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2,2-dimethyl-1-{7-[(4-methylpiperazin-1-yl)sulfonyl]-1,2,3,4-tetrahydroisoquinolin-2-yl}propan-1-one
1-{[3,5-dimethyl-2-(1H-pyrazol-1-yl)phenyl]methyl}-4-(1H-pyrazol-3-yl)piperidine
(3aS,6aS)-2-methanesulfonyl-5-[3-(2-methyl-1H-imidazol-1-yl)propyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
3-chloro-6-{4-[(4-methylphenyl)methyl]-3-oxopiperazin-1-yl}pyridine-2-carboxylic acid
propan-2-yl 4-{2-chloro-4-[(2-methoxyethyl)carbamoyl]phenoxy}piperidine-1-carboxylate
methyl 6-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-2-[ethyl(2-methylprop-2-en-1-yl)sulfamoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
1-cyclopropanecarbonyl-2-(3-methyl-1H-1,2,4-triazol-5-yl)piperidine
dimethyl(2-{[(3-methylthiophen-2-yl)methyl](pyridin-3-ylmethyl)amino}ethyl)amine
3-[(2-methyl-5-oxo-1,4-diazepan-1-yl)methyl]-7-(methylsulfanyl)-1,2-dihydroquinolin-2-one
(4aS,7aR)-1-(6-methylpyridine-2-carbonyl)-4-(pyrimidin-2-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-[2-(morpholin-4-yl)ethyl]-5,5-diphenylpiperidin-2-one
N-methyl-2-(pyridin-3-yl)-N-[2-(pyridin-4-yl)ethyl]acetamide
ethyl 4-[(4-methoxyphenyl)methyl]-1-[2-(pyridin-4-ylsulfanyl)acetyl]piperidine-4-carboxylate
N-(1-hydroxybutan-2-yl)-3-propyl-N-(pyridin-2-ylmethyl)-1H-pyrazole-5-carboxamide
(1S,5R)-3-(1-benzofuran-2-ylmethyl)-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
2-methyl-4-(4-methyl-3-oxopiperazine-1-carbonyl)-1,2-dihydrophthalazin-1-one
N-(4-butanamido-3-methoxyphenyl)-5,7-dimethyl-[1,2,4]triazolo[4,3-a]pyrimidine-3-carboxamide
N-({7-[(2-chloro-6-fluorophenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)benzamide
(5S,9aS,9bS)-2-cyclopentyl-5-(2-methyl-1H-imidazol-4-yl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
8-methoxy-N-methyl-N-[2-(1H-pyrazol-4-yl)ethyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
2-[3-(2-methoxyphenoxy)azetidine-1-carbonyl]-1-methyl-1H-pyrrole
(4S)-3-[2-(4,4-difluoropiperidin-1-yl)-2-oxoethyl]-4-phenyl-1,3-oxazolidin-2-one
2-(adamantan-1-yl)-N-{[1-(2-methoxyethyl)-5-oxopyrrolidin-3-yl]methyl}acetamide
3-{[(1H-indazol-4-yl)carbamoyl](methyl)amino}-N-methylbutanamide
[1-(1-phenyl-1H-pyrazole-4-carbonyl)-3-(3-phenylpropyl)piperidin-3-yl]methanol
4-(furan-3-carbonyl)-9-methoxy-7-(2-methoxyphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
4-(2,3-dihydro-1H-inden-2-yl)-3-[2-oxo-2-(4-phenylpiperidin-1-yl)ethyl]piperazin-2-one
(3S,4R)-1-(5-methoxyfuran-2-carbonyl)-4-(pyridin-3-yl)pyrrolidine-3-carboxylic acid
2-(4-{[propyl(pyridin-4-ylmethyl)amino]methyl}phenyl)-3,4,5,6,7,8-hexahydroquinazolin-4-one
1-{2-ethyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl}-3-(3-methoxyphenoxymethyl)piperidine
4-[(3,4-difluorophenyl)methyl]-7-(thiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
methyl 9-(cyclopentyloxy)-3-[3-(dimethyl-1,2-oxazol-4-yl)propanoyl]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
N-[2-(4-fluorophenyl)ethyl]-N-{[7-methoxy-2-(morpholin-4-yl)quinolin-3-yl]methyl}propanamide
2-[2-(4-methanesulfonylphenyl)-1H-1,3-benzodiazol-1-yl]ethan-1-ol
N-[2-(diethylamino)ethyl]-3-(4-methylthiophen-2-yl)-5-(morpholine-4-sulfonyl)benzamide
4-(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)-N-[1-(pyridin-4-yl)propan-2-yl]pyrimidin-2-amine
ethyl 1-[(3-methylquinoxalin-2-yl)methyl]-4-(oxan-2-ylmethyl)piperidine-4-carboxylate
3-[7-(1,3-benzothiazol-2-yl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-N-ethylpropanamide
2-{1-cyclohexyl-4-[(1-ethyl-1H-1,3-benzodiazol-2-yl)methyl]piperazin-2-yl}ethan-1-ol
(3S,4S)-3-[(1-benzylpiperidin-4-yl)(methyl)amino]-4-hydroxy-1λ6-thiolane-1,1-dione
7-(2-methoxyethyl)-2-[4-(trifluoromethyl)pyrimidin-2-yl]-2,7-diazaspiro[4.5]decan-6-one
3-{[(3-methylthiophen-2-yl)methyl]amino}-N-[3-(pyrrolidin-1-yl)propyl]benzamide
3-[2-(furan-2-yl)azepane-1-carbonyl]-6-(propan-2-yl)-1,2-dihydropyridin-2-one
N-[(5-amino-1,3,4-thiadiazol-2-yl)(phenyl)methyl]-3-phenyl-1H-pyrazole-4-carboxamide
1-[1,3-dioxo-2-(oxolan-2-ylmethyl)-2,3-dihydro-1H-isoindol-4-yl]-N-methyl-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]piperidine-4-carboxamide
N-[1-(1,3-benzothiazol-2-yl)piperidin-3-yl]-2-(propan-2-yloxy)acetamide
3-methyl-8-[3-(2-methylpropyl)-1,2-oxazole-5-carbonyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-[(3,4-difluorophenyl)methyl]-3-{[(1,3-dihydroxy-2-methylpropan-2-yl)amino]methyl}-3-hydroxypiperidin-2-one
1-[4-(2-methylpropyl)-3-oxo-6-(pyridin-3-ylmethoxy)-1,4-diazepan-1-yl]-4-phenylbutane-1,4-dione
N-(furan-2-ylmethyl)-N,1-dimethyl-5-{[3-(propan-2-yloxy)propyl]amino}-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide