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dimethyl[2-(2-{3-oxa-9-azaspiro[5.5]undecan-9-ylmethyl}phenoxy)ethyl]amine
3-(4-methoxyphenyl)-N-[(3-methyloxetan-3-yl)methyl]-3-phenylpropanamide
3-(3-fluorophenyl)-4-[3-(1-methyl-1H-pyrrol-2-yl)-1H-pyrazole-5-carbonyl]piperazin-2-one
4-(6-{3-[1-(pyrrolidin-1-yl)ethyl]phenyl}pyrazine-2-carbonyl)morpholine
N-{[2-(2,5-dimethoxyphenyl)-8-methylquinolin-3-yl]methyl}-N-(furan-2-ylmethyl)-3-(3-methyl-1H-pyrazol-1-yl)propanamide
2-methyl-5-(4-{[4-(pyridin-2-yl)phenyl]methyl}piperazin-1-yl)-2,3-dihydropyridazin-3-one
methyl 3-[(2-ethylbutanamido)methyl]-5-(2-methoxybenzamido)benzoate
2-{6-chloro-1H,2H,3H,4H,5H-pyrido[4,3-b]indol-2-yl}-5-propyl-1,3,4-oxadiazole
3-[(3,4-difluorophenyl)methyl]-9-methoxy-7-oxo-N-(thiophen-3-ylmethyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
2-[5-(2-methoxyethyl)-3-(pyridin-4-yl)-1H-1,2,4-triazol-1-yl]ethan-1-ol
3-methyl-7-[1-(2-methylpropyl)-5-oxopyrrolidine-3-carbonyl]-5,6,7,8-tetrahydro-2,7-naphthyridine-4-carbonitrile
7-(3-methoxyphenyl)-2-(3-propyl-1,2-oxazol-5-yl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
ethyl 1-ethyl-5-(1H-indol-3-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
5,7-dimethyl-4-(2-methylpyrrolidine-1-carbonyl)-2-(1-propyl-1H-pyrazol-4-yl)quinoline
1-[4-(1-{[(1,3-dimethyl-1H-pyrazol-4-yl)methyl](methyl)amino}-2-phenylethyl)piperidin-1-yl]-2-(1,3-thiazol-4-yl)ethan-1-one
N-cyclopentyl-1-{1-[(2E)-3-(thiophen-2-yl)prop-2-enoyl]piperidin-4-yl}-1H-1,2,3-triazole-4-carboxamide
N-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl]-N-methyl-4-oxo-4,5,6,7-tetrahydro-1-benzofuran-3-carboxamide
(1-ethyl-5-{[2-(pyrrolidin-1-yl)-1,3-thiazol-5-yl]methyl}-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-3-yl)methanol
3-[(3S,4R)-1-[(2,3-dimethoxyphenyl)methyl]-4-[4-(2-fluorophenyl)piperazin-1-yl]piperidin-3-yl]-N-(4-methoxyphenyl)propanamide
(1R,2R,6S,7S)-4-[(3-fluoropyridin-2-yl)methyl]-10-oxa-4-azatricyclo[5.2.1.02,6]decane
2-(2,3-dihydro-1H-inden-1-yl)-N-{[4-(pyrrolidine-1-carbonyl)phenyl]methyl}acetamide
1-{2-[4-(2-methylphenoxy)piperidin-1-yl]-2-oxoethyl}piperidin-2-one
1-(5-methyl-2-phenyl-1H-imidazole-4-carbonyl)-4-phenylpiperidine-4-carbonitrile
5-(4-methoxyphenyl)-N-[(2-phenyl-1,3-thiazol-5-yl)methyl]-1,2,4-triazin-3-amine
N-({7-[2-(2H-1,3-benzodioxol-5-yl)acetyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)oxolane-3-carboxamide
3-{1-[1-(3-ethyl-1-methyl-1H-pyrazole-5-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}-1-(3-fluorophenyl)urea
N-[2-(5-cyclopentyl-1,2,4-oxadiazol-3-yl)ethyl]-5-oxo-1-phenyl-2,5-dihydro-1H-pyrazole-3-carboxamide
6-{4H,5H,6H,7H,8H-cyclohepta[b]thiophene-2-carbonyl}-2-ethyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine
methyl({3-[1-(4-methylphenyl)cyclopentyl]-1,2,4-oxadiazol-5-yl}methyl)[4-(morpholin-4-yl)butyl]amine
methyl 2-{[(1R,2S,9R)-6-oxo-7,11-diazatricyclo[7.3.1.02,7]tridecan-11-yl]methyl}-1,3-oxazole-4-carboxylate
N-(1-{4-[4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazine-1-carbonyl]phenyl}-1H-pyrazol-4-yl)acetamide
3-{2-oxo-2-[2-(pyridin-2-yl)piperidin-1-yl]ethyl}-1,3-oxazolidin-2-one
(3S,4R)-1-(1-methyl-4,5,6,7-tetrahydro-1H-indazole-3-carbonyl)-4-phenylpyrrolidine-3-carboxylic acid
2-cyclopentyl-N-({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)-N-(2-methoxyethyl)acetamide
2-{4-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]-1-[(4-methoxy-2,3-dimethylphenyl)methyl]piperazin-2-yl}ethan-1-ol
3,5-dimethyl-2-[2-(trifluoromethyl)morpholine-4-carbonyl]-1H-indole
N-({3-[4-(1-methoxyethyl)phenyl]phenyl}methyl)acetamide
1-(furan-2-ylmethyl)-3-[5-oxo-1-(3-phenylpropyl)pyrrolidin-3-yl]urea
1-{3-[4-(4-methoxyphenyl)piperazin-1-yl]piperidin-1-yl}-3-phenylprop-2-yn-1-one
N-({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)-N-(pyridin-3-ylmethyl)oxan-4-amine
N-ethyl-2-fluoro-N-[2-(pyrrolidin-1-yl)ethyl]-5-sulfamoylbenzamide
N-(1-ethyl-1H-pyrazol-4-yl)-4-(1-hydroxy-3-phenylpropyl)piperidine-1-carboxamide
[(3R,4R)-4-{[(2-methoxyethyl)(methyl)amino]methyl}-1-[(5-methylthiophen-2-yl)methyl]pyrrolidin-3-yl]methanol
methyl 6-(azepan-1-ylmethyl)-3-(5-methylthiophene-2-amido)thieno[2,3-b]pyridine-2-carboxylate
ethyl 2-[3-(2,5-dimethoxyphenyl)pyrrolidin-1-yl]-1,3-oxazole-4-carboxylate
N4-[1-(cyclohexylmethyl)piperidin-3-yl]pyrimidine-4,6-diamine
N-[2-({3-[(2-methylprop-2-en-1-yl)oxy]phenyl}formamido)ethyl]acetamide
N-[2-(3,4-dimethylphenoxy)ethyl]-1-methyl-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
ethyl 3-[(2-fluorophenyl)methyl]-1-[3-(1H-pyrazol-1-yl)benzoyl]piperidine-3-carboxylate
4-(1-{1-[(5-methylfuran-2-yl)methyl]piperidin-4-yl}piperidine-4-carbonyl)morpholine