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[(5-{[(2-chlorophenyl)methyl]sulfanyl}-4-methyl-4H-1,2,4-triazol-3-yl)methyl](cyclohex-3-en-1-ylmethyl)methylamine
5-(3-methylbutyl)-5-[1-(3-methylfuran-2-carbonyl)piperidin-4-yl]-3-(pyridin-2-ylmethyl)imidazolidine-2,4-dione
3-(4-benzylpiperazine-1-carbonyl)-2-ethyl-6-methyl-1-(thiophen-2-ylmethyl)-1,4-dihydropyridin-4-one
1-(3-cyclohexyl-1H-pyrazole-4-carbonyl)-4-cyclopentyl-1,4-diazepane
1-[4-(trifluoromethyl)pyridin-2-yl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
N-{[2-(3-hydroxypiperidin-1-yl)-8-methylquinolin-3-yl]methyl}-2,3-dimethoxy-N-[(4-methoxyphenyl)methyl]benzamide
4,6-dimethyl-3-[4-(4H-1,2,4-triazol-3-ylmethyl)piperazine-1-carbonyl]-1,2-dihydropyridin-2-one
3-[(2,4-difluorophenyl)methyl]-1-(2-methylpyrimidin-4-yl)piperidine-3-carboxylic acid
N-(2,2-dimethyloxan-4-yl)-2-{5-[(4-methylpiperidin-1-yl)methyl]-1H-1,2,3,4-tetrazol-1-yl}acetamide
3-{[(cyclopropylmethyl)amino]methyl}-1-(2,2-dimethylpropyl)-3-hydroxypiperidin-2-one
3-[1-(2-methyloxane-2-carbonyl)piperidin-4-yl]-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
4-[4-ethyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(1-ethylpiperidin-4-yl)piperidine
4-(2-methyl-1H-imidazol-1-yl)-1-[3-(pyridin-3-yl)propanoyl]piperidine-4-carboxylic acid
6-[1-(2,1,3-benzothiadiazol-5-ylmethyl)piperidin-4-yl]-2-methylpyrimidin-4-ol
N-(prop-2-en-1-yl)-N-(pyridin-3-ylmethyl)-1,3-benzothiazole-2-carboxamide
N-cyclopropyl-N-{[4-methoxy-3-(pyridin-4-ylmethoxy)phenyl]methyl}-3-(2-oxoimidazolidin-1-yl)benzamide
1-(6-ethoxy-4-methylquinazolin-2-yl)-N-[(2-methyl-1,3-thiazol-4-yl)methyl]piperidine-4-carboxamide
N-[2-(1-methylpiperidin-2-yl)ethyl]-6-[(pyridin-2-ylmethyl)amino]pyridine-3-carboxamide
3-phenyl-1-[3-(propan-2-yl)-1,2-oxazole-5-carbonyl]piperidine
1-[(4-fluorophenyl)methyl]-N-[3-(1H-indol-1-yl)propyl]-1H-1,2,3-triazole-4-carboxamide
4-{[2-(cyclohex-1-en-1-yl)ethyl]amino}-N-ethyl-5-methylthieno[2,3-d]pyrimidine-6-carboxamide
5-[4-(3-benzyl-1H-pyrazol-5-yl)piperidine-1-carbonyl]-3,4-dihydropyrimidin-4-one
5-({4-[(3-fluorophenyl)methyl]piperazin-1-yl}methyl)-2,1,3-benzoxadiazole
methyl 2-[(2,3-dihydro-1H-inden-5-yl)sulfamoyl]-6-(oxolane-2-carbonyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
2-(dimethylamino)-1-[9-hydroxy-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]ethan-1-one
2-(2-butoxyacetyl)-N-(pyridin-3-yl)-1,2,3,4-tetrahydroisoquinoline-6-sulfonamide
1-(2-methylpropyl)-4-(3-oxo-2,3-dihydro-1H-indene-1-carbonyl)-6-(pyridin-2-ylmethoxy)-1,4-diazepan-2-one
N-[(4-methoxyphenyl)methyl]-3-(1-methyl-1H-pyrazol-5-yl)-N-(oxolan-2-ylmethyl)propanamide
5-[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]-N-(pyridin-2-ylmethyl)pyridin-2-amine
1-phenyl-4-[4-(thiophen-2-ylmethyl)-1,4-diazepan-1-yl]butane-1,4-dione
[(4-{[1-(furan-3-carbonyl)piperidin-4-yl]oxy}phenyl)methyl](methyl)[(1-methyl-1H-pyrazol-4-yl)methyl]amine
1-{2-[(2,3,4,9-tetrahydro-1H-carbazol-6-ylmethyl)amino]pyrimidin-4-yl}pyrrolidin-3-ol
3-({4-[(1R,5S,8R)-8-(dimethylamino)-3-azabicyclo[3.2.1]octan-3-yl]-6-methylpyrimidin-2-yl}amino)phenol
N-{[7-(2H-1,3-benzodioxole-5-carbonyl)-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}-2-(methylsulfanyl)benzamide
1-[5-(1-cyclohexyl-1H-1,2,4-triazol-5-yl)-1H-pyrazol-3-yl]ethan-1-one
2-{1-[(3,4-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-ethyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]acetamide
(4aR,8aR)-4a-hydroxy-N,N-dimethyl-7-(2-methylpyrimidin-4-yl)-decahydro-2,7-naphthyridine-2-sulfonamide
2-(2,3-dihydro-1-benzofuran-7-yl)-3-(pyrrolidine-1-carbonyl)pyridine
N-[2-(1H-indol-3-yl)ethyl]-2-(1H-1,2,3,4-tetrazol-5-yl)benzamide
2-{4-[(1-ethyl-1H-pyrazol-4-yl)methyl]-1-(thiophen-2-ylmethyl)piperazin-2-yl}ethan-1-ol
N-cyclopropyl-1-(1-{[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]methyl}piperidin-4-yl)-1H-1,2,3-triazole-4-carboxamide
(2S,4R)-1-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]-4-(1H-1,2,3,4-tetrazol-1-yl)-N-(thiophen-2-ylmethyl)pyrrolidine-2-carboxamide
1-cyclohexyl-4-[3-(2,3-dimethoxyphenyl)pyrrolidine-1-carbonyl]-1H-1,2,3-triazole
2-(1-benzothiophen-2-yl)pyridine-3-carboxamide
2-[4-(4-{[2-(furan-2-yl)ethyl]amino}piperidin-1-yl)phenyl]-N-[2-(2-methoxyphenyl)ethyl]acetamide
3-cyclohexyl-N-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-N-methyl-1H-pyrazole-4-carboxamide
2-[5-(5-chloro-6-oxo-1,6-dihydropyridin-3-yl)-3-methyl-1H-1,2,4-triazol-1-yl]benzoic acid
N-[2-hydroxy-2-(prop-2-en-1-yl)pent-4-en-1-yl]-6-oxo-1-(3-phenylpropyl)piperidine-3-carboxamide
1'-{[1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}-1,2-dihydrospiro[indole-3,4'-piperidine]-2-one
N-methyl-3-[(3S,4R)-1-(2-methylpropyl)-4-{4-[3-(trifluoromethyl)phenyl]piperazin-1-yl}piperidin-3-yl]-N-[2-(pyridin-2-yl)ethyl]propanamide