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N-[4-(3-fluorophenyl)phenyl]-1-(5-methyl-1,3-oxazole-4-carbonyl)pyrrolidine-2-carboxamide
2-(ethoxymethyl)-N-[2-(2-fluorophenyl)ethyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
1-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-3-[(dimethylamino)methyl]pyrrolidin-3-ol
6-[4-(1-hydroxy-3-methylbutyl)piperidine-1-carbonyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-{[7-(6-methoxypyridazin-3-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-4-methyl-1,3-oxazole-5-carboxamide
1-[2-methoxy-5-({methyl[(5-methyl-1H-pyrazol-3-yl)methyl]amino}methyl)phenoxy]-3-(4-methylpiperazin-1-yl)propan-2-ol
1-[1-(furan-2-ylmethyl)piperidine-4-carbonyl]-4-(pyridin-4-ylmethyl)-1,4-diazepane
N-(1-{[(furan-2-ylmethyl)carbamoyl]methyl}-1H-pyrazol-4-yl)-4-oxo-4-phenylbutanamide
4-({1-[(4-fluorophenyl)methyl]-3-hydroxy-2-oxopiperidin-3-yl}methyl)piperazine-1-sulfonamide
4-(1H-imidazol-1-yl)-N-[2-(4-phenylpiperidin-1-yl)ethyl]benzamide
N-[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]-2-(pyridin-3-yl)pyrimidine-5-carboxamide
4-{4-[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]pyrimidin-2-yl}-1,4-oxazepane
2-[(dimethylamino)methyl]-N-methyl-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}-1,3-thiazole-4-carboxamide
N-tert-butyl-5-chloro-2-{[1-(pyridin-4-ylmethyl)piperidin-4-yl]oxy}benzamide
3-hexyl-8-(6-methylpyridine-2-carbonyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
4-[2-amino-3-cyano-6-(2,2-dimethyloxan-4-yl)-5-methylpyridin-4-yl]benzamide
2-(6-aminopyrimidin-4-yl)-7-(oxan-4-yl)-2,7-diazaspiro[4.5]decan-6-one
1-(1-benzylpiperidin-4-yl)-3-(3-methyl-1,2,4-thiadiazol-5-yl)urea
1-[(5-methylthiophen-2-yl)methyl]-4-[5-(trifluoromethyl)-1,3,4-thiadiazol-2-yl]piperazine
1-[2-(dimethylamino)propanoyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
N-[(2R,3R)-1'-(2,6-difluorobenzoyl)-2-(2-methoxyethoxy)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-methylpropanamide
1-(2-{5,6-dimethyl-4-oxo-3H,4H-thieno[2,3-d]pyrimidin-3-yl}ethyl)imidazolidin-2-one
6-[(2,3-dimethoxyphenyl)methyl]-N-(2-methyl-1,3-benzothiazol-5-yl)-6-azaspiro[2.5]octane-1-carboxamide
4-{3-[4-(4-methoxyphenyl)piperazin-1-yl]piperidine-1-carbonyl}-N,N-dimethylaniline
1-methyl-5-[(2-{2-[4-(trifluoromethyl)phenyl]-1H-imidazol-1-yl}ethyl)sulfanyl]-1H-1,2,3,4-tetrazole
4-phenyl-1-{[6-(piperidine-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl}-1,2,3,6-tetrahydropyridine
(1S,5R)-3-[3-(2-methyl-1H-imidazol-1-yl)propanoyl]-6-(3-methylbut-2-en-1-yl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N-(4-cyano-2-fluorophenyl)-4-(3-methylpyridin-4-yl)-1,4-diazepane-1-carboxamide
N-benzyl-N-(cyclobutylmethyl)-2-(5,5-dimethyl-2,4-dioxo-1,3-oxazolidin-3-yl)acetamide
1-{5-ethyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-2-(3-fluoro-4-hydroxyphenyl)ethan-1-one
3-(2,3-dihydro-1H-inden-2-yl)-1-(2-methylpropyl)-8-[(1-phenyl-1H-pyrazol-4-yl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
6-cyclopentyl-3-{[(4-hydroxybutan-2-yl)amino]methyl}-2-methoxy-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
1-[1-(4-fluorobenzenesulfonyl)piperidin-3-yl]-N-(propan-2-yl)-1H-1,2,3-triazole-4-carboxamide
1-[(2S,6S)-6-butyl-2-(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridin-1-yl]-3-[5-(1H-indol-3-ylmethyl)-1,3,4-oxadiazol-2-yl]propan-1-one
[7-(4-chloro-2-methylphenyl)-2,3-dihydro-1-benzofuran-2-yl]methanamine
5-(piperazin-1-yl)-2-{[6-(trifluoromethyl)pyridin-3-yl]methyl}-2,3-dihydropyridazin-3-one
(1S,5R)-6-(1-methyl-1H-indole-2-carbonyl)-3-(oxan-4-yl)-3,6-diazabicyclo[3.2.2]nonane
2-(2,3-dihydro-1H-inden-1-yl)-N-[(4-phenyloxan-4-yl)methyl]acetamide
N-[2-(1-benzylpiperidin-2-yl)ethyl]-4-(pyridin-2-yl)pyrimidin-2-amine
(3aR,7aS)-2-[1-(furan-2-ylmethyl)piperidine-4-carbonyl]-2,3,3a,4,7,7a-hexahydro-1H-isoindole
3-{[(3-hydroxypyrrolidin-3-yl)methyl]sulfamoyl}-N-phenylbenzamide
1-[(4aS,8aS)-4a-hydroxy-7-(pyridin-2-ylmethyl)-decahydro-2,7-naphthyridin-2-yl]-2-cyclobutylethan-1-one
1,3-dimethyl-5-{[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]methyl}imidazolidine-2,4-dione
1-{[4-(methylsulfanyl)phenyl]methyl}-N-[3-(1H-1,2,3,4-tetrazol-1-yl)phenyl]pyrrolidine-2-carboxamide
1-(2-methyl-4-{[3-(pyridin-3-yloxy)propyl]amino}-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl)ethan-1-one
(4S)-3-({2-methyl-5-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidin-7-yl}methyl)-4-phenyl-1,3-oxazolidin-2-one
N-{2-cyclobutyl-7-[3-(2-fluorophenyl)pyrrolidine-1-carbonyl]-1-methyl-1H-1,3-benzodiazol-5-yl}-2-methoxyacetamide
(2S,4S)-4-amino-1-[3-(3-chloro-1H-1,2,4-triazol-5-yl)propanoyl]-N-(propan-2-yl)pyrrolidine-2-carboxamide
3-{[7-(2,6-dimethoxyphenyl)-9-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]methyl}-6-methyl-4H-chromen-4-one
(3S)-1-({5-[(4,5-dimethylfuran-2-yl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-3-fluoropyrrolidine