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methyl 9-[(4-fluorophenyl)methoxy]-7-oxo-3-(1H-pyrazol-3-ylmethyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
N-[(1S,2S)-1-amino-2,3-dihydro-1H-inden-2-yl]-2-(2-oxopiperidin-1-yl)acetamide
2-{[methyl({[4-(1H-pyrazol-1-yl)phenyl]methyl})amino]methyl}quinolin-4-ol
2-(dimethylamino)-8-{[2-(thiophen-2-yl)pyrimidin-5-yl]methyl}-1,3,8-triazaspiro[4.5]dec-1-en-4-one
3-[({pyrazolo[1,5-a]pyrimidin-3-ylmethyl}amino)methyl]pyrrolidin-3-ol
(3R,9aR)-3-benzyl-8-(naphthalene-2-sulfonyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
1-[(1-ethyl-5-methyl-1H-pyrazol-4-yl)methyl]-N-[4-(1,3-thiazol-4-yl)phenyl]pyrrolidine-2-carboxamide
1-propanoyl-N-[2-(1H-pyrrol-1-yl)ethyl]piperidine-3-carboxamide
2-chloro-4-({ethyl[(1-ethyl-1H-pyrazol-4-yl)methyl]amino}methyl)phenol
3-({1,4-dimethyl-1,4,9-triazaspiro[5.5]undecan-9-yl}methyl)-7-methylquinolin-2-ol
1-[3-(3-oxopiperazin-1-yl)propyl]-3-[3-(1H-1,2,3,4-tetrazol-1-yl)phenyl]urea
(2S,4S)-4-[4-(2-methoxyphenyl)-1H-1,2,3-triazol-1-yl]pyrrolidine-2-carboxylic acid
2-[(3-cyclopropyl-1H-pyrazol-5-yl)methyl]-7-(oxan-4-yl)-2,7-diazaspiro[4.5]decan-6-one
[(5-methoxy-3-methyl-1H-indol-2-yl)methyl](methyl)(1H-pyrazol-3-ylmethyl)amine
7-[(5-methoxy-2-methyl-3-phenyl-1-benzofuran-6-yl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine
N-[2-(1H-indol-3-yl)ethyl]-2-[1-(naphthalen-2-ylmethyl)-3-oxopiperazin-2-yl]acetamide
1-[(3S,4R)-3-(dimethylamino)-4-(propan-2-yl)pyrrolidin-1-yl]-4-phenoxybutan-1-one
N-({3-[2-(4-fluorophenyl)ethoxy]phenyl}methyl)-2,3-dimethoxy-N-(pyridin-4-ylmethyl)benzamide
5,6-dimethyl-2-(2-{4-[(3-methylphenyl)sulfanyl]piperidin-1-yl}-2-oxoethyl)-2,3-dihydropyridazin-3-one
2-methyl-6-{[5-(pyrazin-2-yl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}-3H,4H,5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-one
1-(2-methylpropyl)-5-oxo-N-[(1r,4r)-4-(4H-1,2,4-triazol-4-yl)cyclohexyl]pyrrolidine-3-carboxamide
5-hydroxy-N,1,2-trimethyl-N-(quinolin-5-ylmethyl)-1H-indole-3-carboxamide
N2-benzyl-6-(2-fluorophenyl)-1,3,5-triazine-2,4-diamine
1-ethyl-4-{[3-fluoro-4-(trifluoromethyl)phenyl]methyl}piperazine-2,3-dione
(4aS,8aR)-6-[(4-acetyl-1-methyl-1H-pyrrol-2-yl)methyl]-1-(3-methylbutyl)-decahydro-1,6-naphthyridin-2-one
methyl (2S,4S)-4-(5-chloro-3-phenyl-1H-indole-2-amido)-1-[(2-methoxyphenyl)methyl]pyrrolidine-2-carboxylate
8-{[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]methyl}-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
N-(furan-2-ylmethyl)-N-[2-(morpholin-4-yl)ethyl]-3-(trimethyl-1H-pyrazol-4-yl)propanamide
2-{4-[(2-chloro-3,4-dimethoxyphenyl)methyl]-1-(2-methylpropyl)piperazin-2-yl}ethan-1-ol
9-[4-(ethylamino)pyrimidin-2-yl]-2-[2-(pyridin-3-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
7,7-dimethyl-2-(5-phenyl-1,3,4-oxadiazol-2-yl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
N-(furan-2-ylmethyl)-1-methyl-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
6-fluoro-4-[2-(3-methyl-1H-1,2,4-triazol-5-yl)pyrrolidine-1-carbonyl]-1,2-dihydroquinolin-2-one
N-(2H-1,3-benzodioxol-5-ylmethyl)-N-methyl-4-oxo-3,4-dihydroquinazoline-2-carboxamide
1-(3-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidine-1-carbonyl)cyclobutan-1-amine
2-[3-benzyl-1-(4-methoxyphenyl)-5-oxo-4,5-dihydro-1H-1,2,4-triazol-4-yl]-N-propylacetamide
1-[1-(dimethyl-1,3-thiazole-5-carbonyl)piperidin-3-yl]-4-(4-fluorophenyl)piperazine
N-{2-[1-(2-{1-[(4-methylphenyl)methyl]-3-oxopiperazin-2-yl}acetyl)piperidin-4-yl]ethyl}acetamide
5-(pyridin-3-yl)-5-{1-[2-(1,3-thiazol-4-yl)acetyl]piperidin-4-yl}-3-(thiophen-3-ylmethyl)imidazolidine-2,4-dione
1-[1-(2-methylpropyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]-4-(1H-1,2,4-triazol-1-yl)butan-1-one
1-[7-(3-chlorophenyl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-4-methylpentan-1-one
(2,1,3-benzothiadiazol-5-ylmethyl)(methyl){[5-methyl-2-(5-methylfuran-2-yl)-1,3-oxazol-4-yl]methyl}amine
N-[(3R,5S)-1-[(2-aminopyridin-3-yl)methyl]-5-(ethylcarbamoyl)pyrrolidin-3-yl]-1,3-thiazole-4-carboxamide
5-{4-[1-(2,2-dimethylpropyl)pyrrolidin-3-yl]piperidine-1-carbonyl}pyridin-2-ol
1-[3-(5-methyl-1,3,4-thiadiazol-2-yl)phenyl]-N-{[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}piperidin-4-amine
3-[1-(1H-indol-2-ylmethyl)piperidin-4-yl]-N-phenylpropanamide
4-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-(pyridin-4-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
5-{4-[1-(morpholin-4-yl)ethyl]phenyl}-1H-indazole
4-{[2-(4-chlorophenyl)-7-(methylsulfanyl)quinolin-3-yl]methyl}piperazin-2-one
2-methoxy-5-({methyl[2-(oxan-4-yl)ethyl]amino}methyl)benzoic acid