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N-[3-(3-methoxyphenyl)phenyl]-1-(1,2-oxazol-3-ylmethyl)piperidine-4-carboxamide
{1-[6-(4-fluorophenyl)pyridazin-3-yl]-3-(prop-2-en-1-yl)piperidin-3-yl}methanol
7-cyclohexyl-2-[2-(methylsulfanyl)acetyl]-2,7-diazaspiro[4.5]decan-6-one
3-(1-methyl-1H-imidazol-2-yl)-1-(2-propoxyethyl)piperidine
3-(methylsulfanyl)-5-[3-(1H-pyrazol-1-yl)phenyl]-1H-1,2,4-triazole
5-[4-(4-fluorophenyl)-4-oxobutanoyl]-1-(2-methylpropyl)-N-(pyridin-3-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
(1S,6R)-9-{6-methyl-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-yl}-3,9-diazabicyclo[4.2.1]nonan-4-one
2-methoxy-2-methyl-N-({2-[3-(trifluoromethyl)phenoxy]pyridin-3-yl}methyl)propanamide
N-(2-{1-[2-(dimethylamino)ethyl]-5-oxopyrrolidin-2-yl}ethyl)-4,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
ethyl 5-(2,3-dihydro-1-benzofuran-5-ylmethyl)-1-(2-hydroxyethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
N-{2-[7-(naphthalen-2-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]ethyl}oxane-4-carboxamide
N-[(3,5-dimethoxyphenyl)methyl]-1-(4,7-dimethylquinazolin-2-yl)piperidine-4-carboxamide
{[1-(2,4-difluorophenyl)-3-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]amine
N-{1-[1-(3-acetamidopropanoyl)piperidin-4-yl]-2-(2-methylphenyl)ethyl}-N-methyl-2-(1H-pyrazol-1-yl)acetamide
7-[ethoxy(phenyl)methyl]-4-(4-methyl-1,2,3-thiadiazole-5-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-{[2-(2-benzamidophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-5-(methoxymethyl)thiophene-2-carboxamide
(3S,4R)-4-phenyl-1-[2-(1H-1,2,3,4-tetrazol-5-yl)benzoyl]pyrrolidine-3-carboxylic acid
N-{[1-(thiophene-3-carbonyl)piperidin-3-yl]methyl}naphthalene-1-carboxamide
4-[2-methyl-5-(1,2-oxazol-5-yl)benzenesulfonyl]-2-(trifluoromethyl)morpholine
(1R,7S)-3-cycloheptyl-N-methyl-4-oxo-N-[2-(1H-pyrazol-4-yl)ethyl]-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
5-(3-fluorophenyl)-N-[3-(propan-2-yloxy)propyl]-1,2,4-triazin-3-amine
4-[4-(3-hydroxy-3-methylbutyl)benzoyl]morpholine-2-carboxamide
1-(3-phenylpropyl)-N-{[3-(trifluoromethoxy)phenyl]methyl}-1H-1,2,3-triazole-4-carboxamide
4-{2-[3-(thiophen-3-yl)-1,2,4-oxadiazol-5-yl]ethyl}morpholine
2-ethyl-4-methyl-N-[1-(3-phenylpropyl)piperidin-3-yl]-1,3-oxazole-5-carboxamide
2-(4-{[7-methyl-2-(3-methylphenyl)quinolin-3-yl]methyl}morpholin-2-yl)ethan-1-ol
4-{4-[3-(pyrrolidine-1-carbonyl)piperidin-1-yl]piperidine-1-carbonyl}pyridine
2-[(dimethyl-1,2-oxazol-4-yl)methyl]-5-(dimethylamino)-2,3-dihydropyridazin-3-one
N-[(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)methyl]-1,9-dioxaspiro[5.5]undecan-4-amine
N-(4-{5H,6H,7H,8H-imidazo[1,5-a]pyrazine-7-carbonyl}-3-methylphenyl)acetamide
5-(2,6-difluorophenoxymethyl)-N-[2-(3-methoxyphenyl)ethyl]-1,2-oxazole-3-carboxamide
N-{[3-(cycloheptyloxy)-4-methoxyphenyl]methyl}-N-cyclopropyl-2,2-dimethyloxane-4-carboxamide
6-[3-(2-methoxybenzoyl)piperidine-1-carbonyl]-2,2-dimethyl-3,4-dihydro-2H-pyran-4-one
2-(2-methoxyphenoxy)-N-{[1-(1,2-oxazole-3-carbonyl)piperidin-3-yl]methyl}acetamide
3-[1-(1-ethyl-1H-pyrazole-3-carbonyl)piperidin-3-yl]benzoic acid
N-(3-{[(4-chlorophenyl)methyl]sulfanyl}propyl)-2-(2-oxo-1,2-dihydropyrimidin-1-yl)acetamide
N-{[2-(1H-imidazol-1-yl)pyridin-3-yl]methyl}-3-(1H-pyrazol-1-yl)benzamide
4-{5-[(2,4-difluorophenyl)methyl]-3-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazol-1-yl}-1-methylpiperidine
ethyl 2-[4-(4-fluorobenzenesulfonyl)-1-(pyridin-4-ylmethyl)piperidin-4-yl]acetate
{[2-(2-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(ethyl)(2-methylprop-2-en-1-yl)amine
N-{1-[1-(4-chlorobenzoyl)piperidin-4-yl]-2-(3-methoxyphenyl)ethyl}-N,3-dimethylbutanamide
3-{[(3-{1-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl}phenyl)methyl]amino}propan-1-ol
2-[(4-ethylcyclohexyl)formamido]-N-[(1-methylpyrrolidin-3-yl)methyl]acetamide
(5S,9aS,9bS)-2-[(4-methoxyphenyl)methyl]-5-(5-methylfuran-2-yl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
1-(1-{[1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}piperidin-3-yl)-2-phenylethan-1-one
N-[2-(2-chloro-6-methylphenoxy)ethyl]cyclopentanamine
(3R,4R)-4-(2-ethyl-4-methyl-1H-imidazol-5-yl)-N-(hexahydro-1H-pyrrolizin-7a-ylmethyl)-1-methylpyrrolidine-3-carboxamide
(2R,3S,6R)-3-phenyl-5-(2-propyl-1,3-thiazole-4-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
N-methyl-5-{[(2-methyl-1,3-benzothiazol-5-yl)oxy]methyl}-N-(oxolan-3-yl)-1,2-oxazole-3-carboxamide
3-(morpholin-4-yl)-N-[1-(2-phenylethyl)piperidin-3-yl]propanamide