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methyl 1-{[2-(6-chloro-2H-1,3-benzodioxol-5-yl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidine-2-carboxylate
5-(1H-imidazol-2-ylmethyl)-2-[3-(trifluoromethyl)phenyl]-2,3,4,5-tetrahydro-1,5-benzothiazepine
N-{1-[1-(5-methoxyfuran-2-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}-2-methylbenzamide
2-methyl-N-[2-(4-phenylpyrimidin-2-yl)ethyl]-1-benzofuran-5-carboxamide
5-hydroxy-N-{2-[1-(2-methylpropyl)piperidin-3-yl]ethyl}-4-oxo-4H-pyran-2-carboxamide
5-cyclopropanecarbonyl-1'-(3-methyl-1H-pyrazole-5-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
N-[3-(2,6-dimethylphenoxy)propyl]-N-methyl-5-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxamide
5-[7-(cyclopropylmethyl)-6-oxo-2,7-diazaspiro[4.5]decane-2-carbonyl]-1-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
3-[2-(2,6-difluorophenyl)ethyl]-1-[3-(1H-1,2,3,4-tetrazol-1-yl)propyl]piperidine
3-(5-{1-[(2R)-3,4-dihydro-2H-1-benzopyran-2-ylmethyl]-1H-imidazol-2-yl}thiophen-2-yl)prop-2-yn-1-ol
2-(propan-2-yl)-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}-1,3-benzoxazole-5-carboxamide
N-[2-(2,3-dihydro-1H-indol-1-yl)ethyl]-2-(morpholin-4-yl)pyrimidine-5-carboxamide
2-{1-[(4-ethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-(2-methylpropyl)acetamide
2-[2-methyl-4-(pyrrolidin-1-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl]pyridin-3-ol
2-[(3-methoxyphenyl)methyl]-8-[2-(1H-pyrazol-1-yl)acetyl]-2,8-diazaspiro[4.5]decan-3-one
2-methyl-4-{3-[2-(5-methyl-1,2-oxazol-3-yl)piperidine-1-carbonyl]phenyl}butan-2-ol
N-[3-(5-amino-1,3,4-thiadiazol-2-yl)propyl]-4-(pyridin-4-yl)pyrimidin-2-amine
2-[(2H-1,3-benzodioxol-5-yloxy)methyl]-N-[1-(3-methylpyridin-2-yl)ethyl]-1,3-oxazole-4-carboxamide
7-(2-methylphenyl)-4-(pyrrolidin-3-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
3-methoxy-2-({3-[methyl(2-phenylethyl)amino]piperidin-1-yl}methyl)phenol
9-(4-chloro-1,5-dimethyl-1H-pyrazole-3-carbonyl)-2-ethyl-2,9-diazaspiro[5.5]undecan-3-one
(2S,4S)-N-ethyl-4-(2-hydroxyacetamido)-1-({7-methylimidazo[1,2-a]pyridin-2-yl}methyl)pyrrolidine-2-carboxamide
1-[(dimethyl-1H-1,2,4-triazol-5-yl)methyl]-3-(trifluoromethyl)-1,2-dihydropyridin-2-one
4-(methoxymethyl)-6-(4-methoxynaphthalen-1-yl)pyrimidine
N-{[4-(2-methylphenyl)-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}thiophene-2-sulfonamide
2-{4-[(3,4-difluorophenyl)methyl]-3-(2-hydroxyethyl)piperazin-1-yl}ethan-1-ol
(3S,5R,9R)-11-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]-5-hydroxy-1,7,11-triazatricyclo[7.4.0.03,7]tridecane-2,8-dione
1-{[(3R,4R)-1-[2-(dimethylamino)benzoyl]-4-(hydroxymethyl)pyrrolidin-3-yl]methyl}piperidin-4-ol
4-[(2-butyl-5-chloro-1H-imidazol-4-yl)methyl]-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
(1S,5R)-3-(2,3-dihydro-1H-inden-2-yl)-6-[1-(propan-2-yl)-1H-pyrazole-4-carbonyl]-3,6-diazabicyclo[3.2.2]nonane
methyl 4-(4-{[2-(furan-2-yl)pyrimidin-5-yl]methyl}piperazin-1-yl)benzoate
6,8-dimethyl-2-{[(pyridin-2-ylmethyl)amino]methyl}quinolin-4-ol
N-[2-methoxy-1-(pyridin-2-yl)ethyl]-N-methyl-2-(2,4,7-trimethyl-1H-indol-3-yl)acetamide
1-{7-[(4-acetylpiperazin-1-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl}-2-(3,5-difluorophenyl)ethan-1-one
N-(3-carbamoylphenyl)-4-[(1-methylpiperidin-4-yl)methyl]piperazine-1-carboxamide
N-methyl-N-[(3-{1-[2-(1H-pyrrol-1-yl)ethyl]-1,2,3,6-tetrahydropyridin-4-yl}-1,2-oxazol-5-yl)methyl]acetamide
N-(2-{7-[(4-ethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-2-(4-fluorophenyl)acetamide
5-fluoro-N,N-dimethyl-2-{4-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyrimidin-4-amine
N-[2-(5-amino-1,3,4-thiadiazol-2-yl)propan-2-yl]-2-(thiophen-2-yl)-1,3-thiazole-4-carboxamide
2-[3-({methyl[2-(pyridin-2-yl)ethyl]amino}methyl)phenyl]-6-(pyridin-3-yl)-3,4-dihydropyrimidin-4-one
3-{[1-(1-propyl-1H-pyrazole-5-carbonyl)pyrrolidin-3-yl]methyl}benzamide
ethyl 4-{2-[6-oxo-4-(pyrrolidin-1-yl)-1,6-dihydropyridazin-1-yl]acetyl}piperazine-1-carboxylate
{[2-(cycloheptanesulfonyl)-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}(methyl)[(4-methyl-1H-imidazol-2-yl)methyl]amine
(1S,5R)-3-[(6-methoxy-2H-chromen-3-yl)methyl]-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
3-(pyridin-4-yl)-5-(pyrrolidine-1-sulfonyl)benzoic acid
9-[1-(2-hydroxyethyl)-1H-1,3-benzodiazole-5-carbonyl]-1-oxa-9-azaspiro[5.5]undecan-5-ol
1-(4-{4-[(4-fluorophenyl)methyl]piperidin-1-yl}-4-oxobutyl)piperidin-2-one
N-({1-[ethyl(methyl)amino]cyclohexyl}methyl)-4,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
(1S,5R)-3-(2,3-dihydro-1H-inden-2-yl)-6-(3-ethyl-5-methyl-1,2-oxazole-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
5-(3-chloro-4-methoxyphenyl)-1-(propan-2-yl)-1H,4H-pyrazolo[3,4-d]imidazole