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N-[2-(6-methylpyridin-2-yl)ethyl]-N'-[2-(methylsulfanyl)phenyl]butanediamide
3-{2-ethyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}-1,4,6-trimethyl-1,2-dihydropyridin-2-one
methyl 3-[({1-[2-(2-methoxyphenyl)ethyl]piperidin-3-yl}methyl)(methyl)carbamoyl]propanoate
5-ethyl-N-{[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl}-N,2,3-trimethylpyrazolo[1,5-a]pyrimidin-7-amine
4-[1-(2-fluorophenyl)piperidin-4-yl]-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
1-[2-(2-ethyl-1H-imidazol-1-yl)ethyl]-2-oxo-3-[2-(pyridin-2-yl)ethyl]-1H,2H,3H-imidazo[4,5-b]pyridine-6-carboxylic acid
6-(2-aminoethyl)-2-methyl-N-[4-(pyrrolidin-1-yl)butyl]pyrimidin-4-amine
3-{2-[(4-ethyl-5-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}-1-(1-methyl-1H-indazol-6-yl)urea
N-[(2,4-dimethoxyphenyl)methyl]-3-{1-[2-(1H-pyrazol-1-yl)acetyl]piperidin-3-yl}propanamide
6-{3-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyridine-2-carboxylic acid
8-[2-(dimethyl-1,2-oxazol-4-yl)acetyl]-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
4-(2-methyl-2-{1-phenyl-1H,4H-pyrazolo[3,4-d]imidazol-5-yl}propyl)morpholine
1-benzyl-N,N-dimethyl-5-{[2-(4-phenylpiperidin-1-yl)ethyl]amino}-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
N-[(1-ethyl-1H-imidazol-2-yl)methyl]-N-methyl-5-[4-(1H-1,2,4-triazol-1-yl)phenoxymethyl]-1,2-oxazole-3-carboxamide
4-[3-(2,5-dimethoxyphenyl)pyrrolidine-1-carbonyl]benzonitrile
5-oxo-1-(pyridin-2-ylmethyl)-N-{2-[2-(thiophen-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]ethyl}pyrrolidine-3-carboxamide
N-[2-(benzyloxy)ethyl]-1,1-dioxo-1λ6-thiolane-3-carboxamide
N-[(2-chloropyridin-3-yl)methyl]-4-(2,4-dioxoimidazolidin-1-yl)-N-methylbenzamide
1-methyl-4-[2-(methylamino)pyridine-3-carbonyl]piperazin-2-one
ethyl 4-({4-[3-(1H-indol-3-yl)propanoyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}methyl)piperazine-1-carboxylate
(2R,3R)-3-amino-1'-(1,3-benzothiazol-2-yl)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
N-(2-{1-[2-(dimethylamino)ethyl]-5-oxopyrrolidin-2-yl}ethyl)-1-methyl-1H-indole-4-carboxamide
5-acetyl-2,4-dimethyl-N-[2-(4-methylmorpholin-2-yl)ethyl]-1H-pyrrole-3-carboxamide
6-{[3-(butan-2-yloxy)phenyl]methyl}-2,5-dioxo-1,2,5,6-tetrahydro-1,6-naphthyridine-3-carbonitrile
1-(2-methoxy-4-{[(thiophen-3-ylmethyl)amino]methyl}phenoxy)-3-(morpholin-4-yl)propan-2-ol
ethyl 3-[(3-methoxyphenyl)methyl]-1-[3-(methylsulfanyl)propanoyl]piperidine-3-carboxylate
N-methyl-N-{2-[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]ethyl}-2-propyl-1,3-thiazole-4-carboxamide
N-[2-(2-methyl-1H-indol-1-yl)ethyl]-3-(pyridin-2-yl)-1H-pyrazole-5-carboxamide
4-{4-phenyl-1-[(1-propyl-1H-pyrazol-4-yl)methyl]-1H-imidazol-5-yl}benzonitrile
1-(4-{4-[1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]piperazin-1-yl}phenyl)ethan-1-one
3-(2-amino-1,3-thiazol-4-yl)-1-[4-(2,3-dihydro-1H-inden-2-yl)-1,4-diazepan-1-yl]propan-1-one
2-[(4aS,8aR)-6-butyl-4a-(hydroxymethyl)-decahydro-1,6-naphthyridin-1-yl]-N-(1-methyl-1H-pyrazol-4-yl)acetamide
2-(dimethylamino)-N-[5-oxo-1-(2-phenylethyl)pyrrolidin-3-yl]acetamide
3-[1-(1-ethyl-3-methyl-1H-pyrazole-5-carbonyl)piperidin-3-yl]-1-[4-(pyridin-2-yl)piperazin-1-yl]propan-1-one
6-[(2E)-3-(3,4-difluorophenyl)prop-2-enoyl]-N-[3-(pyridin-4-yl)propyl]-6-azaspiro[2.5]octane-1-carboxamide
5-methyl-1-(4-methylphenyl)-4-{4-oxo-4H-pyrido[1,2-a]pyrimidine-3-carbonyl}piperazin-2-one
N-methyl-N-[(3-phenyl-1H-pyrazol-5-yl)methyl]-1-(propan-2-yl)-1H-pyrazole-4-carboxamide
2-(cyclohex-1-en-1-yl)-N-({5-methyl-2-[2-(2-phenylacetamido)phenyl]-1,3-oxazol-4-yl}methyl)acetamide
1-[(4aS,8aR)-1-(3-aminopropyl)-2-oxo-decahydro-1,6-naphthyridine-6-carbonyl]cyclopropane-1-carbonitrile
(3S,4S)-4-propyl-1-{[6-(trifluoromethyl)pyridin-3-yl]methyl}pyrrolidine-3-carboxylic acid
4-{3-[(3aR,7aS)-5-methyl-2,3,3a,4,7,7a-hexahydro-1H-isoindole-2-carbonyl]phenyl}-2-methylbutan-2-ol
methyl({[5-(oxan-2-yl)thiophen-2-yl]methyl}){[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl}amine
3-{[3-(2-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-(3-hydroxypropyl)-N-(pyridin-3-ylmethyl)-1H-1,2,3-triazole-5-carboxamide
N-[(5-chloro-1H-indol-2-yl)methyl]-1-[3-(morpholin-4-yl)propyl]-6-oxopiperidine-3-carboxamide
2-(3-{[(1R,5R)-3-cyclobutanecarbonyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}phenoxy)ethan-1-ol
2-(5-{[4-(2,6-dimethylpyridin-4-yl)piperazin-1-yl]methyl}-1,2,4-oxadiazol-3-yl)pyrazine
4-methyl-N-{4-[(2-phenylethyl)carbamoyl]phenyl}-1,4-diazepane-1-carboxamide
[2-(dimethylamino)-2-(thiophen-2-yl)ethyl]({[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl})amine
N-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]methyl}-N-[3-(dimethylamino)propyl]-3-(1H-pyrazol-1-yl)propanamide