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1-(2-{[benzyl(methyl)amino]methyl}phenoxy)-3-(piperidin-1-yl)propan-2-ol
2-(4-{4-[3-(pyrrolidine-1-carbonyl)piperidin-1-yl]piperidine-1-carbonyl}-1H-1,2,3-triazol-1-yl)ethan-1-amine
3-[3-(2-ethoxyethyl)-5-methyl-1H-1,2,4-triazol-1-yl]-4-fluorobenzene-1-sulfonamide
1-[(4-chlorophenyl)methyl]-5-[4-(furan-2-carbonyl)-1,4-diazepane-1-carbonyl]piperidin-2-one
1-(5-chloropyridin-2-yl)-4-{5-[(methylsulfanyl)methyl]furan-2-carbonyl}piperazine
(1S,5R)-3-(3-{[(4-fluorophenyl)methyl]sulfanyl}propanoyl)-6-methyl-3,6-diazabicyclo[3.2.2]nonan-7-one
methyl (2S,4R)-4-(dimethylamino)-1-[1-(3,5-dimethylphenyl)piperidin-4-yl]pyrrolidine-2-carboxylate
(1R,5R)-3-(5-methoxy-2,4-dimethylbenzenesulfonyl)-6-methyl-3,6-diazabicyclo[3.2.2]nonane
(6R)-6-[3-(2-phenylethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine-7-carbonyl]-1,3-diazinane-2,4-dione
1-[(1S,2R)-2-butylcyclopropanecarbonyl]-4-[4-(2-methylpropyl)-1H-1,2,3-triazol-1-yl]piperidine
[(5-methoxy-1H-indol-2-yl)methyl]({[2-(3-methylphenyl)pyrimidin-5-yl]methyl})amine
3-fluoro-N-[1-(2-hydroxyphenyl)ethyl]-7-methylimidazo[1,2-a]pyridine-2-carboxamide
1-[7-(1-benzothiophen-3-yl)-9-ethoxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-(dimethyl-1,2-oxazol-4-yl)ethan-1-one
4-(2,5-dimethoxyphenyl)-3-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-4H-1,2,4-triazole
N-({1-[2-(2-methoxyphenyl)ethyl]piperidin-4-yl}methyl)-N-methylfuran-2-carboxamide
1-(2-methyl-1H-pyrrole-3-carbonyl)-3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidine
methyl 2-[1-(2-methoxyethyl)-2,4-dioxo-8-(pyridin-4-ylmethyl)-1,3,8-triazaspiro[4.5]decan-3-yl]acetate
(1S,5R)-3-{6-methylpyrazolo[1,5-a]pyrimidine-3-carbonyl}-6-propyl-3,6-diazabicyclo[3.2.2]nonan-7-one
(2S,4R)-4-amino-1-{[3-(4-chlorophenoxy)phenyl]methyl}-N-methylpyrrolidine-2-carboxamide
5-methoxy-1-methyl-N-{2-[(pyridin-3-yl)amino]ethyl}-1H-indole-2-carboxamide
5-(furan-2-yl)-3-methyl-1-(2-methylpropyl)-1H,4H-pyrazolo[3,4-d]imidazole
N-[1-(6-methylpyridin-2-yl)propan-2-yl]-9H-purin-6-amine
5-[4-(3-methylphenoxy)piperidine-1-carbonyl]-1-[3-(2-oxopyrrolidin-1-yl)propyl]piperidin-2-one
3-(2,3-dihydro-1H-inden-2-yl)-8-[(2-fluorophenyl)methyl]-1-(2-methoxyethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-(3-chlorobenzoyl)-1-[(trimethyl-1H-pyrazol-4-yl)sulfonyl]piperidine
5-butyl-1-(3-phenylphenyl)-4-(1H-pyrazole-3-carbonyl)piperazin-2-one
N-[(2R,4R,6S)-2-cyclohexyl-6-(isoquinolin-5-yl)oxan-4-yl]acetamide
3-(2,3-dimethoxyphenyl)-1-{2-methyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl}pyrrolidine
1-[(1s,4s)-4-aminocyclohexyl]-N-[1-(thiophen-2-yl)propan-2-yl]-1H-1,2,3-triazole-4-carboxamide
2-[ethyl({[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl})amino]-2-(4-fluoro-3-methylphenyl)acetic acid
N-cyclohexyl-N-(pyridin-2-ylmethyl)-[1,2,4]triazolo[4,3-a]pyridine-7-carboxamide
2-[3-(pyridin-3-yl)propyl]-1H,2H-pyrrolo[1,2-d][1,2,4]triazin-1-one
N-(3-chloro-4-methoxyphenyl)-6-[(2-fluorophenyl)methyl]-6-azaspiro[2.5]octane-1-carboxamide
N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-N-methyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxamide
1-methanesulfonyl-4-(2,3,4,5-tetrahydro-1-benzoxepine-4-carbonyl)-1,4-diazepane
1-[(1-methyl-1H-imidazol-4-yl)sulfonyl]-4-(5-methylpyridin-2-yl)piperidin-4-ol
N-({5-methyl-2-[4-(2-phenylacetamido)phenyl]-1,3-oxazol-4-yl}methyl)cyclohex-3-ene-1-carboxamide
7-{[(2S)-2-(methoxymethyl)pyrrolidin-1-yl]methyl}-2,3-dimethyl-1H-indole
8-(9H-purin-6-yl)-1-oxa-8-azaspiro[4.5]decane
1-[(5-{1-methyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazine-2-carbonyl}furan-2-yl)methyl]-1H-imidazole
N,N-diethyl-1-(4-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}benzoyl)pyrrolidin-3-amine
5-[1-(2,5-dimethylphenyl)-3-methyl-1H-1,2,4-triazol-5-yl]-2-methyl-1,4-dihydropyridin-4-one
N-(isoquinolin-5-ylmethyl)-N-methyl-1-(pyrimidin-2-yl)piperidin-4-amine
2-{[8-(2-hydroxyethyl)-9-oxo-2,8-diazaspiro[5.5]undecan-2-yl]methyl}benzonitrile
(1S,2S)-2-[4-(7-methoxy-4-methylquinazolin-2-yl)piperazin-1-yl]cyclohexan-1-ol
(3aS,6aS)-2-(4-cyanopyridin-2-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
6-tert-butyl-1-methyl-N-{[5-(2-methylpropyl)-1,2-oxazol-3-yl]methyl}-1H-pyrazolo[3,4-d]pyrimidin-4-amine
2-[3-(2-ethyl-1H-imidazol-1-yl)propanoyl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
2-[1-benzyl-3-(1-phenylcyclopropyl)-1H-1,2,4-triazol-5-yl]morpholine
(4aS,8aR)-6-{[2-(furan-2-yl)pyrimidin-5-yl]methyl}-1-propyl-decahydro-1,6-naphthyridin-2-one