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2-(1-{8-methylimidazo[1,2-a]pyridine-2-carbonyl}piperidin-3-yl)-1,2,3,4-tetrahydroisoquinoline
(2R)-2-amino-N-{[2-(3,4-difluorophenoxy)pyridin-3-yl]methyl}-3-hydroxypropanamide
[(3R,4R)-4-[(dimethylamino)methyl]-1-[2-methyl-5-(propan-2-yl)furan-3-carbonyl]pyrrolidin-3-yl]methanol
1-({3-[3-(3,5-dimethyl-1H-pyrazol-1-yl)azetidine-1-carbonyl]-1H-pyrazol-5-yl}methyl)-1H-indole
2-[3-(hydroxymethyl)-3-(3-methylbut-2-en-1-yl)piperidin-1-yl]acetic acid
8-[(4-chloro-1-methyl-1H-indazol-3-yl)methyl]-1-ethyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-[3-chloro-4-(2,2-dimethylpropanamido)phenyl]-2,1-benzoxazole-3-carboxamide
4-(furan-3-ylmethyl)-2-[(3-methoxyphenyl)methyl]morpholine
4-[5-methoxy-2-(pyrrolidine-1-carbonyl)phenoxy]-1-{[(4S)-4-(prop-1-en-2-yl)cyclohex-1-en-1-yl]methyl}piperidine
5-[(2-chlorophenyl)methyl]-5-[1-(2,4-dimethoxybenzoyl)piperidin-4-yl]imidazolidine-2,4-dione
6-amino-N-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}-N-(oxolan-2-ylmethyl)pyridine-3-carboxamide
5-(3-fluorophenyl)-N-[2-(2-methoxyphenyl)ethyl]-1,2,4-triazin-3-amine
ethyl 5-[(4-acetamidophenyl)methyl]-1-[2-(4-methoxyphenyl)ethyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
N-[4-(4-{[2-(methylsulfanyl)ethyl]amino}piperidin-1-yl)phenyl]-2-phenoxyacetamide
5-(2H-1,3-benzodioxol-5-ylmethyl)-1-[3-(1H-imidazol-1-yl)propyl]-5-methylpiperidin-2-one
4-(2-methylphenoxy)-1-(6-oxo-1,4,5,6-tetrahydropyridazine-3-carbonyl)piperidine-4-carboxylic acid
7-methyl-3-({3-methyl-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl}methyl)-2-(thiophen-2-yl)quinoline
N-[(4-chloro-3-methyl-1H-pyrazol-5-yl)methyl]-N-ethyloxan-4-amine
5-methoxy-2-({3-[3-(propan-2-yloxy)benzoyl]piperidin-1-yl}methyl)pyridin-4-ol
N-(dicyclopropylmethyl)-1-[(4-methoxyphenyl)methyl]-N-methyl-1H-1,2,3-triazole-4-carboxamide
(2R)-2-({6-[(diethylamino)methyl]pyrazolo[1,5-a]pyrimidin-3-yl}formamido)propanamide
9-[2-(methylamino)pyridine-4-carbonyl]-2-(pyridin-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
N-[1-(4-fluorophenyl)-2-methylpropan-2-yl]-6-oxopiperazine-2-carboxamide
3-acetamido-N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}thiophene-2-carboxamide
N,N-dimethyl-2-[(1S,5R)-6-[2-(4-methyl-1,2,5-oxadiazol-3-yl)acetyl]-3,6-diazabicyclo[3.2.2]nonan-3-yl]acetamide
N-(1-{[2-(2,5-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-4-yl)acetamide
(1R,5R)-N,N-dimethyl-6-[5-(propan-2-yl)-1,2-oxazole-3-carbonyl]-3,6-diazabicyclo[3.2.2]nonane-3-sulfonamide
3-(5-{pyrazolo[1,5-a]pyridine-3-carbonyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl)propanoic acid
4-(2,3-dimethylphenyl)-3-(1H-1,2,3,4-tetrazol-5-ylmethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
5-methoxy-2-[2-(3-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl]phenol
7-cyclopropanecarbonyl-N-methyl-N-[(3-methylpyridin-2-yl)methyl]-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
1-benzyl-5-(3-methylpiperidine-1-carbonyl)-4-oxo-N-(prop-2-en-1-yl)-1,4-dihydropyridine-3-carboxamide
6-(3-methyl-1H-pyrazol-1-yl)-2,3,4,9-tetrahydro-1H-carbazol-1-one
2-(2,4-dichlorophenoxy)-N-{1-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]ethyl}acetamide
2-({[(3R,4R)-1-(2,3-dimethyl-1H-indole-5-carbonyl)-4-(hydroxymethyl)pyrrolidin-3-yl]methyl}(ethyl)amino)ethan-1-ol
1-(5-cyanopyridin-2-yl)-N-[2-(pyridin-3-yloxy)phenyl]piperidine-3-carboxamide
(2S,4S)-1-acetyl-N,N-diethyl-4-[3-(pyridin-4-yl)propanamido]pyrrolidine-2-carboxamide
2-(1H-imidazol-4-yl)-1-[3-(propan-2-yl)phenyl]-1H-imidazole
N-[4-(1H-1,3-benzodiazol-2-yl)phenyl]-1-{[5-(methoxymethyl)furan-2-yl]methyl}piperidine-4-carboxamide
1-[2-(4-chlorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]-2-(1H-pyrazol-1-yl)butan-1-one
4-{[4-(dimethylamino)-5-methylpyrimidin-2-yl]amino}-1λ6-thiane-1,1-dione
5-[(1S,5R)-3-(3-phenylpropyl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-1,2-dihydropyridin-2-one
N-{[3-(propan-2-yl)-1,2-oxazol-5-yl]methyl}-2-[5-(pyrrolidin-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]acetamide
6-(cyclopentylamino)-N-[(3-propyl-1,2-oxazol-5-yl)methyl]pyridine-3-carboxamide
3-amino-N-[1-(6-chloropyridazin-3-yl)piperidin-4-yl]-1H-1,2,4-triazole-5-carboxamide
1-(cyclopropylmethyl)-4-{5-[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}piperazine
(2S)-2-acetamido-N-{[7-(3-methylpyridin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-4-(methylsulfanyl)butanamide
5-[1-(2-aminoacetyl)pyrrolidin-2-yl]-N-[(5-cyclopropyl-1H-pyrazol-3-yl)methyl]thiophene-2-carboxamide
N-[1-({[(5-tert-butyl-1H-pyrazol-3-yl)methyl]carbamoyl}methyl)-1H-pyrazol-4-yl]pyridine-2-carboxamide
N-benzyl-2-[(1R,5R)-3-(pyridine-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]acetamide