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N-methyl-N-({1-[2-(2-methylphenyl)ethyl]piperidin-3-yl}methyl)-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide
(1R,9aR)-1-[({[5-(2-methylpropyl)-1,2-oxazol-3-yl]methyl}amino)methyl]-octahydro-1H-quinolizin-1-ol
3,4,7-trimethyl-2-[2-(1,3-thiazol-2-yl)piperidine-1-carbonyl]-1H-indole
2-({[(3R,4R)-4-(hydroxymethyl)-1-[3-(piperidine-1-carbonyl)pyridin-2-yl]pyrrolidin-3-yl]methyl}(methyl)amino)ethan-1-ol
N-methyl-1-[4-(methylsulfanyl)benzoyl]-N-(2-phenylethyl)piperidin-3-amine
1-(6-{1H-pyrrolo[2,3-b]pyridin-4-yl}pyridin-3-yl)ethan-1-one
7-(4-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-[2-(2-fluorophenyl)ethyl]-3-[(4-methoxyphenyl)methyl]-4,5-dihydro-1,2-oxazole-5-carboxamide
4-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)-N-methyl-N-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]benzamide
N-{2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]ethyl}-2-(pyridin-3-yl)-2-(pyrrolidin-1-yl)acetamide
N-{[2-(2,6-dimethylphenoxy)pyridin-3-yl]methyl}-3-methyl-1H-pyrazole-5-carboxamide
1-methyl-N-{[1-(piperidin-1-yl)cyclohexyl]methyl}-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
1-[3-(4-chlorophenyl)-1-(2-hydroxyethyl)-1H-1,2,4-triazol-5-yl]-3-methylbutan-1-ol
N-cyclopropyl-N-[(4-ethoxyphenyl)methyl]-1H-1,2,3-benzotriazole-5-carboxamide
3-{5-[2-(4H-1,2,4-triazol-4-yl)pyridine-4-carbonyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanoic acid
5-(2,6-dimethylphenoxymethyl)-N-[(4-fluorophenyl)methyl]-N-methyl-1,2-oxazole-3-carboxamide
N-[(2-methoxyphenyl)methyl]-4-oxo-N-propyl-4H-chromene-2-carboxamide
2-(4-fluorophenyl)-N-[1-(thiophen-2-yl)ethyl]imidazo[1,2-a]pyridine-6-carboxamide
3-fluoro-N-(1-{1-[2-(3-methyl-1H-pyrazol-1-yl)acetyl]piperidin-4-yl}-1H-pyrazol-5-yl)benzamide
(3aR,7aS)-2-[(1-ethyl-1H-pyrazol-4-yl)sulfonyl]-5-methyl-2,3,3a,4,7,7a-hexahydro-1H-isoindole
1-{3-[4-(dimethylamino)azepan-1-yl]-3-oxopropyl}-6-methyl-1,2-dihydropyridin-2-one
1-{3-[3-(2-fluorophenyl)phenyl]-1H-pyrazol-1-yl}butan-2-ol
3-{[1-ethyl-3-(pyrrolidine-1-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}-1H-indole
3-[5-(2H-1,3-benzodioxol-5-ylmethyl)-1,3,4-oxadiazol-2-yl]-1-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-1-one
5-[({1-[2-(4-fluorophenyl)ethyl]piperidin-4-yl}methyl)(methyl)carbamoyl]-2,1,3-benzoxadiazol-1-ium-1-olate
(1S,2S)-2-{[2-amino-6-(propan-2-yl)pyrimidin-4-yl]amino}-1-phenylpropane-1,3-diol
3-[4-(2-methoxyphenyl)piperazine-1-carbonyl]-N,N-dimethyl-6-(2-methylphenyl)pyridin-2-amine
N-[(2-chlorophenyl)methyl]-1-[(2-fluorophenyl)methyl]-N-methyl-1H-1,2,3-triazole-4-carboxamide
N-cyclopropyl-5-[(1-methyl-1H-imidazol-4-yl)sulfonyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
3-chloro-N-[2-(ethanesulfonyl)ethyl]-4-fluoro-1-benzothiophene-2-carboxamide
2-({[(3R,4R)-4-(hydroxymethyl)-1-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepine-3-carbonyl}pyrrolidin-3-yl]methyl}(methyl)amino)ethan-1-ol
1-(4-{1-[methyl(pyridin-4-ylmethyl)amino]-2-phenylethyl}piperidin-1-yl)-3-(thiophen-2-yl)propan-1-one
1-(2-{[1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl]amino}ethyl)-4,6-dimethyl-1,2-dihydropyrimidin-2-one
3-benzyl-4-[4-(dimethylamino)benzoyl]piperazin-2-one
1-(3,3-dimethyl-4-phenylpyrrolidin-1-yl)-3-methanesulfonylpropan-1-one
9-[(2-butyl-1H-imidazol-4-yl)methyl]-2-[(1r,4r)-4-hydroxycyclohexyl]-2,9-diazaspiro[5.5]undecan-3-one
1-(2-{imidazo[2,1-b][1,3]thiazol-6-yl}acetyl)-4-phenylpiperidine-4-carbonitrile
N-{2-ethyl-4-[2-(hydroxymethyl)-1H-1,3-benzodiazol-1-yl]phenyl}acetamide
1-[benzyl(methyl)amino]-3-[4-({[(3-methylphenyl)methyl]amino}methyl)phenoxy]propan-2-ol
4-[4-(5-methyl-1-propyl-1H-pyrazole-4-carbonyl)piperazin-1-yl]quinazoline
3-{2-[4-(1-butyl-1H-imidazol-2-yl)piperidin-1-yl]-2-oxoethyl}-1λ6-thiolane-1,1-dione
2-(1-{[1-(propan-2-yl)-1H-imidazol-2-yl]methyl}piperidine-3-carbonyl)pyridine
3-[3-(3-oxopiperazin-1-yl)propyl]-1-[2-(propan-2-ylsulfanyl)phenyl]urea
(1R,5R)-6-[(4-fluoro-3-methoxyphenyl)methyl]-3-(pyrazine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
4-methyl-14-[2-(pyridin-2-yl)pyrimidin-5-yl]-2,8,11-triazatricyclo[7.5.0.02,7]tetradeca-1(9),3,5,7-tetraen-12-one
N-cyclopentyl-4-(1H-imidazol-1-yl)-N-propylbenzamide
N-({1-[2-(4-methoxyphenyl)ethyl]piperidin-4-yl}methyl)-N,1-dimethylpiperidine-2-carboxamide
(2S,4R)-1-[(2-chlorophenyl)methyl]-4-{[(2,5-difluorophenyl)methyl]amino}-N-(2-methoxyethyl)pyrrolidine-2-carboxamide
(4aR,8aR)-4a-hydroxy-N,N-dimethyl-7-[(4-methylphenyl)methyl]-decahydro-2,7-naphthyridine-2-sulfonamide
2-{5H,6H,7H-[1,3]thiazolo[3,2-a]pyrimidin-3-yl}-N-{1-[5-(trifluoromethyl)pyridin-2-yl]piperidin-3-yl}acetamide