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N-cyclopentyl-N-{[4-methoxy-3-(thiophen-2-ylmethoxy)phenyl]methyl}cyclobutanecarboxamide
N-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-5-(2,5-dimethylphenoxymethyl)-1,2-oxazole-3-carboxamide
1-[3-(2,5-difluorobenzoyl)piperidin-1-yl]-4-(thiophen-2-yl)butan-1-one
N-[(2-amino-1,3-thiazol-4-yl)methyl]-4-(3,3,3-trifluoropropyl)pyrimidin-2-amine
5-{[3-(5-chloro-2-methoxybenzoyl)piperidin-1-yl]methyl}-2,1,3-benzothiadiazole
(3R,4S)-3,4-dimethyl-1-(2-propyl-1,3-thiazole-4-carbonyl)piperidin-4-ol
4-(3-fluorophenoxy)-1-[2-(2-methyl-1,3-thiazol-4-yl)ethyl]piperidine
2-{[(1-ethyl-1H-imidazol-2-yl)methyl]sulfamoyl}-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
4-(2-phenylethyl)-7-{[4-(pyridin-3-yloxy)piperidin-1-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepine
2-[2-(4-fluorophenyl)pyrrolidine-1-carbonyl]-1-methyl-1H-imidazole
2-{1-[(2-chloro-6-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-[3-(pyridin-3-yloxy)propyl]acetamide
N,N-diethyl-3-[5-(methoxymethyl)-3-methyl-1H-pyrazol-4-yl]benzamide
3-{3-[2-(2,6-difluorophenyl)ethyl]piperidine-1-carbonyl}-2-methylphenol
2-[4-(2H-1,3-benzodioxol-4-ylmethyl)-1-[(3,4-difluorophenyl)methyl]piperazin-2-yl]ethan-1-ol
N-(pyridin-3-ylmethyl)-4-[4-({[3-(trifluoromethoxy)phenyl]methyl}amino)piperidin-1-yl]benzamide
1-[1'-(5-fluoropyridine-3-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]-2-methoxyethan-1-one
2-{2-[2-(methoxymethyl)piperidin-1-yl]-2-oxoethyl}-1,2-dihydroisoquinolin-1-one
methyl 3-({1-[(2-chloro-4-fluorophenyl)methyl]-1H-1,2,3-triazol-4-yl}formamido)propanoate
N-[1-(1-ethyl-1H-1,2,4-triazol-5-yl)ethyl]-4-hydroxy-2-(thiophen-2-yl)pyrimidine-5-carboxamide
N-[1-methyl-3-(pyridin-2-yl)-1H-pyrazol-5-yl]-2-(1H-pyrazol-1-ylmethyl)-1,4-oxazepane-4-carboxamide
1-[2-(dimethylamino)-4-{[2-(4-ethyl-4H-1,2,4-triazol-3-yl)ethyl]amino}-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]ethan-1-one
2,6-dimethyl-4-({[1-(3-methyl-1,2,4-oxadiazol-5-yl)propyl]amino}methyl)phenyl acetate
2-phenyl-1-[4-(piperidine-1-sulfonyl)-1,4-diazepan-1-yl]ethan-1-one
2-(diethylamino)-1-{4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1,4-diazepan-1-yl}ethan-1-one
1-ethyl-4-[2-(4-methoxypiperidine-1-carbonyl)-2,3-dihydro-1H-inden-2-yl]piperazine
2-[1-(1-methylpiperidin-4-yl)-4-phenyl-1H-imidazol-5-yl]-1H-indole
2-(2,4-dichlorophenoxy)-1-[4-(4-methyl-4H-1,2,4-triazol-3-yl)piperidin-1-yl]ethan-1-one
2-fluoro-N-({6-methyl-2-[methyl(1H-pyrazol-5-ylmethyl)amino]quinolin-3-yl}methyl)-N-(oxolan-2-ylmethyl)benzamide
2-benzyl-N-(isoquinolin-5-ylmethyl)-N-methyl-1,3-thiazole-4-carboxamide
4-[2-(dimethylamino)-4-oxo-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-4-oxobutane-1-sulfonamide
5-acetyl-N-butyl-N-[(2-fluorophenyl)methyl]-6-methyl-2-oxo-1,2-dihydropyridine-3-carboxamide
N-(2-{7-[(2,4-dimethylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-4-methylbenzamide
5,6-dimethyl-3-{2-[2-(2-oxopyrrolidin-1-yl)ethyl]piperidine-1-carbonyl}-1,2-dihydropyridin-2-one
2,N4-dimethyl-N4-(4,5,6,7-tetrahydro-1,2-benzoxazol-3-ylmethyl)pyrimidine-4,6-diamine
ethyl 2-({[2-(dimethylamino)pyridin-3-yl]methyl}amino)-6-methylpyrimidine-4-carboxylate
N-(2,3-dihydro-1H-inden-2-yl)-2-(2,4-dioxo-1,3-diazinan-1-yl)benzamide
1-[2-(4-fluorophenyl)morpholin-4-yl]-3-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propan-1-one
[(2S,6S)-4-[(5-ethylfuran-2-yl)methyl]-11-methoxy-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-trien-6-yl]methanol
methyl 5-{[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]amino}-1-methyl-3-(3-phenylpropanamido)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
2-{[4-(2H-1,3-benzodioxol-5-ylmethyl)piperazin-1-yl]methyl}-7-chloro-4-(morpholin-4-yl)quinazoline
7-(2,2-dimethylpropyl)-2-(1H-imidazol-2-ylmethyl)-2,7-diazaspiro[4.5]decan-6-one
2-(3-hydroxypyridine-2-carbonyl)-N-(5-methyl-1,2-oxazol-3-yl)-1,2,3,4-tetrahydroisoquinoline-7-sulfonamide
1-{4-[3-(1H-pyrazol-3-yl)phenyl]phenyl}ethan-1-one
5-fluoro-4-(pyrrolidin-1-yl)-N-(1H-1,2,3,4-tetrazol-5-ylmethyl)pyrimidin-2-amine
1-ethyl-N-[(2-methoxyphenyl)methyl]-3-(morpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
2-{[3-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]methyl}-4H,5H,6H,7H,8H,9H-[1,2,4]triazolo[3,2-b]quinazolin-9-one
N-[(2-methoxyphenyl)methyl]-2-[3-(1-methyl-1H-imidazol-2-yl)piperidin-1-yl]acetamide
N-cyclobutyl-3-{[(5-ethyl-1,3,4-thiadiazol-2-yl)methyl]sulfamoyl}benzamide
1-(1-benzofuran-2-ylmethyl)-3-(2-methoxyethyl)piperidine
4-{[3-(3,4-difluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}-1,5-dimethyl-1H-pyrazole