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N-[2-(1H-1,3-benzodiazol-2-yl)ethyl]-2-cyclohexyl-1,3-benzoxazole-6-carboxamide
(1S,6R)-9-(pyridazine-4-carbonyl)-3,9-diazabicyclo[4.2.1]nonan-4-one
2-[(3-ethyl-1H-1,2,4-triazol-5-yl)sulfanyl]-N-[3-hydroxy-3-(prop-2-en-1-yl)hex-5-en-2-yl]acetamide
2-(3-{1,9-dimethyl-1,4,9-triazaspiro[5.5]undecane-4-carbonyl}piperidin-1-yl)acetamide
1-methyl-4-[3-(trifluoromethyl)-1H-pyrazole-5-carbonyl]piperazine-2-carboxylic acid
N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-2-hydroxy-4-methylpentanamide
4-[2,4-dimethyl-5-(1H-1,2,4-triazol-1-ylmethyl)phenyl]-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
[1-({1-[(2,5-dimethylthiophen-3-yl)sulfonyl]piperidin-4-yl}methyl)-1H-1,2,3-triazol-4-yl]methanamine
(4aS,8aR)-6-[(2-oxo-1,2-dihydroquinolin-3-yl)methyl]-1-propyl-decahydro-1,6-naphthyridin-2-one
(1S,5R)-3-benzyl-6-(3-propyl-1H-pyrazole-5-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
N-(2-methoxyethyl)-2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]-N-(1,3-thiazol-2-ylmethyl)acetamide
(4aS,7aR)-1-(3-ethyl-4-methyl-1H-pyrazole-5-carbonyl)-4-(2-methylpropanoyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
{[3-(3-chlorophenyl)-1-methyl-1H-pyrazol-4-yl]methyl}(oxolan-2-ylmethyl)(pyridin-4-ylmethyl)amine
1-[(1R,5R)-6-(3-methylbut-2-en-1-yl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]-3-(1H-pyrazol-1-yl)propan-1-one
N-methyl-N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-3-(5-methylthiophen-2-yl)-5-(morpholine-4-sulfonyl)benzamide
7-(cyclobutylmethyl)-2-(morpholine-4-sulfonyl)-2,7-diazaspiro[4.5]decan-6-one
1-[(4-methyl-1H-imidazol-5-yl)methyl]-4-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
N-({7-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)-2-phenylacetamide
N-{2-[(2-methylquinolin-8-yl)oxy]ethyl}-4-(trifluoromethyl)pyrimidin-2-amine
[1-(2,3-dihydro-1-benzofuran-5-ylmethyl)-4-{[2-(trifluoromethyl)phenyl]methyl}piperidin-4-yl]methanol
3-benzyl-8-[1-(methylsulfanyl)propan-2-yl]-1-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
({2,5-dimethyl-3-[(4-methylpiperazin-1-yl)methyl]phenyl}methyl)(methyl)[(5-methylfuran-2-yl)methyl]amine
3-(2-ethyl-7-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-1-{4-[(1-methyl-1H-imidazol-2-yl)methyl]piperazin-1-yl}propan-1-one
2-(3-chlorophenoxy)-N-[(1S,2R)-2-[(1-ethylpiperidin-4-yl)amino]cyclobutyl]acetamide
2-({[2-(2,4-dimethylphenoxy)ethyl](methyl)amino}methyl)phenol
N-[2-(1H-imidazol-1-yl)-1-phenylethyl]-1H-1,2,3-triazole-5-carboxamide
ethyl 1-{1-[4-(cyclopentylcarbamoyl)phenyl]piperidin-4-yl}piperidine-2-carboxylate
2-(3-fluorophenyl)-N-(4-{4-[4-(pyridin-2-yl)piperazin-1-yl]piperidin-1-yl}phenyl)acetamide
(1S,5R)-3-[(4-fluorophenyl)methyl]-6-[5-(methoxymethyl)thiophene-2-carbonyl]-3,6-diazabicyclo[3.2.2]nonane
2-acetyl-8-(5-acetylpyridin-2-yl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
methyl (2S)-2-{[2-(3-fluorophenoxymethyl)-1,3-oxazol-4-yl]formamido}-3-methylbutanoate
3-(2H-1,3-benzodioxol-5-yl)-5-[(3-fluorophenyl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
4-{[5-(4-chlorophenyl)furan-2-yl]methyl}-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
4-{[2-(2-methoxyethyl)morpholin-4-yl]methyl}quinoline
3-(4-{3-cyclopropyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-6-yl)pyridine
N-[(3-methylphenyl)methyl]-1-(prop-2-en-1-yl)-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
1-{1-[(2-chlorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}-3-(2-methylphenoxymethyl)piperidine
N-ethyl-N-{[1-(1-methylpiperidin-4-yl)piperidin-4-yl]methyl}-4-phenylbenzamide
(3S,9aR)-3-(4-aminobutyl)-8-[(3-methylthiophen-2-yl)methyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
4-[(1-ethyl-1H-pyrazol-4-yl)methyl]-1-[(4-methylphenyl)methyl]piperazin-2-one
2-{5H,6H-imidazo[2,1-b][1,3]thiazol-3-yl}-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}acetamide
2-ethyl-5-{3-[(methylsulfanyl)methyl]piperidine-1-carbonyl}pyrimidine
(2S)-2-{[2-(adamantan-1-yl)-4-hydroxypyrimidin-5-yl]formamido}-3-methylbutanamide
3-ethyl-8-[1-ethyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
6-(3-methylbenzoyl)-N-[(6-methylpyridin-2-yl)methyl]-6-azaspiro[2.5]octane-1-carboxamide
N-(2,1,3-benzothiadiazol-5-ylmethyl)-4-ethyl-2-methyl-1,3-thiazole-5-carboxamide
(2S)-N-[(3,5-dimethyl-2-phenyl-1H-indol-7-yl)methyl]oxolane-2-carboxamide
2-(4-fluorophenyl)-N-[2-(2-methylpropoxy)phenyl]-3-oxopiperazine-1-carboxamide
6-{1-[(2,3-dimethyl-1H-indol-7-yl)methyl]piperidin-4-yl}-2-methylpyrimidin-4-ol
4-fluoro-N-[2-({5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}amino)ethyl]benzamide