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3-(1-methyl-1H-pyrazol-4-yl)-1-(2-{[(2-methylphenyl)methyl]sulfanyl}ethyl)urea
5-{3-oxo-2-[2-(pyridin-3-yl)ethyl]-2,9-diazaspiro[5.5]undecane-9-carbonyl}pyridine-2-carbonitrile
(2R,3R,6R)-5-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]-3-(3-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
(4aS,8aR)-6-(5-methyl-1,3-oxazole-4-carbonyl)-1-[2-(thiophen-2-yl)ethyl]-decahydro-1,6-naphthyridin-2-one
N-benzyl-1-cyclopropyl-6-oxo-N-(2-phenylethyl)piperidine-3-carboxamide
2-phenyl-1-[4-(quinolin-5-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl]ethan-1-ol
(3S)-2-[3-(5-amino-1H-1,2,4-triazol-3-yl)propanoyl]-N-tert-butyl-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
3-(4-methoxyphenyl)-1-[(1R,5R)-6-(3-methylbut-2-en-1-yl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]propan-1-one
1-{2-[(1S,5R)-3-(2,3-dihydro-1H-inden-2-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-oxoethyl}-3,3-dimethylurea
2,8-dimethyl-N-[1-(pyrazin-2-yl)piperidin-4-yl]quinoline-4-carboxamide
5-methyl-N-[2-methyl-2-(4-methylpiperazin-1-yl)propyl]pyrimidin-2-amine
4-{4-[6-(methylamino)-1H-pyrrolo[2,3-b]pyridin-4-yl]phenyl}-4-oxobutanoic acid
ethyl 4-{[(3aS,6aR)-3-cyclopentyl-2-oxo-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-5-yl]methyl}-1H-pyrazole-3-carboxylate
5-(furan-2-yl)-1-[(2-methoxyphenyl)methyl]-1H,4H-pyrazolo[3,4-d]imidazole
5-{[(1S,5R)-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]methyl}-1,2,4-oxadiazole-3-carboxamide
N-[2-methoxy-1-(pyridin-2-yl)ethyl]-3-[3-(2-methoxyphenyl)-1,2,4-oxadiazol-5-yl]-N-methylpropanamide
4-[(4-fluorophenyl)methyl]-1-(2-methylpyridine-3-carbonyl)-3-(propan-2-yl)-1,4-diazepan-5-one
1-(4-chloro-3-{2-ethyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}phenyl)-1H-pyrazole
3-(3-methoxyphenyl)-5-{8-methyl-octahydro-1H-pyrazino[1,2-a]piperazine-2-carbonyl}-1H-pyrazole
5-fluoro-N-methyl-N-[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]quinazolin-4-amine
3-chloro-N-{[3-(cyclopentyloxy)phenyl]methyl}-N-[(3S)-2-oxoazepan-3-yl]benzamide
N-[(4-chlorophenyl)methyl]-N-(3-hydroxypropyl)-2-[methyl(piperidin-4-yl)amino]acetamide
N-[2-(3-methoxyphenyl)-1-{1-[(2E)-3-(thiophen-2-yl)prop-2-enoyl]piperidin-4-yl}ethyl]-N-methyl-3-(methylsulfanyl)propanamide
1-{1-[(3-methylphenyl)methyl]piperidin-4-yl}-N-(pyridin-3-ylmethyl)piperidine-3-carboxamide
2-{1-[(2-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-[2-(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)ethyl]acetamide
N-[2-(7-{[3-(2-hydroxyethoxy)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)ethyl]-4-methylbenzamide
2-{1-[(2-ethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-methyl-N-(1,3-thiazol-2-ylmethyl)acetamide
2-{4-[5-(1H-imidazol-1-ylmethyl)pyridin-2-yl]phenyl}-2-methylpropanenitrile
N-cyclopropyl-2-(1,3-dimethyl-2,5-dioxoimidazolidin-4-yl)-N-(1H-indol-5-ylmethyl)acetamide
5-methyl-N4-{[1-(1H-pyrazol-1-ylmethyl)cyclopropyl]methyl}pyrimidine-2,4-diamine
2-(2-acetyl-4,5-dimethoxyphenyl)-1-[(3S,4S)-3,4-dihydroxy-4-methylpiperidin-1-yl]ethan-1-one
N-[(2,6-dimethoxyphenyl)methyl]-5-{1-[(2-fluorophenyl)methyl]-1H-pyrazol-3-yl}-4-methyl-1,3-thiazol-2-amine
4-{2-methyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-5-carbonyl}-1,2-dihydroquinolin-2-one
5-(pyrrolidine-1-carbonyl)-N-[(2,3,5-trimethyl-1H-indol-7-yl)methyl]pyridin-2-amine
(4S)-3-{2-[4-(3-methylphenoxy)piperidin-1-yl]-2-oxoethyl}-4-(propan-2-yl)-1,3-oxazolidin-2-one
N-cyclobutyl-3-[(2-acetamidoethyl)sulfamoyl]benzamide
5-{[2-(2,2-dimethyloxan-4-yl)-1H-imidazol-1-yl]methyl}-N,N-dimethylfuran-2-carboxamide
N-methyl-N-(1,2-oxazol-5-ylmethyl)-2-(pyrrolidin-3-yl)benzamide
1-{2-methyl-5-[4-(oxolan-2-ylmethyl)piperazine-1-carbonyl]phenyl}imidazolidin-2-one
1-{[4-(trifluoromethoxy)phenyl]methyl}azepan-4-amine
N-({5-methanesulfonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-4-methylpiperazine-1-carboxamide
N-[1-(1,5-dimethyl-1H-pyrazol-4-yl)ethyl]-2-(4-fluorophenyl)imidazo[1,2-a]pyridine-6-carboxamide
3-[(1-propyl-1H-imidazol-2-yl)methyl]-3,9-diazaspiro[5.5]undecane
4-(hydroxymethyl)-1-{[7-methyl-2-(3-methylphenyl)quinolin-3-yl]methyl}piperidin-4-ol
2,6-difluoro-3-methoxy-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]benzamide
N-[1-(dimethylamino)propan-2-yl]-6-(2,5-dimethylfuran-3-yl)-7-methyl-8-oxo-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
N-ethyl-2-(4-{2-[4-(methylsulfanyl)phenyl]acetyl}piperazin-1-yl)acetamide
N-(2-{5-[(2-chloroprop-2-en-1-yl)sulfanyl]-4-(4-fluorophenyl)-4H-1,2,4-triazol-3-yl}ethyl)acetamide
8-cyclohexyl-3-{3-[3-(dimethylamino)pyrrolidin-1-yl]propyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-(oxan-2-ylmethyl)-2-{[4-(pyrimidin-2-yl)piperazin-1-yl]methyl}-1,3-oxazole-4-carboxamide