromethyl)phenyl]methyl}piperidin-4-yl)methanol
1-{[2-(3-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-4-ol
2-(ethylsulfanyl)-N-({2-[(6-methylpyridin-3-yl)oxy]pyridin-3-yl}methyl)propanamide
2-[2-methyl-6-(4H-1,2,4-triazol-4-yl)pyridin-3-yl]-N,N-bis(propan-2-yl)benzamide
N-[2-({[2-(dimethylamino)ethyl](thiophen-3-ylmethyl)amino}methyl)quinolin-6-yl]acetamide
(2R,3R,6R)-3-(4-methylphenyl)-5-[3-(propan-2-yl)-1H-pyrazole-5-carbonyl]-1,5-diazatricyclo[5.2.2.02,6]undecane
N-[3-(methylsulfamoyl)phenyl]-3-(pyrimidin-4-yl)piperidine-1-carboxamide
1-{4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazin-1-yl}-3-(trimethyl-1H-pyrazol-4-yl)propan-1-one
2-{[(8-chloro-4-hydroxyquinolin-2-yl)methyl]amino}acetamide
N-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)-2-{4-[hydroxy(1-methyl-1H-imidazol-2-yl)methyl]piperidin-1-yl}acetamide
methyl 2-(2-{1-[(4-methoxy-2,3-dimethylphenyl)methyl]-3-oxopiperazin-2-yl}-N-methylacetamido)acetate
N-(2-methoxyethyl)-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-2-[(2-methylprop-2-en-1-yl)oxy]benzamide
4-({3-phenylpyrazolo[1,5-a]pyrimidin-6-yl}methyl)-2-(trifluoromethyl)morpholine
1-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-3-[5-(thiophen-2-yl)-1,3,4-thiadiazol-2-yl]urea
methyl 5-[4-({[(1S)-1-carbamoylethyl]amino}methyl)phenoxymethyl]furan-2-carboxylate
1-{4-[({1-[2-(4-methoxyphenyl)ethyl]piperidin-4-yl}methyl)(methyl)amino]piperidin-1-yl}ethan-1-one
(3R,7S,8aS)-7-{[(2,4-dimethylphenyl)methyl]amino}-3-[(1S)-1-hydroxyethyl]-octahydropyrrolo[1,2-a]piperazine-1,4-dione
2-(2-methoxy-5-methylphenyl)-5,6-dimethylpyridine-3-carboxamide
(4aS,8aR)-6-(1H-pyrrole-2-carbonyl)-1-[2-(thiophen-2-yl)ethyl]-decahydro-1,6-naphthyridin-2-one
4-{5-[(4-methylpiperidin-1-yl)methyl]-1H-1,2,3,4-tetrazol-1-yl}-1-[2-(1,3-thiazol-2-yl)pyrrolidin-1-yl]butan-1-one
1-(cyclohexylmethyl)-3-[(dimethylamino)methyl]-3-hydroxypiperidin-2-one
3-({3-azaspiro[5.5]undecan-9-yl}amino)-2,3-dihydro-1λ6-thiophene-1,1-dione
2-phenoxy-N-[1-(7-{[4-(pyrrolidin-1-yl)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)ethyl]acetamide
1-({1-[2-(4-chlorophenyl)ethyl]piperidin-3-yl}methyl)-1-methyl-3-propylurea
2-(3,5-dimethyl-1H-pyrazol-4-yl)-2-[2-(2H-indazol-2-yl)acetamido]acetic acid
1-{2,5-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}-4-(2-methylphenyl)-1,4-diazepane
N-[(3S,4R)-1-[(8-methoxy-3,4-dihydro-2H-1,5-benzodioxepin-7-yl)methyl]-4-propylpyrrolidin-3-yl]acetamide
2,3,5-trimethyl-6-{[3-(thiophen-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}pyrazine
1-[(2,5-difluorophenyl)methyl]-N-[4-(1H-pyrazol-5-yl)phenyl]piperidine-3-carboxamide
(2E)-N-[1-(3,5-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-3-(furan-2-yl)prop-2-enamide
1-methyl-4-{[3-(thiophen-3-yl)-1,2,4-oxadiazol-5-yl]methyl}-1,4-diazepane
N-[2-(3-methoxyphenyl)-1-[1-(3-phenylpropyl)piperidin-4-yl]ethyl]-N-methylpyridine-2-carboxamide
(2S,4S)-N-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-1-[(4-chlorophenyl)methyl]-4-{[(4-methoxy-2,3-dimethylphenyl)methyl]amino}pyrrolidine-2-carboxamide
N-[3-(4-chloro-1H-pyrazol-1-yl)propyl]-5-oxo-1-(pyridin-2-ylmethyl)pyrrolidine-3-carboxamide
2-cyclobutyl-5-(2-methoxyacetamido)-1-methyl-N-[(2-methylphenyl)(pyridin-4-yl)methyl]-1H-1,3-benzodiazole-7-carboxamide
4-(azepane-1-carbonyl)-6-methyl-2-[1-(propan-2-yl)-1H-pyrazol-4-yl]quinoline
2-[4-(hydroxymethyl)-4-{[3-(trifluoromethyl)phenyl]methyl}piperidin-1-yl]pyridine-4-carbonitrile
(1S,5R)-6-(1H-imidazol-2-ylmethyl)-3-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
N-cyclohexyl-3-(1-methyl-1H-pyrazol-4-yl)-N-(pyridin-2-ylmethyl)propanamide