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1-[(dimethyl-1H-1,2,4-triazol-5-yl)methyl]-4-(2-methylpropyl)pyrrolidin-2-one
N-(3-hydroxy-3-methylbutyl)-N-methyl-2-(3-methyl-4,5-dihydro-1H-pyrazol-1-yl)acetamide
1-{5-[(2,3-dimethoxyphenyl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carbonyl}pyrrolidine
1-{[5-(propan-2-yl)-1H-pyrazol-3-yl]methyl}-3-[3-(trifluoromethyl)benzoyl]piperidine
1-[2-(4-fluorophenoxymethyl)-1,3-oxazole-4-carbonyl]-4-(pyrrolidin-1-yl)piperidine
N-methyl-3-(2-methylpropyl)-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}-1,2-oxazole-5-carboxamide
2-butyl-4-methyl-3-oxo-N-[2-(trifluoromethoxy)phenyl]piperazine-1-carboxamide
N-({1-[2-(4-chlorophenyl)ethyl]piperidin-3-yl}methyl)-N-methyl-2-[methyl(pyridin-3-ylmethyl)amino]acetamide
(1S,5R)-3-benzoyl-N-phenyl-3,6-diazabicyclo[3.2.2]nonane-6-carboxamide
1-(butan-2-yl)-N3-(cyclopropylmethyl)-4-oxo-N5-(prop-2-en-1-yl)-N3-propyl-1,4-dihydropyridine-3,5-dicarboxamide
(1S,4S)-2-methyl-5-{2-[4-(trifluoromethyl)phenyl]-1,3-thiazole-4-carbonyl}-2,5-diazabicyclo[2.2.1]heptane
4-[1-ethyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]-1-(4-methoxyphenyl)piperazin-2-one
4-(3-tert-butyl-1H-pyrazol-1-yl)-1-(4-cyanopyridin-2-yl)piperidine-4-carboxylic acid
2-{[2-(propan-2-yl)pyrimidin-5-yl]methyl}-9-oxa-2-azaspiro[5.5]undecane
N-{2-[3-(pyridin-3-yl)-1H-1,2,4-triazol-5-yl]ethyl}morpholine-2-carboxamide
N-{2-[2-(pyrimidin-2-ylsulfanyl)acetyl]-1,2,3,4-tetrahydroisoquinolin-7-yl}oxolane-2-carboxamide
3-{5-[(2,5-dimethoxyphenyl)methyl]-1,3,4-oxadiazol-2-yl}-1-[2-(pyridin-2-yl)piperidin-1-yl]propan-1-one
{1-[2-({dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}amino)ethyl]piperidin-2-yl}methanol
N-{[3-(methylcarbamoyl)phenyl]methyl}-N'-[2-(methylsulfanyl)phenyl]butanediamide
N-(2,6-dichloropyridin-4-yl)-5H,6H,7H,8H,9H-imidazo[1,5-a][1,4]diazepine-8-carboxamide
N-({1-[2-(4-fluorophenyl)ethyl]piperidin-3-yl}methyl)-N,2-dimethyl-1-benzofuran-5-carboxamide
2-(4-chlorophenyl)-4-(5,6-dimethylpyrimidin-4-yl)morpholine
methyl 3-(1-benzofuran-2-ylmethyl)-9-[(4-fluorophenyl)methoxy]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
N-[(3R,4S)-1-[(methylcarbamoyl)methyl]-4-(propan-2-yl)pyrrolidin-3-yl]-3-phenoxypropanamide
1,3-dimethyl-N-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
1-{4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-2-(1H-indol-1-yl)ethan-1-one
1-(furan-2-ylmethyl)-N-[(2,3,5-trimethyl-1H-indol-7-yl)methyl]piperidine-4-carboxamide
N-[2-(1H-imidazol-1-yl)-1-phenylethyl]-2-(pyridin-3-yl)pyrimidine-5-carboxamide
N-cyclopentyl-3-(dimethyl-1,2-oxazol-4-yl)-N-({1-[2-(2-methylphenyl)ethyl]piperidin-4-yl}methyl)propanamide
N-[2-(oxan-2-yl)ethyl]-2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
1-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}-3-(4-fluorophenoxymethyl)piperidine
1-{3-[3-(5-propylpyrimidin-2-yl)phenyl]-1H-pyrazol-1-yl}butan-2-ol
3-[methyl({2-methyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl})amino]-1-phenylpropan-1-ol
1-{3-[methyl(2-phenylethyl)amino]piperidin-1-yl}-3-(1,2-oxazinan-2-yl)propan-1-one
N-(5-cyclobutyl-1,3,4-oxadiazol-2-yl)-1-(thiophen-2-ylmethyl)piperidin-4-amine
N-(1-{imidazo[1,2-a]pyrimidin-2-yl}propyl)-6-methoxy-3-methyl-1-benzofuran-2-carboxamide
N-{3-[(furan-2-ylmethyl)sulfanyl]propyl}-4-methylpiperidine-4-carboxamide
N-(2-fluoro-4-methylphenyl)-2,3-dimethyl-4-oxo-3H,4H,5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carboxamide
3-chloro-4-methoxy-N-methyl-N-{[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl}benzamide
5-fluoro-3-(2-hydroxybutyl)-3,4-dihydroquinazolin-4-one
2-{2-[5-fluoro-2-(1H-pyrazol-1-yl)phenyl]-1H-imidazol-1-yl}-1-phenylethan-1-ol
4-[4-({[1-(hydroxymethyl)cyclobutyl]methyl}amino)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-2-yl]benzamide
4-[(5-{1-[(1-ethyl-1H-imidazol-2-yl)methyl]piperidin-3-yl}-4-methyl-4H-1,2,4-triazol-3-yl)methyl]morpholine
1-(3-methylbutyl)-N-[3-(1,3-thiazol-4-yl)phenyl]piperidine-4-carboxamide
(2S,4R)-4-amino-N-ethyl-1-[2-(1H-1,2,4-triazol-3-yl)benzoyl]pyrrolidine-2-carboxamide
9-ethyl-1-methyl-4-(4,5,6,7-tetrahydro-1-benzothiophene-3-carbonyl)-1,4,9-triazaspiro[5.6]dodecan-10-one
benzyl({[1-(1,3-thiazol-2-yl)-1H-pyrrol-2-yl]methyl})(1,3-thiazol-2-ylmethyl)amine
2-{2-[1-benzyl-3-(1H-1,2,4-triazol-1-ylmethyl)-1H-1,2,4-triazol-5-yl]ethyl}-1-methylpiperidine
(1S,5R)-6-[5-(propan-2-yl)-1,2-oxazole-3-carbonyl]-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
2-(1,3-benzoxazol-2-yl)-1-[6-hydroxy-4-(2-hydroxyethyl)-1,4-diazepan-1-yl]ethan-1-one