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N-({7-[(4-ethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)benzenesulfonamide
N-(furan-2-ylmethyl)-2-oxo-1-phenyl-N-(pyridin-2-ylmethyl)pyrrolidine-3-carboxamide
1-[3-(2-hydroxyethyl)-4-methylpiperazin-1-yl]-3-{imidazo[1,2-a]pyridin-2-yl}propan-1-one
4-[3-(pyridin-4-yl)propyl]-11-{[(3,4,5-trifluorophenyl)methyl]amino}-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
2-[3-(dimethylamino)pyrrolidin-1-yl]-N-{5-[2-(3-methylphenoxy)ethyl]-1,3,4-thiadiazol-2-yl}acetamide
N-[(1-ethylpyrrolidin-2-yl)methyl]-3-[1-(2-methylpyridine-3-carbonyl)piperidin-4-yl]propanamide
N-{2-[(3-methylpyridin-4-yl)amino]ethyl}-3,4-dihydro-2H-1-benzopyran-3-carboxamide
N-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-{[4-(methylsulfanyl)phenyl]methyl}piperidin-3-amine
(2S)-2-hydroxy-4-[5-(1-methyl-1H-imidazol-2-yl)-4-phenyl-1H-imidazol-1-yl]butanoic acid
6-[3-(2,5-dimethoxyphenyl)pyrrolidine-1-carbonyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
9-[2-(dimethylamino)-2-(4-methylphenyl)acetyl]-3,9-diazaspiro[5.5]undecane-2,4-dione
5-{4-hydroxy-1-[(4-methylphenyl)methyl]piperidin-4-yl}-N-(oxolan-2-ylmethyl)-1-benzofuran-2-carboxamide
3-({3-[4-(methylsulfanyl)benzoyl]piperidin-1-yl}methyl)pyridine
4-(1,3-dimethyl-1H-pyrazole-5-carbonyl)-7-(phenoxathiin-4-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
3-(azocan-1-yl)-N-[2-(4-hydroxypiperidin-1-yl)ethyl]propanamide
1-[4-(methoxymethyl)piperidin-1-yl]-3-[5-(4-phenylbutyl)-1,3,4-oxadiazol-2-yl]propan-1-one
6-(3-{5-[(dimethylamino)methyl]-4-methyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)pyridine-3-carboxylic acid
1-{[(4S)-4-(prop-1-en-2-yl)cyclohex-1-en-1-yl]methyl}-4-[3-(pyrrolidine-1-carbonyl)phenoxy]piperidine
2-{4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]benzoyl}-2,3-dihydro-1H-isoindole
(3aR,6aS)-2-[(3-fluoro-2-methoxyphenyl)methyl]-5-methyl-octahydropyrrolo[3,4-c]pyrrole
1-(2-phenylmorpholine-4-carbonyl)isoquinoline
(2R)-2-[(3-propyl-1H-pyrazol-5-yl)formamido]propanamide
5-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl}-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxylic acid
5-(2-{[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]amino}ethyl)-1-[(4-methylphenyl)methyl]pyrrolidin-2-one
3-{[7-(hydroxymethyl)-9-(pyridin-3-ylmethyl)-3,9-diazaspiro[5.5]undecan-3-yl]methyl}phenol
1-(2-methoxyethyl)-6-oxo-N-[2-(4-phenyl-1,3-thiazol-2-yl)ethyl]piperidine-3-carboxamide
6-{[cyclohexyl(methyl)amino]methyl}-2-oxo-N-{[3-(trifluoromethyl)phenyl]methyl}-1,2-dihydropyridine-3-carboxamide
1-[2-amino-4-(2,5-dihydro-1H-pyrrol-1-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl]-2-(1-methyl-1H-pyrrol-3-yl)ethan-1-one
5-(4-{2-chloro-5H,6H,7H-cyclopenta[b]pyridine-3-carbonyl}piperazin-1-yl)-2-methyl-2,3-dihydropyridazin-3-one
N-[3-(3-fluorophenyl)phenyl]-1-{[5-(2-methylpropyl)-1H-pyrazol-3-yl]methyl}piperidine-4-carboxamide
3-[({[3-(2-methylpropyl)-1,2-oxazol-5-yl]methyl}amino)methyl]pyrrolidin-3-ol
1-{[2-methyl-4-(1H-pyrazol-1-yl)phenyl]methyl}-3-(piperidin-1-ylmethyl)pyrrolidin-3-ol
1-benzyl-3-(2-methoxyethyl)-8-(pyridin-4-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-(2-amino-1,3-thiazol-4-yl)-N-{[1-(4-methoxyphenyl)cyclopentyl]methyl}propanamide
3-(3-{[(3-methoxy-2,2-dimethylpropyl)carbamoyl]amino}phenyl)-N,N-dimethylpropanamide
2-(3-{1-[3-(dimethylamino)propyl]-1H-imidazol-2-yl}piperidin-1-yl)pyrimidin-4-amine
3-hydroxy-1-[(3-methoxyphenyl)methyl]-3-[({pyrazolo[1,5-a]pyridin-3-ylmethyl}amino)methyl]piperidin-2-one
N-{[3-fluoro-5-(trifluoromethyl)phenyl]methyl}-5-[(3-hydroxypiperidin-1-yl)methyl]-1,2-oxazole-3-carboxamide
6-[(1-phenyl-1H-pyrazol-4-yl)methyl]-N-[2-(pyridin-2-yl)ethyl]-6-azaspiro[2.5]octane-1-carboxamide
1-(4-{[4-(4-chlorobenzoyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl]methyl}piperazin-1-yl)ethan-1-one
(3R,4S)-1-{imidazo[2,1-b][1,3]thiazole-6-carbonyl}-4-(3-methoxyphenyl)pyrrolidin-3-amine
1-[(4-methoxyphenyl)methyl]-4-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidine
(3S,4R)-1-(2-methanesulfonylethyl)-4-(pyridin-4-yl)pyrrolidine-3-carboxylic acid
(1R,3S)-7-[2-(2-ethylphenoxy)ethyl]-7-azaspiro[3.5]nonane-1,3-diol
1-(3-chloro-2-propoxyphenyl)-3-[1-(5-methyl-1H-1,2,4-triazol-3-yl)ethyl]urea
ethyl 1-(3-methylbutyl)-5-[2-(1H-pyrazol-1-yl)benzoyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
N-cyclopropyl-5-[1-(3-methylbutyl)-1H-pyrazol-4-yl]thiophene-2-carboxamide
4-[(1S,5R)-3-methyl-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]benzene-1-sulfonamide
2-[5-(2-ethylpyridin-4-yl)-3-methyl-1H-1,2,4-triazol-1-yl]-6-methylpyridine
2-cyclopentyl-9-[(3-methylpyridin-2-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one