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N-(1-{1-[1-(methylsulfanyl)propan-2-yl]piperidin-4-yl}-1H-pyrazol-5-yl)-1-phenylmethanesulfonamide
2-({4-[2-(ethylamino)pyrimidin-5-yl]-1H-1,2,3-triazol-1-yl}methyl)-3,4-dihydroquinazolin-4-one
(1R,5S,6S)-6-{[4-(4-methoxyphenoxy)piperidin-1-yl]methyl}-3-azabicyclo[3.1.0]hexane
2-amino-4-(4-fluorophenyl)-6-(trimethyl-1H-pyrazol-4-yl)pyridine-3-carbonitrile
1-(5-oxo-1-{[2-(trifluoromethyl)phenyl]methyl}pyrrolidin-3-yl)-3-(prop-2-en-1-yl)urea
2-(dimethylamino)-N-{[7-(pyrimidin-5-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}acetamide
5-(2-cyclopentylacetamido)-1-methyl-N-[(3-methylpyridin-2-yl)methyl]-2-(oxolan-2-yl)-1H-1,3-benzodiazole-7-carboxamide
1-(dimethyl-1,2-oxazole-4-carbonyl)-3-[4-(4-fluorophenyl)-1H-pyrazol-5-yl]piperidine
N-{1-[1-(cyclohex-1-ene-1-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}oxolane-3-carboxamide
2-(6-methoxynaphthalen-2-yl)-4-(5-propyl-1,2-oxazole-3-carbonyl)morpholine
4-(3,3-diphenylpiperidin-1-yl)-4-oxobutanamide
3-[(1R,4R)-2-azabicyclo[2.2.1]heptan-2-yl]-N-{[2-(3,4-difluorophenoxy)pyridin-3-yl]methyl}propanamide
3-amino-N-[(3,5-dimethoxyphenyl)methyl]-N-(1-methoxypropan-2-yl)benzamide
4-[4-(4-methoxybenzoyl)piperazin-1-yl]-4-oxobutane-1-sulfonamide
N-(cyclobutylmethyl)-2-{2,5-dioxo-3-phenyl-1-[2-(pyridin-2-yl)ethyl]pyrrolidin-3-yl}-N-(oxolan-2-ylmethyl)acetamide
1-[5-(1,5-dimethyl-1H-pyrazol-4-yl)-1,2-oxazole-3-carbonyl]-3-(1H-imidazol-1-ylmethyl)piperidine
5-[6-oxo-2-(propan-2-yl)-1,6-dihydropyrimidine-5-carbonyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylic acid
8-{10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-yl}-1-oxa-8-azaspiro[4.5]decan-3-ol
2-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-4-[4-(3-fluorobenzoyl)piperazin-1-yl]-2,3-dihydro-1H-isoindole-1,3-dione
1-(2,3-dihydro-1,4-benzodioxin-6-yl)-3-methyl-3-{[5-(propan-2-yl)-1,2-oxazol-3-yl]methyl}urea
methyl (2S,3S)-3-methyl-2-({1-[(5-methylfuran-2-yl)methyl]-4-oxo-5-[(prop-2-en-1-yl)carbamoyl]-1,4-dihydropyridin-3-yl}formamido)pentanoate
2-ethyl-N-(6-methoxy-1,3-benzothiazol-2-yl)-4-methyl-1,3-oxazole-5-carboxamide
6-ethoxy-3-{[(1R,3S,5S)-3-hydroxy-8-azabicyclo[3.2.1]octan-8-yl]methyl}-1,2-dihydroquinolin-2-one
methyl 3-[2-(3-fluorophenyl)acetamido]-6-{[methyl(1,3-thiazol-4-ylmethyl)amino]methyl}thieno[2,3-b]pyridine-2-carboxylate
2-[(1S,4R)-2-azabicyclo[2.2.1]heptan-2-yl]-N-methyl-N-{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}acetamide
2-methanesulfonamido-N-methyl-N-[(3-phenyl-1,2-oxazol-5-yl)methyl]acetamide
N-[1-({[(1R)-1-(4-methoxyphenyl)ethyl]carbamoyl}methyl)-1H-pyrazol-4-yl]furan-2-carboxamide
1-ethyl-3-(piperidine-1-carbonyl)-N-[2-(thiophen-2-yl)ethyl]-4,5,6,7-tetrahydro-1H-indazol-5-amine
4-({[(3-ethoxyphenyl)methyl](2-hydroxyethyl)amino}methyl)-N-methylbenzene-1-sulfonamide
N-methyl-N-(oxan-4-yl)-2-oxo-1-phenylpyrrolidine-3-carboxamide
3-ethyl-8-({5-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]furan-2-yl}methyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N,N-diethyl-4-[4-ethyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carboxamide
(2R,3R,6R)-5-(2,5-dimethylfuran-3-carbonyl)-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
N-ethyl-2-(7-fluoro-2-methyl-1H-indol-3-yl)-N-[2-hydroxy-2-(3-hydroxyphenyl)ethyl]acetamide
N-{1-[5-methyl-1-(2-methylphenyl)-1H-pyrazol-4-yl]ethyl}-3-(trimethyl-1H-pyrazol-4-yl)propanamide
2-(1-benzothiophen-7-yl)-2-[4-hydroxy-4-(pyridin-3-yl)piperidin-1-yl]acetic acid
6-(2-methoxyethyl)-2-[4-({methyl[(5-methyl-1H-pyrazol-3-yl)methyl]amino}methyl)phenyl]-3,4-dihydropyrimidin-4-one
2-cyclopropyl-N-{[1-(hydroxymethyl)cyclobutyl]methyl}-N-methylpyrimidine-5-carboxamide
ethyl 4-[6-(2,3-dimethylbenzoyl)-6-azaspiro[2.5]octane-1-amido]piperidine-1-carboxylate
3-(1-cyclopentyl-4-methyl-1H-pyrazol-5-yl)-1-[1-(pyrazin-2-yl)propan-2-yl]urea
1-{3-[(2,2-dimethylpyrrolidin-1-yl)methyl]phenoxy}-3-(morpholin-4-yl)propan-2-ol
2-(4-{[5-methyl-2-(4-phenylphenyl)-1,3-oxazol-4-yl]methyl}piperazin-1-yl)pyrazine
N-{1-[(2-fluorophenyl)methyl]piperidin-3-yl}-N-methyl-3-(1-methyl-1H-pyrrol-2-yl)-1H-pyrazole-5-carboxamide
6-({[3-(1,2,3,4-tetrahydroquinolin-1-yl)propyl]amino}methyl)-1,4-oxazepan-6-ol
N-[3-methyl-1-(pyridin-3-yl)butyl]-2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
N-[(1-ethyl-5-methyl-1H-pyrazol-4-yl)methyl]-1-methyl-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
5-{1-[(4-ethylphenyl)methyl]piperidin-4-yl}-3-(2-methoxyethyl)-5-[(3-methoxyphenyl)methyl]imidazolidine-2,4-dione
N-{2-[(4-ethyl-5-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}-8-fluoroquinoline-2-carboxamide
ethyl 1-[2-(1H-imidazol-4-yl)ethyl]-4-oxo-5-phenoxy-1,4-dihydropyridine-3-carboxylate
N-[1-(3-methyl-1,2,4-oxadiazol-5-yl)propyl]-3-(pyrrolidine-1-carbonyl)benzene-1-sulfonamide