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4-(2-methyl-2H-1,2,3,4-tetrazol-5-yl)-N-[(5-methylthiophen-2-yl)methyl]-N-(prop-2-en-1-yl)benzamide
4'-{[4-(1H-pyrazol-1-yl)phenyl]methyl}-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
3-(2-amino-1,3-thiazol-4-yl)-N-[(1-methyl-1H-imidazol-2-yl)methyl]-N-propylpropanamide
N-{2-[1-(4-fluorophenyl)-3-(2-methylpropyl)-1H-1,2,4-triazol-5-yl]ethyl}-N-methylmethanesulfonamide
6-{3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-(methylsulfanyl)pyrimidin-4-amine
(3S,9aR)-8-(4-ethylbenzoyl)-3-[(1R)-1-hydroxyethyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
propyl 3-{1-[3-(dimethylamino)propyl]-1H-imidazol-2-yl}piperidine-1-carboxylate
4-[1-(2-chlorobenzenesulfonyl)piperidin-3-yl]benzoic acid
N-methyl-N-(1,2-oxazol-3-ylmethyl)-2-(3-oxo-1-{[3-(trifluoromethyl)phenyl]methyl}piperazin-2-yl)acetamide
3-({3-[(2-chloro-6-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-4-ethylpiperazin-2-one
N-[(1-methyl-1H-imidazol-2-yl)methyl]-1-[3-(morpholin-4-yl)propyl]-6-oxopiperidine-3-carboxamide
4-(pyridin-2-yl)-N-[1-(pyridin-2-ylmethyl)piperidin-4-yl]pyrimidin-2-amine
6-fluoro-2-[({1-oxaspiro[4.4]nonan-3-yl}amino)methyl]quinolin-4-ol
N-{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N,5-dimethyl-1,3-oxazole-4-carboxamide
2-{3'-oxo-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-1-yl}-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
3-(benzenesulfonyl)-1-[6-(hydroxymethyl)-1,4-oxazepan-4-yl]propan-1-one
2-(4-chlorophenyl)-4-(3-phenyl-1,2,4-oxadiazol-5-yl)morpholine
ethyl 4-{[3-(3-fluoro-4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}piperazine-1-carboxylate
N-{[5-(naphthalen-2-ylmethyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}cyclobutanecarboxamide
1-{3-methoxy-4-[(1-methylpiperidin-4-yl)oxy]benzoyl}-4-(2-methoxyethoxy)piperidine
1-methyl-3-(2-methylpropyl)-N-[2-(2-oxopyrrolidin-1-yl)ethyl]-1H-pyrazole-5-carboxamide
9-(7-methoxy-4-methylquinazolin-2-yl)-1-methyl-1,4,9-triazaspiro[5.5]undecan-5-one
1-(4-ethyl-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-7-yl)-3-[3-(2-oxopyrrolidin-1-yl)propyl]urea
N-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-N-methyl-5-oxo-1-phenyl-2,5-dihydro-1H-pyrazole-3-carboxamide
N-({2-[(methylsulfanyl)methyl]-1,3-thiazol-4-yl}methyl)-5-oxo-1-(pyridin-3-ylmethyl)pyrrolidine-3-carboxamide
N,5-dimethyl-N-[2-(morpholin-4-yl)propyl]pyrazolo[1,5-a]pyrimidin-7-amine
N-benzyl-N-(2-hydroxyethyl)-1-methyl-2-oxo-1,2-dihydropyridine-3-carboxamide
2-(2-methoxy-5-{3-oxa-9-azaspiro[5.5]undecan-9-ylmethyl}phenoxy)acetic acid
1-(benzyloxy)-8-{2-[(4-methyl-1,3-thiazol-2-yl)sulfanyl]acetyl}-1,8-diazaspiro[4.5]decan-2-one
N-[(3S,4R)-4-ethoxyoxolan-3-yl]-6-methylimidazo[2,1-b][1,3]thiazole-5-carboxamide
1-{[3-(butan-2-yloxy)phenyl]methyl}-4-(pyridin-2-ylmethyl)-1,4-diazepane
3-{[(3-methyloxetan-3-yl)methyl]sulfamoyl}-N-(2-methylphenyl)benzamide
3-[5-(2H-1,3-benzodioxol-5-ylmethyl)-1,3,4-oxadiazol-2-yl]-N-[(1R,4S,6S)-spiro[bicyclo[2.2.1]heptane-7,1'-cyclopropan]-2-en-6-ylmethyl]propanamide
N-methyl-N-[2-(4-phenylphenyl)ethyl]oxan-4-amine
1-(1H-imidazol-4-ylmethyl)-3-{2-[2-(trifluoromethyl)phenyl]ethyl}piperidine
ethyl 3-({3-[ethyl(pyridin-4-ylmethyl)amino]piperidine-1-carbonyl}amino)propanoate
(3S,4S)-4-methoxy-N-{2-methylthieno[3,2-d]pyrimidin-4-yl}-1-(propan-2-yl)pyrrolidin-3-amine
N-cyclopropyl-1-[1-(dimethyl-1,3-thiazole-5-carbonyl)piperidin-4-yl]piperidine-3-carboxamide
5-(adamantan-1-yl)-3-(oxolan-3-yl)-1,2,4-oxadiazole
(3S,4R)-4-(2H-1,3-benzodioxol-5-yl)-1-[3-(2-methyl-1H-imidazol-1-yl)propanoyl]pyrrolidine-3-carboxylic acid
4-[2-(7-methyl-2-oxo-2H-chromen-4-yl)acetyl]-1-(2-methylpropyl)-6-(pyridin-2-ylmethoxy)-1,4-diazepan-2-one
5-(2-chloro-4-methoxyphenoxymethyl)-N-(2-oxopiperidin-3-yl)-1H-pyrazole-3-carboxamide
methyl 3-({[4-(dimethylamino)phenyl]formamido}methyl)-5-(furan-3-amido)benzoate
1-{imidazo[2,1-b][1,3]thiazole-6-carbonyl}-4-(1H-pyrazol-1-yl)piperidine-4-carboxylic acid
2-{1-[(6-methylpyridin-2-yl)methyl]-4-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}piperazin-2-yl}ethan-1-ol
1-{3-[(3-chlorophenyl)methyl]-3-(hydroxymethyl)piperidin-1-yl}-4-(1H-1,2,4-triazol-1-yl)butan-1-one
ethyl 5-(2,2-dimethylpropanoyl)-1-[(3-methoxyphenyl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
3-({[(1-hydroxycyclohexyl)methyl]carbamoyl}methyl)-N,N,4-trimethyl-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
N-[(3,5-dimethyl-2-phenyl-1H-indol-7-yl)methyl]-2-(2,5-dioxoimidazolidin-1-yl)acetamide
N-ethyl-N-(pyridin-4-ylmethyl)quinoxaline-5-carboxamide