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6-[4-(6-cyclopropylpyrimidin-4-yl)piperazin-1-yl]-9H-purine
4-ethyl-3-[1-(1H-indole-2-carbonyl)piperidin-3-yl]-1-methyl-4,5-dihydro-1H-1,2,4-triazol-5-one
methyl[2-(2-methyl-1H-imidazol-1-yl)ethyl]{[5-(1H-pyrazol-3-yl)furan-2-yl]methyl}amine
2-[4-(2-fluorophenyl)piperazin-1-yl]-6-(2-methoxyphenyl)-N-[2-(morpholin-4-yl)ethyl]pyridine-3-carboxamide
N-(cyclohexylmethyl)-2-{2-[(dimethylamino)methyl]-4-phenylphenoxy}acetamide
N-[(7S,8aS)-2-methyl-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-2-oxo-1,2-dihydroquinoline-3-carboxamide
1-(4,7-dimethylquinazolin-2-yl)-N-methyl-N-[2-(oxan-2-yl)ethyl]piperidine-3-carboxamide
N-[2-(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)ethyl]-3-(1H-pyrazol-1-yl)benzamide
N-[2-(diethylamino)ethyl]-N-methyl-5-[2-(methylsulfanyl)phenoxymethyl]-1,2-oxazole-3-carboxamide
N,1-dimethyl-N-[3-(1-methyl-1H-pyrazol-4-yl)propyl]-1H-pyrazolo[1,5-a]imidazole-7-carboxamide
[(5-{[4-(ethoxymethyl)piperidin-1-yl]methyl}thiophen-3-yl)methyl]dimethylamine
3-{[1-(3,5-dimethylbenzoyl)pyrrolidin-3-yl]methyl}benzoic acid
N-[(2,5-dimethylphenyl)(pyridin-3-yl)methyl]imidazo[1,2-a]pyridine-6-carboxamide
N-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-1-(furan-2-ylmethyl)-N-methylpiperidine-3-carboxamide
1-{[1-(2-fluorophenyl)-1H-pyrazol-4-yl]methyl}-4-(1,2,4-oxadiazol-3-yl)piperidine
N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-2,4-dimethyl-1,3-thiazole-5-carboxamide
4-phenyl-N-(3-{4-[(pyridin-3-ylmethyl)amino]piperidin-1-yl}phenyl)butanamide
2-(3,6,7-trimethyl-1-benzofuran-2-carbonyl)-octahydropyrrolo[1,2-a]piperazine
1'-[1-ethyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]-3,4-dihydrospiro[1-benzopyran-2,3'-pyrrolidine]-4-one
2-(3,4-dimethylphenoxy)-1-[(3R,4R)-3-(hydroxymethyl)-4-(piperidin-1-ylmethyl)pyrrolidin-1-yl]ethan-1-one
N-[(5-tert-butyl-1,2,4-oxadiazol-3-yl)methyl]-N-(pyridin-3-ylmethyl)-1-azabicyclo[2.2.2]octan-3-amine
N3,N3-diethyl-N1-(2-methyl-1-benzofuran-5-yl)piperidine-1,3-dicarboxamide
1-(4-cyclohexylphenyl)-3-[2-(1H-imidazol-4-yl)ethyl]urea
N-methyl-6-(1-methyl-1H-imidazol-2-yl)-N-[(3-methylthiophen-2-yl)methyl]pyridazin-3-amine
N-[(5-chloro-2-propoxyphenyl)methyl]-2-methyl-[1,3]oxazolo[5,4-d]pyrimidin-7-amine
2-[(2-chlorophenyl)methyl]-4-(2,5-dimethylbenzoyl)morpholine
1-(4-methyl-1,3-thiazol-2-yl)-3-(piperidin-1-ylmethyl)piperidine
2-hydroxy-1-{2-[(4-methoxyphenyl)methyl]-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-4-(methylsulfanyl)butan-1-one
1-[3-(4-methyl-2-phenylpiperazine-1-carbonyl)phenyl]imidazolidin-2-one
methyl (2R,4S)-4-hydroxy-1-[3-(2-methylphenoxy)propanoyl]piperidine-2-carboxylate
N-[(3S,4R)-4-ethoxyoxolan-3-yl]-6-methylpyrazolo[1,5-a]pyrimidine-3-carboxamide
2-(dimethylamino)-N-({2-methoxy-5-oxo-6-[2-(pyridin-2-yl)ethyl]-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)propanamide
3-(3-fluorophenyl)-N-[1-(1,3-thiazol-5-yl)propan-2-yl]-1H-pyrazole-4-carboxamide
N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]-5-(oxolan-2-yl)thiophene-2-carboxamide
N-[(3,5-dimethyl-2-phenyl-1H-indol-7-yl)methyl]-3-methyl-1H-pyrazole-5-carboxamide
N-[1-(1H-imidazol-2-ylmethyl)azepan-3-yl]-2-methoxy-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
2-cyclopentyl-N-{[4-(2,3-dihydro-1H-inden-2-yloxy)-3-methoxyphenyl]methyl}-N-(oxolan-2-ylmethyl)acetamide
5-[6-amino-5-cyano-4-(3,4-dihydroxyphenyl)pyridin-2-yl]-2,4-dimethyl-1H-pyrrole-3-carboxylic acid
1-[4-(3-methoxybenzoyl)piperazin-1-yl]-2-(oxan-2-ylmethoxy)ethan-1-one
2-[2-(1H-imidazol-4-yl)ethyl]-9-(6-methylpyridine-2-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
N-({5-[(3,4-dimethoxyphenyl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)acetamide
5-(4-benzoylpiperidine-1-carbonyl)-1-cyclopropylpiperidin-2-one
4-{[(2R,3R,6R)-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]methyl}benzonitrile
N-(1-{7-[(2,4-difluorophenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}-3-methylbutyl)furan-2-carboxamide
1-[(2-chlorophenyl)methyl]-N-[(5-chlorothiophen-2-yl)methyl]-1H-1,2,3-triazole-4-carboxamide
1-methyl-1-[3-(oxolan-2-yl)propyl]-3-(2-phenyl-1,3-benzoxazol-5-yl)urea
3,5-dichloro-N-[(3R,4R)-4-hydroxypiperidin-3-yl]-4-methylbenzamide
1-(azepan-1-yl)-3-(3-{[(1H-imidazol-2-ylmethyl)(methyl)amino]methyl}phenoxy)propan-2-ol
4-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]-1-(4-methoxyphenyl)-6,6-dimethylpiperazin-2-one
N-cyclopropyl-5-methyl-4-(piperidin-1-yl)thieno[2,3-d]pyrimidine-6-carboxamide