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2-methyl-4-(3-{7-methyl-2,7-diazaspiro[4.4]nonane-2-carbonyl}phenyl)butan-2-ol
1-cyclopropyl-4-({4-[2-(5-methylfuran-2-yl)phenyl]-1H-1,2,3-triazol-1-yl}methyl)pyrrolidin-2-one
1-(3-aminothiophene-2-carbonyl)-4-(2-methylquinolin-6-yl)piperidin-4-ol
1-[1-(2-hydroxyethyl)-3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl]-3-(methylsulfanyl)propan-1-ol
[(3R,4R)-1-(3,5-dimethyl-1H-indole-2-carbonyl)-4-(morpholin-4-ylmethyl)pyrrolidin-3-yl]methanol
N-[1-(2,2-dimethylpropyl)-5-oxopyrrolidin-3-yl]-2,5-dimethylthiophene-3-sulfonamide
1-[(1S,5R)-6-(1-benzothiophene-2-sulfonyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]ethan-1-one
5-methyl-N-({2-[4-(pyridin-2-yl)piperazin-1-yl]pyridin-3-yl}methyl)-1,2-oxazole-3-carboxamide
N-{2-fluoro-5-[({2-[(3-methylpyridin-4-yl)amino]ethyl}carbamoyl)amino]phenyl}-2-methylpropanamide
3-[2-(2H-1,3-benzodioxol-5-ylmethyl)-5-oxopyrrolidin-2-yl]-N-[3-(1H-imidazol-1-yl)-1-phenylpropyl]propanamide
3-[(2,5-dimethoxyphenyl)methyl]-9-methoxy-N-methyl-7-oxo-N-(1,3-thiazol-2-ylmethyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
(3S,4R)-1-[3-(azepan-1-ylmethyl)benzoyl]-N,N-dimethyl-4-(propan-2-yl)pyrrolidin-3-amine
4-[1-(1,1-dioxo-1λ6-thiolan-3-yl)-5-(1,2-oxazol-3-yl)-1H-1,2,4-triazol-3-yl]benzamide
2-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl]-6-phenylpyridine-3-carboxylic acid
methyl({4-methyl-5-[(pyridin-4-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl)(2-phenylpropyl)amine
3-{2-[(3aS,6aS)-1-cyclobutanecarbonyl-octahydropyrrolo[2,3-c]pyrrol-5-yl]-2-oxoethyl}-2,3-dihydro-1,3-benzoxazol-2-one
1'-{imidazo[2,1-b][1,3]thiazole-6-carbonyl}-3,4-dihydrospiro[1-benzopyran-2,3'-pyrrolidine]-4-one
1-(2-chlorophenyl)-5-methyl-4-{2-[(5-methyl-1,3,4-oxadiazol-2-yl)sulfanyl]acetyl}piperazin-2-one
4-[(4-fluorophenyl)methyl]-1-(2-methylpyrimidin-4-yl)-3-(propan-2-yl)-1,4-diazepan-5-one
6-[7-(1,3-benzothiazol-2-yl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]pyridine-3-carboxamide
1-[(1R,3R,5S)-3-hydroxy-8-azabicyclo[3.2.1]octan-8-yl]-2-(pyridin-4-yl)ethan-1-one
1-(3-hydroxypropanoyl)-4-(pyrimidin-2-ylmethyl)-1,4-diazepane-6-carboxylic acid
4-methyl-6-(3-methyl-1H-pyrazol-4-yl)-2-(piperidin-1-yl)pyrimidine
N-[(1-ethyl-1H-imidazol-5-yl)methyl]-4-[3-(furan-2-yl)-1,2,4-oxadiazol-5-yl]butanamide
methyl({4-methyl-5-[(pyridin-4-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl)(3-phenylpropyl)amine
N-[3-(1H-indazol-1-yl)propyl]-3-(2-methylpropyl)-1,2-oxazole-5-carboxamide
2-amino-4-[5-(hydroxymethyl)furan-2-yl]-5-methyl-6-phenylpyridine-3-carbonitrile
2-{5-[2-(3-chloro-1,2-oxazol-5-yl)ethyl]-3-cyclopropyl-1H-1,2,4-triazol-1-yl}acetic acid
1-ethyl-2-{1-[3-(pyrrolidin-1-yl)propyl]-1H-imidazol-2-yl}-1H-imidazole
1-[3-(2-chlorophenyl)-5-methyl-1,2-oxazole-4-carbonyl]-3-[(dimethylamino)methyl]piperidin-3-ol
N-(1,1-dioxo-1λ6-thiolan-3-yl)-2-(2-phenylethyl)-1,3-benzoxazole-5-carboxamide
{4-[3-(pyrrolidine-1-carbonyl)pyridin-2-yl]phenyl}methanol
N-(furan-2-ylmethyl)-3-{[4-(pyridin-3-yl)-1H-1,2,3-triazol-1-yl]methyl}piperidine-1-carboxamide
5-butyl-4-(3-cyclopropyl-1H-pyrazole-5-carbonyl)-1-(3-methylphenyl)piperazin-2-one
(1S,5R)-3-[4-methoxy-3-(morpholin-4-yl)benzoyl]-6-methyl-3,6-diazabicyclo[3.2.2]nonan-7-one
N-{2-[(2,6-dimethylphenyl)carbamoyl]phenyl}-3-oxo-2,3-dihydro-1H-indene-1-carboxamide
N-[(1-methyl-2-oxo-1,2,3,4-tetrahydroquinolin-4-yl)methyl]-6-(2-methylpropyl)-2-oxo-1,2-dihydropyrimidine-4-carboxamide
6-[4-(3-fluorophenoxy)piperidine-1-carbonyl]quinoxaline
4-{1-[3-(2H-1,3-benzodioxol-5-yl)-2-methylpropyl]piperidin-4-yl}-5-methylpyrimidine
3-butyl-1-methyl-4-[5-(pyrrolidin-1-ylmethyl)furan-2-carbonyl]piperazin-2-one
3-methyl-7-{5-methylimidazo[1,2-a]pyridine-2-carbonyl}-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
3-(azocan-1-yl)-N-[2-(2-hydroxyethoxy)ethyl]propanamide
2-(2-methyl-1,3-thiazol-4-yl)-N-[2-(6-oxo-3-phenyl-1,4,5,6-tetrahydropyridazin-1-yl)ethyl]acetamide
3-ethyl-N-[2-(4-methoxyphenyl)ethyl]-N-(pyridin-2-ylmethyl)-1,2-oxazole-5-carboxamide
N-[(3-{[1-(3-fluorobenzoyl)piperidin-3-yl]methoxy}phenyl)methyl]-N,1-dimethylpiperidin-4-amine
(2R,3S,6R)-3-(2H-1,3-benzodioxol-5-yl)-5-(1,3-thiazol-2-yl)-1,5-diazatricyclo[5.2.2.02,6]undecane
(2R,3S,6R)-3-(4-methylphenyl)-5-(4-methylpyridine-3-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
N-{1-[7-(1-benzofuran-2-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]-3-methylbutyl}acetamide
(4aR,8aR)-4-({4-[3-(1H-imidazol-1-yl)propoxy]phenyl}methyl)-octahydro-2H-1,4-benzoxazine
N-methyl-6-phenyl-N-{[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}pyridazin-3-amine