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4-(1-benzyl-1H-imidazol-2-yl)-1-(3-ethyl-5-methyl-1,2-oxazole-4-carbonyl)piperidine
(3S,4S)-4-(naphthalen-2-yl)-1-[3-(propan-2-yl)-1,2-oxazole-5-carbonyl]piperidin-3-ol
3-[(2,5-dimethoxyphenyl)methyl]-3H,4H-pyrido[4,3-d]pyrimidin-4-one
(3R,4S)-4-{[(3,5-dichloropyridin-4-yl)methyl](ethyl)amino}oxolan-3-ol
N-[(4,5-dimethyl-1H-1,3-benzodiazol-2-yl)methyl]-2-(1H-1,2,3,4-tetrazol-5-yl)acetamide
N-(but-2-yn-1-yl)-N-(furan-2-ylmethyl)-1H-imidazole-5-carboxamide
6-methyl-N4-[1-(pyrimidin-2-yl)piperidin-3-yl]pyrimidine-2,4-diamine
3-(3,5-dimethyl-1H-pyrazol-1-yl)-N-(2-methanesulfonylethyl)benzamide
N-[(4-hydroxy-1-{[(5-methyl-1,2-oxazol-3-yl)carbamoyl]methyl}azepan-4-yl)methyl]pyrrolidine-1-carboxamide
3-[({1-[1-(4-methylphenyl)cyclopropanecarbonyl]piperidin-4-yl}oxy)methyl]pyridine
3-[5-oxo-2-(thiophen-2-ylmethyl)pyrrolidin-2-yl]-N-[(4-phenyloxan-4-yl)methyl]propanamide
N-[4-(ethylsulfanyl)phenyl]-4-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carboxamide
1-[benzyl(methyl)amino]-3-[2-methoxy-5-({methyl[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]amino}methyl)phenoxy]propan-2-ol
1-[(3aS,6aR)-3-[(2-methoxyphenyl)methyl]-2-oxo-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-5-yl]-2-(furan-2-yl)ethane-1,2-dione
ethyl 1-(1-methyl-2-oxo-1,2-dihydroquinolin-4-yl)-5-({methyl[2-(1H-pyrazol-1-yl)ethyl]amino}methyl)-1H-pyrazole-4-carboxylate
4-[4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazine-1-carbonyl]piperidin-4-amine
4-(1-ethyl-1H-imidazol-2-yl)-1-{[4-(trifluoromethoxy)phenyl]methyl}piperidine
2-[4-(4-{[2-hydroxy-2-(prop-2-en-1-yl)pent-4-en-1-yl]amino}piperidin-1-yl)phenyl]-1-(4-hydroxypiperidin-1-yl)ethan-1-one
2-[(4aR,7aS)-6,6-dioxo-4-(4,4,4-trifluorobutyl)-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]-N,N-dimethylacetamide
1-{1-[3-(4-methoxyphenyl)propanoyl]piperidin-3-yl}-N-(propan-2-yl)-1H-1,2,3-triazole-4-carboxamide
6-(4-acetyl-4-phenylpiperidine-1-carbonyl)-1,3-dimethyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
2-(2-methylpropyl)-6-{thieno[3,2-d]pyrimidin-4-yl}-5H,6H,7H-pyrrolo[3,4-d]pyrimidine
(3S,4S)-1-(1,3-dimethyl-1H-pyrazole-4-carbonyl)-4-(naphthalen-2-yl)piperidin-3-ol
1-(1-acetylpiperidin-3-yl)-3-(3-chloro-2-propoxyphenyl)urea
N-{[2-(1H-imidazol-1-yl)phenyl]methyl}-7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carboxamide
2-{1-[3-(5-methylfuran-2-yl)-1H-pyrazole-5-carbonyl]pyrrolidin-2-yl}-1,3-thiazole
3-[(3R,4S)-1-(2-chloro-5-fluorobenzoyl)-4-(morpholin-4-yl)piperidin-3-yl]propan-1-ol
1-(2,4-dimethoxybenzenesulfonyl)-2-(3-methoxypropyl)piperidine
9-(5-methylpyrazine-2-carbonyl)-2-(pyridin-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
3-(3-fluoro-4-methoxybenzoyl)-1-[(1-methyl-3-phenyl-1H-pyrazol-4-yl)methyl]piperidine
4-methyl-N-(3-{[4-(pyridin-3-yl)pyrimidin-2-yl]amino}propyl)benzene-1-sulfonamide
2-(dimethyl-1,2-oxazol-4-yl)-1-{4-[2-(1H-pyrazol-1-yl)ethyl]piperidin-1-yl}ethan-1-one
1-[(2-fluorophenyl)methyl]-5-{3-[(1-methylpiperidin-4-yl)methyl]-1,2,4-oxadiazol-5-yl}piperidin-2-one
2-(3-chloro-2,4-difluorophenyl)-1-[(3R,4S)-4-hydroxy-3,4-dimethylpiperidin-1-yl]ethan-1-one
N-cycloheptyl-1-{2-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl}piperidine-3-carboxamide
1-(furan-2-yl)-2-[9-oxo-8-(pyridin-3-ylmethyl)-2,8-diazaspiro[5.5]undecan-2-yl]ethane-1,2-dione
[2-(2-{6-chloroimidazo[2,1-b][1,3]thiazol-5-yl}-1H-imidazol-1-yl)ethyl]diethylamine
1-ethyl-2-({4-[3-(propan-2-yl)-1H-pyrazol-5-yl]piperidin-1-yl}methyl)-1H-1,3-benzodiazole
1-[(1S,5R)-3-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]cyclopropane-1-carboxamide
methyl[(4-{2-[1-(quinoline-2-carbonyl)piperidin-2-yl]ethoxy}phenyl)methyl](thiophen-2-ylmethyl)amine
2-ethyl-5-(3-{[4-(2-methylpropyl)-1H-1,2,3-triazol-1-yl]methyl}piperidine-1-carbonyl)pyrimidine
1-{7-[ethoxy(phenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl}-2-(pyridin-4-ylsulfanyl)ethan-1-one
(3S,9aR)-3-benzyl-8-[(3,4-difluorophenyl)methyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
2-{2-[2-(3-methylthiophen-2-yl)-1H-imidazol-1-yl]ethyl}-6-phenyl-2,3,4,5-tetrahydropyridazin-3-one
2-(3-methoxypropyl)-8-{thieno[3,2-d]pyrimidin-4-yl}-2,8-diazaspiro[4.5]decan-3-one
3-{2-[({5-[(dimethylamino)methyl]furan-2-yl}methyl)sulfanyl]ethyl}-1-(1H-indazol-5-yl)urea
2-(pyrrolidin-3-ylmethyl)-2,3-dihydro-1,2-benzothiazol-3-one
1-[3-(2-fluorophenyl)pyrrolidin-1-yl]-3-[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]propan-1-one
5-[4-(4-methoxyphenyl)-3,3-dimethylpiperazine-1-carbonyl]-4-methyl-1,3-thiazol-2-amine
1-(4-{2-[(2-chlorophenyl)methyl]morpholin-4-yl}-4-oxobutyl)pyrrolidin-2-one