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N,N-diethyl-1-({4-[(3-hydroxyphenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}methyl)piperidine-3-carboxamide
5-[(1-phenyl-1H-1,2,3-triazol-4-yl)methyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxylic acid
5-cyclopropyl-1-{9-methoxy-5H,6H-benzo[h]quinazolin-2-yl}-N-methyl-N-[2-(pyridin-2-yl)ethyl]-1H-pyrazole-4-carboxamide
5-{2-[(1R,5R)-6-(cyclobutylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]-2-oxoethyl}-2-methyl-3,4-dihydropyrimidin-4-one
(3S,4R)-1-{5H,6H,7H,8H-imidazo[1,2-a]pyrazine-2-carbonyl}-4-(3-methylthiophen-2-yl)piperidin-3-ol
3-(6-methoxyhexanoyl)-3,9-diazaspiro[5.6]dodecan-10-one
1-[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]-3-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]piperidine
methyl[(1-methyl-1H-indol-2-yl)methyl]{[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]methyl}amine
N-[(3,4-dimethoxyphenyl)methyl]-N-(pyridin-2-ylmethyl)naphthalene-1-carboxamide
(propan-2-yl)({[2-(propylsulfanyl)pyrimidin-5-yl]methyl})[(trimethyl-1H-pyrazol-4-yl)methyl]amine
(1R,6S)-N-[4-(1H-1,3-benzodiazol-2-yl)phenyl]-9-methyl-3,9-diazabicyclo[4.2.1]nonane-3-carboxamide
2-{4-[5-(methoxymethyl)thiophene-2-carbonyl]piperazin-1-yl}-1,3-benzothiazole
3,5-dimethyl-6-[3-(1-methyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-3H,4H-thieno[2,3-d]pyrimidin-4-one
1-{3-[(3-chlorophenyl)methyl]-3-(hydroxymethyl)piperidin-1-yl}-2-(methylsulfanyl)ethan-1-one
2-(3,4-dimethoxyphenyl)-3-{[3-(methoxymethyl)pyrrolidin-1-yl]methyl}-7-methylquinoline
3-({2-[1-(5-methoxyfuran-2-carbonyl)piperidin-4-yl]-1H-imidazol-1-yl}methyl)pyridine
4-(3,6-dimethylpyrazin-2-yl)-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-({3,5-dimethoxy-4-[2-(thiophen-3-yl)ethoxy]phenyl}methyl)-N-[(3S)-2-oxoazepan-3-yl]-2-(trifluoromethyl)benzamide
(2S,4R)-4-amino-1-(2,1,3-benzothiadiazole-4-sulfonyl)-N-(propan-2-yl)pyrrolidine-2-carboxamide
N-(1,1-dioxo-1λ6-thiolan-3-yl)-3-(3-hydroxy-3-methylbutyl)-N-(2-hydroxyethyl)benzamide
N-(2-ethoxyphenyl)-3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidine-1-carboxamide
N-[(1-ethylpyrrolidin-2-yl)methyl]-2-methyl-6-(piperidin-4-yl)pyrimidin-4-amine
1-[2-(3-fluorophenyl)ethyl]-N-[(4-methyl-1H-imidazol-2-yl)methyl]-6-oxopiperidine-3-carboxamide
4-phenyl-3-{[1-(3,3,3-trifluoropropyl)piperidin-4-yl]methyl}-4,5-dihydro-1H-1,2,4-triazol-5-one
1-[2-(4-methoxyphenyl)ethyl]-N-(1,2-oxazol-3-ylmethyl)-6-oxopiperidine-3-carboxamide
(3aS,6aR)-5-[(2E)-3-phenylprop-2-en-1-yl]-3-(pyridin-2-ylmethyl)-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
3-(2,3-dihydro-1H-inden-2-yl)-1-ethyl-8-{[2-(furan-2-yl)phenyl]methyl}-1,3,8-triazaspiro[4.5]decane-2,4-dione
(2S,4S)-1-[(2-chlorophenyl)methyl]-4-{[(4-methoxy-2,3-dimethylphenyl)methyl]amino}-N-(propan-2-yl)pyrrolidine-2-carboxamide
1-ethyl-5-oxo-N-(3-{[1,2,4]triazolo[4,3-a]pyridin-3-yl}propyl)pyrrolidine-3-carboxamide
8-methoxy-N-[3-(4-methyl-1H-pyrazol-1-yl)propyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
N-[1-(2-cyclopentylacetyl)azepan-3-yl]thiophene-2-sulfonamide
2-(3-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-5-yl)-N-[(4-phenyloxan-4-yl)methyl]acetamide
4-(4-hydroxyphenyl)-N-methyl-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}benzamide
N-cyclopropyl-5-[2-(prop-2-en-1-ylsulfanyl)propanoyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
2-(3-{1-[2-(dimethylamino)ethyl]-1H-imidazol-2-yl}piperidin-1-yl)-N-ethylpyridine-4-carboxamide
9-(2,5-dimethylbenzoyl)-2-(2-methoxyethyl)-2,9-diazaspiro[5.5]undecan-3-one
4-chloro-N,N-bis(pyridin-3-ylmethyl)-1H-pyrrole-2-carboxamide
2-[4-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-1-[(2-fluorophenyl)methyl]piperazin-2-yl]ethan-1-ol
3-(2H-1,3-benzodioxol-5-ylmethyl)-5-ethyl-5-[1-(3-methylpentanoyl)piperidin-4-yl]imidazolidine-2,4-dione
[1-(3-fluoropyridin-2-yl)-3-(2-phenylethyl)piperidin-3-yl]methanol
N-[2-(1H-1,3-benzodiazol-2-yl)ethyl]-5-(1-benzofuran-2-yl)-N-methyl-1,2,4-triazin-3-amine
1-methyl-4-phenyl-3-[1-(piperidin-4-yl)piperidin-3-yl]-4,5-dihydro-1H-1,2,4-triazol-5-one
3-methyl-N-[(2-{methyl[2-(pyridin-2-yl)ethyl]amino}pyridin-3-yl)methyl]pyridine-4-carboxamide
2-methyl-6-{3-[1-(pyrrolidin-1-yl)ethyl]phenyl}-2,3-dihydropyridazin-3-one
1-{furo[3,2-c]pyridin-4-yl}-3-[(3-methoxyphenyl)methyl]piperidine-3-carboxylic acid
4-[(2-tert-butyl-1H-imidazol-1-yl)methyl]-1-cyclopentylpiperidine
3-methyl-N-[1-(1-{7-methylimidazo[1,2-a]pyridine-2-carbonyl}piperidin-4-yl)-1H-pyrazol-5-yl]butanamide
1-methyl-3-(2-{1-[3-(trifluoromethyl)phenyl]-1H-1,2,4-triazol-5-yl}ethyl)piperidine
2-(1-{1-[(2-methylphenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}piperidin-2-yl)ethan-1-ol
(4aR,7aS)-1-(cyclopropylmethyl)-4-[(3,4-dimethylphenyl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione