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1-[2-(2-{8-oxatricyclo[7.4.0.02,7]trideca-1(9),2(7),3,5,10,12-hexaen-6-yl}-1H-imidazol-1-yl)ethyl]piperidin-4-ol
2-(adamantan-1-yl)-N-methyl-N-(quinolin-3-ylmethyl)acetamide
2-methoxy-N-(2-methyl-1-{7-[(2-phenyl-1,3-thiazol-5-yl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}propyl)acetamide
2-[(4-chlorophenyl)methyl]-N-methyl-N-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]-1,3-benzoxazole-5-carboxamide
2-(3-benzyl-1-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-N-(pyridin-2-ylmethyl)acetamide
2-({6-[2-(methylsulfanyl)phenyl]pyrimidin-4-yl}amino)ethan-1-ol
1-(2H-1,3-benzodioxol-5-ylmethyl)-4-[(2-ethylpyrimidin-4-yl)methyl]piperazin-2-one
2-cyclopropyl-N-[1-(4-fluorophenyl)-2-methylpropan-2-yl]pyrimidine-5-carboxamide
5-methyl-3-[(1E)-pent-1-en-1-yl]-2-(4H-1,2,4-triazol-4-yl)pyridine
3-[(2-fluorophenyl)methyl]-5-{[2-(4-fluorophenyl)pyrrolidin-1-yl]methyl}-1,2,4-oxadiazole
2-(4,6-dimethyl-1-benzofuran-3-yl)-N-(5-oxo-1-phenylpyrrolidin-3-yl)acetamide
N-[2-(4-{[4-(pyridin-2-yl)phenyl]methyl}morpholin-2-yl)ethyl]acetamide
2-oxo-N-[(4-phenyloxan-4-yl)methyl]-2,3-dihydro-1H-imidazole-4-carboxamide
1-(dimethyl-1,2-oxazol-4-yl)-3-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-3-(propan-2-yl)urea
5-({methyl[(3-{2-[4-(naphthalene-2-sulfonyl)piperazin-1-yl]ethoxy}phenyl)methyl]amino}methyl)pyrrolidin-2-one
2-[3-(1H-pyrazol-1-ylmethyl)benzoyl]-1,2,3,4-tetrahydroisoquinoline
3-[(1H-1,3-benzodiazol-2-ylmethyl)sulfamoyl]-N-propylbenzamide
N-{1-[1-(6-chloro-1,3-benzothiazol-2-yl)piperidin-4-yl]pyrrolidin-3-yl}acetamide
(2R,3R,6R)-3-(4-methoxyphenyl)-5-(6-methoxypyrimidin-4-yl)-1,5-diazatricyclo[5.2.2.02,6]undecane
1-(2H-1,3-benzodioxol-5-ylmethyl)-4-(5-fluoro-4-hydroxypyrimidin-2-yl)piperazin-2-one
4-{1-[(5-tert-butyl-1,2,4-oxadiazol-3-yl)methyl]piperidin-4-yl}-6-(pyrrolidin-1-yl)pyrimidine
9-[3-(2-ethyl-1H-imidazol-1-yl)propanoyl]-2-(prop-2-en-1-yl)-2,9-diazaspiro[5.5]undecan-3-one
2-(dimethylamino)-1-[4-(1-methyl-1H-imidazol-2-yl)piperidin-1-yl]-2-(3-methylphenyl)ethan-1-one
2-(2-chlorophenyl)-3-methyl-N-[(4-methyl-1H-imidazol-2-yl)methyl]-3H-imidazo[4,5-b]pyridine-6-carboxamide
7-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-3-(2-phenylethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine
N-[(3S,4R)-4-(5-methylfuran-2-yl)-1-(oxan-4-yl)pyrrolidin-3-yl]acetamide
1-(3-methylphenyl)-3-(2-methylpropyl)-5-(1H-1,2,4-triazol-1-ylmethyl)-1H-1,2,4-triazole
4-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-[3-(2-oxopyrrolidin-1-yl)propyl]benzamide
N-[(7S,8aS)-2-methyl-octahydropyrrolo[1,2-a]piperazin-7-yl]-2-(3-methyl-2-oxo-1,2,3,4-tetrahydroquinazolin-1-yl)acetamide
2-[2-(4-fluorophenyl)-2-(piperidin-1-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
1-{4-[(3-chlorophenyl)methyl]piperazin-1-yl}-2-hydroxy-4-(methylsulfanyl)butan-1-one
N-methyl-N-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]-3-(trimethyl-1H-pyrazol-4-yl)propanamide
4-{5-[1-(2H-1,3-benzodioxol-5-yl)propan-2-yl]-1H,4H-pyrazolo[3,4-d]imidazol-1-yl}-1-methylpiperidine
1-[(3R,5R)-3-(hydroxymethyl)-5-(morpholin-4-ylmethyl)piperidin-1-yl]-3-(1H-1,2,3,4-tetrazol-1-yl)propan-1-one
[(2S)-1-{[2-(3,5-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}pyrrolidin-2-yl]methanol
N-{[5-(4-methanesulfonylphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-(2-methoxyphenoxy)acetamide
N,N-dimethyl-7-[4-(trifluoromethyl)benzamido]-1,2,3,4-tetrahydroisoquinoline-2-carboxamide
1-(4-methylphenyl)-4-[2-(4-propanoylphenoxy)acetyl]piperazin-2-one
1-(3-phenylpropyl)-4-{trimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-1,4-diazepane
{[2-(azocan-1-yl)pyridin-3-yl]methyl}[(trimethylpyrazin-2-yl)methyl]amine
1-methyl-N-({1-[(2-methyl-1H-imidazol-1-yl)methyl]cyclopropyl}methyl)piperidine-2-carboxamide
4-(1-{[1-phenyl-3-(pyridin-4-yl)-1H-pyrazol-4-yl]methyl}azetidin-3-yl)morpholine
3-(oxan-4-yl)-7-(trifluoromethyl)-3,4-dihydroquinazolin-4-one
N-cyclopropyl-2-[(3,4-dimethoxyphenyl)methyl]-N-ethyl-1,3-benzoxazole-6-carboxamide
N-[2-(pyridin-4-yl)ethyl]-5-[(quinolin-6-yloxy)methyl]-1,2-oxazole-3-carboxamide
4-(4-cyclopentylpyrimidin-2-yl)-1-ethyl-3-methylpiperazin-2-one
1-cycloheptyl-6-oxo-N-(quinolin-6-ylmethyl)piperidine-3-carboxamide
2-(4-hydroxyphenyl)-1-[(3R,4S)-3-(3-hydroxypropyl)-4-(4-methylpiperazin-1-yl)piperidin-1-yl]ethan-1-one
methyl[(4-methyl-1,2,5-oxadiazol-3-yl)methyl][(3-{[1-(thiophene-2-carbonyl)piperidin-4-yl]oxy}phenyl)methyl]amine
5-{1-[5-(4,5-dimethylfuran-2-yl)-4-phenyl-1H-imidazol-1-yl]ethyl}-1H-1,2,3,4-tetrazole