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{[3-(2-fluoro-4-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl}(methyl)(pyridin-2-ylmethyl)amine
1-{1,9-dimethyl-1,4,9-triazaspiro[5.5]undecan-4-yl}-3-(2-methoxyphenyl)propan-1-one
2-(furan-2-yl)-N-(furan-2-ylmethyl)-7-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
ethyl 4-(1-{2-[(4-methyl-1,3-thiazol-2-yl)sulfanyl]acetyl}piperidin-3-yl)piperazine-1-carboxylate
3-ethyl-N-[3-(1H-imidazol-1-yl)propyl]-5-methyl-N-(pyridin-3-ylmethyl)-1,2-oxazole-4-carboxamide
3-[3-cyclopropyl-1-(3-fluorophenyl)-1H-1,2,4-triazol-5-yl]-4-fluorobenzene-1-sulfonamide
5-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl]pyridine-2-carbonitrile
4-cyclopentyl-N-methyl-N-{[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}pyrimidin-2-amine
1-[6-methyl-2-(pyrrolidin-1-yl)pyrimidin-4-yl]-N-[3-(1H-1,2,4-triazol-1-yl)propyl]piperidin-4-amine
methyl 4-{[1-(cyclohexylmethyl)-6-oxopiperidin-3-yl]formamido}butanoate
6-(hydroxymethyl)-N-{4-[2-(pyridin-2-yl)ethyl]phenyl}-1,4-oxazepane-4-carboxamide
2-(1-{[3-(2-phenylethyl)-1,2,4-oxadiazol-5-yl]methyl}piperidin-3-yl)-1,3-benzoxazole
2-[4-({methyl[2-(2-methyl-1H-imidazol-1-yl)ethyl]amino}methyl)phenyl]-3,4,5,6,7,8-hexahydroquinazolin-4-one
ethyl 5-{imidazo[1,2-a]pyridine-2-carbonyl}-1-[(4-methoxyphenyl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
3-(4,5-dimethyl-1H-pyrazol-3-yl)-1-{4-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}propan-1-one
N-{[5-(4-methanesulfonylphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-(4-methylphenoxy)acetamide
N-{[5-(1-benzofuran-5-ylmethyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}acetamide
(2R,3R,6R)-N-ethyl-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carboxamide
N-(dimethyl-1,2-oxazol-4-yl)-4-{[2-(4-methyl-1,2,5-oxadiazol-3-yl)pyrrolidin-1-yl]methyl}benzamide
N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-3-(1H-pyrazol-1-ylmethyl)benzamide
5-({[1-(4-fluorophenyl)-3-(2-methylpropyl)-1H-1,2,4-triazol-5-yl]methyl}sulfanyl)-1,3,4-thiadiazol-2-amine
8-[(4-methoxypyridin-2-yl)methyl]-3-(2-phenylethyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-[(2-fluorophenyl)methyl]-4-[2-(2-methoxyphenyl)pyrrolidine-1-carbonyl]-1H-1,2,3-triazole
N-[4-(2-carbamoylethyl)-2-fluorophenyl]-2-phenylbutanamide
N-{1-[1-(2,1,3-benzothiadiazol-5-ylmethyl)piperidin-4-yl]-2-phenylethyl}-N,2-dimethylfuran-3-carboxamide
5-{2-[(2-ethyl-6-methylpyridin-3-yl)oxy]acetyl}-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxylic acid
4-(2H-1,3-benzodioxol-5-yl)-3-(piperidin-1-ylmethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
(1-{imidazo[1,2-a]pyridine-6-carbonyl}piperidin-4-yl)(pyridin-2-yl)methanol
1,3-dimethyl-6-[4-(1-methyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
4-(4-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}benzoyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
2-{[4-(methoxymethyl)piperidin-1-yl]sulfonyl}-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
ethyl 4-[(4-methoxyphenyl)methyl]-1-(1,3-thiazole-5-carbonyl)piperidine-4-carboxylate
5-methoxy-N-methyl-N-(quinolin-4-ylmethyl)furan-2-carboxamide
N-[(2,3-dimethoxyphenyl)methyl]-3-{2-[(4-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}propanamide
6-(methoxymethyl)-N-[2-(5-methylthiophen-2-yl)ethyl]pyrimidin-4-amine
3-benzyl-1-(2-phenylethyl)-8-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
5-(1H-indol-2-ylmethyl)-1-(2-methoxyethyl)-N-(pyridin-3-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
1-(4-{[2-(ethylamino)pyrimidin-5-yl]methyl}-1-methyl-1,4,9-triazaspiro[5.5]undecan-9-yl)-2-methoxyethan-1-one
N-(1-{5-[(cyclohexylmethyl)sulfanyl]-4-methyl-4H-1,2,4-triazol-3-yl}-2-phenylethyl)propanamide
N-(2-phenylpropyl)-3-(5-{[3-(trifluoromethyl)phenyl]methyl}-1,3,4-oxadiazol-2-yl)propanamide
5-{5-[3-(2,3-dimethoxyphenyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}pyrimidine
2-[2-(dimethylamino)ethyl]-8-(5-ethyl-1,2,4-oxadiazol-3-yl)-2,8-diazaspiro[5.5]undecan-3-one
N-[(2,4-dimethoxyphenyl)methyl]-3-[1-(2-methoxypyridine-3-carbonyl)piperidin-3-yl]propanamide
4-({2-ethyl-5-oxo-5H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-yl}methyl)-5-methyl-1-phenylpiperazin-2-one
N-cyclopropyl-6-(1-methyl-1H-indol-2-yl)pyridazin-3-amine
(4-{[2-(2-methylphenyl)pyrimidin-5-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl)methanol
3-(azepane-1-carbonyl)-N,1-dimethyl-N-(1,3-thiazol-4-ylmethyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
N-[2-(4-chloro-1H-pyrazol-1-yl)ethyl]-3-(3-hydroxy-3-methylbutyl)benzamide
2-(2-methoxyethyl)-N-[3-(1,2,3,4-tetrahydroquinolin-1-yl)propyl]-1,3-benzoxazole-6-carboxamide
(2-{2-[1-(2,3-difluorobenzoyl)piperidin-3-yl]-1H-imidazol-1-yl}ethyl)dimethylamine