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3-({4-[1-(4-methoxyphenyl)-1H-imidazol-2-yl]-1H-1,2,3-triazol-1-yl}methyl)-1λ6-thiolane-1,1-dione
N-[(2R,3R)-2-methoxy-1'-(pyridin-4-ylmethyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-(methylsulfanyl)acetamide
N-({3-methoxy-4-[2-(pyridin-2-yl)ethoxy]phenyl}methyl)-N-[(3S)-2-oxoazepan-3-yl]benzenesulfonamide
5-(piperidin-4-yl)-5-(pyridin-2-yl)imidazolidine-2,4-dione
(2R)-2-amino-2-[1-(1-methylpiperidin-4-yl)-3-(oxan-4-yl)-1H-1,2,4-triazol-5-yl]ethan-1-ol
2-{2-[(dimethylamino)methyl]-4-phenylphenoxy}-N-(1,2,3,4-tetrahydronaphthalen-1-yl)acetamide
N-[(1-ethyl-1H-pyrazol-4-yl)methyl]-3-[(oxolan-3-yl)sulfamoyl]benzamide
2-(3,5-dimethyl-1H-pyrazol-4-yl)-2-{[4,5-dimethyl-2-(1H-pyrrol-1-yl)thiophen-3-yl]formamido}acetic acid
(1-methoxypropan-2-yl)({[3-(1H-pyrazol-4-yl)phenyl]methyl})amine
2-{1-[(2-chloro-4-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-[2-(3-methylpyridin-2-yl)ethyl]acetamide
N-{pyrazolo[1,5-a]pyrimidin-3-ylmethyl}-2-(thiophen-2-yl)-1,3-thiazole-4-carboxamide
3-[4-(1-methyl-3-propyl-1H-pyrazole-5-carbonyl)piperazin-1-yl]-1,2-benzothiazole
N-[(1-cyclopentanecarbonylpiperidin-3-yl)methyl]-4-fluorobenzamide
3-({[2-(2,5-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(prop-2-en-1-yl)amino)-1λ6-thiolane-1,1-dione
1-(4-methoxy-2-{[1,2,4]triazolo[4,3-a]pyridin-3-yl}phenyl)-1H-pyrazole
(3R)-1-{[5-(5-methoxy-1H-indole-2-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}pyrrolidin-3-ol
6-(4-ethylphenyl)-N-[2-(pyridin-3-yloxy)ethyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
N4-[(1-cyclopentylpiperidin-4-yl)methyl]-5-methylpyrimidine-2,4-diamine
1-{3-[2-(methylsulfanyl)benzoyl]piperidin-1-yl}-2-(pyrimidin-2-ylsulfanyl)ethan-1-one
2-{3-[1-(2-phenylethyl)piperidin-4-yl]pyrrolidin-1-yl}pyrimidine
methyl 2-({1-cyclohexyl-5-[(2-methylpropyl)carbamoyl]-4-oxo-1,4-dihydropyridin-3-yl}formamido)-4-(methylsulfanyl)butanoate
N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}-2-(pyrrolidin-1-yl)-5,6,7,8-tetrahydroquinazoline-4-carboxamide
4-ethyl-5-[4-(4-methoxybenzoyl)piperazine-1-carbonyl]-1,3-thiazol-2-amine
N-(2,3-dihydro-1-benzofuran-2-ylmethyl)-N-methyl-5-(2-methylpropyl)-1,2-oxazole-3-carboxamide
1-ethyl-4-{[4-methoxy-3-(pyrrolidin-1-ylmethyl)phenyl]methyl}piperazin-2-one
{[2-(1H-1,3-benzodiazol-1-yl)pyridin-3-yl]methyl}[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]amine
[(3-methylthiophen-2-yl)methyl](pyridin-2-ylmethyl)(4,4,4-trifluorobutyl)amine
ethyl 4-[3-(4-tert-butylbenzoyl)piperidin-1-yl]piperidine-1-carboxylate
1-[1-(furan-3-carbonyl)piperidin-4-yl]-2-[2-(2-methoxyphenyl)ethyl]-1H-1,3-benzodiazole
(3aS,6aR)-3-cyclopentyl-5-{[5-(1H-pyrazol-5-yl)thiophen-2-yl]methyl}-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
[1-(2,3-dimethylquinoxaline-6-carbonyl)-3-(2-phenylethyl)piperidin-3-yl]methanol
(1S,2S)-2-[5-(2,6-dimethoxyphenyl)-4-phenyl-1H-imidazol-1-yl]cyclohexan-1-ol
N-cyclopentyl-N-{[4-methoxy-3-(propan-2-yloxy)phenyl]methyl}-3-phenyl-1,2-oxazole-5-carboxamide
N-ethyl-5-{[methyl({[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl})amino]methyl}pyrimidin-2-amine
3-hydroxy-3-({[(6-methylpyridin-2-yl)methyl]amino}methyl)-1-(3-phenylpropyl)piperidin-2-one
N-(2-hydroxybutyl)-4-{5-[(4-methylpiperidin-1-yl)methyl]-1H-1,2,3,4-tetrazol-1-yl}butanamide
3-{5-[methoxy(phenyl)methyl]-1,3,4-oxadiazol-2-yl}-N-{[3-(trifluoromethyl)phenyl]methyl}propanamide
5-cyclopropyl-N-[phenyl(pyridin-4-yl)methyl]-1H-pyrazole-3-carboxamide
8-[3-(dimethylamino)benzoyl]-2-(2-hydroxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
9-[2-(oxolan-2-ylmethoxy)acetyl]-2-(pyridin-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
2-[4-({4-[2,2-bis(prop-2-en-1-yl)piperidine-1-carbonyl]-1,3-oxazol-2-yl}methyl)piperazin-1-yl]pyrimidine
N-({2-[4-(2-methylphenyl)piperazin-1-yl]pyridin-3-yl}methyl)acetamide
N-[3-hydroxy-1-(4-methylphenyl)propyl]-7-oxo-7H-[1,3]thiazolo[3,2-a]pyrimidine-5-carboxamide
N-(furan-3-ylmethyl)-N,2-dimethyl-3-[(pyridin-3-ylmethyl)amino]benzamide
N-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]-4-(4-methylpiperazin-1-yl)benzamide
1-[(3aR,6aR)-3a-{2-methyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-5-carbonyl}-octahydropyrrolo[3,4-c]pyrrol-2-yl]-2-methoxyethan-1-one
{[2-(ethanesulfonyl)-1-(2-phenylethyl)-1H-imidazol-5-yl]methyl}(methyl)[(1-methylpyrrolidin-2-yl)methyl]amine
1-acetyl-N-[2-(5-phenyl-1,2,4-oxadiazol-3-yl)ethyl]piperidine-3-carboxamide
3-[(2-methoxyethyl)sulfamoyl]-5-(6-methoxypyridin-3-yl)benzoic acid
(2E)-N-({7-[3-(2H-1,3-benzodioxol-5-yl)propanoyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-3-(thiophen-2-yl)prop-2-enamide