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1-(2-fluorophenyl)-N-{[4-methoxy-3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}-4,5,6,7-tetrahydro-1H-indazol-4-amine
5-{1-[(2-methoxyphenyl)methyl]piperidin-4-yl}-5-(2-methylpropyl)-3-[2-(thiophen-2-yl)ethyl]imidazolidine-2,4-dione
N-ethyl-N-{[1-(1-methylpiperidin-4-yl)piperidin-4-yl]methyl}-2-(quinazolin-4-yloxy)acetamide
6-[4-(2-fluorophenoxy)piperidine-1-carbonyl]-2,3-dimethylquinoxaline
1-{1,3-dioxo-2-[(3,4,5-trimethoxyphenyl)methyl]-2,3-dihydro-1H-isoindol-4-yl}-N-ethyl-N-(2-methylprop-2-en-1-yl)piperidine-3-carboxamide
5-(2H-1,3-benzodioxole-5-carbonyl)-N-ethyl-1-[(3-methoxyphenyl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
2-(azocan-1-ylmethyl)-4-(2,5-dimethoxyphenyl)phenol
1-(4-{[(3S,4R)-3-[(dimethylsulfamoyl)amino]-4-(propan-2-yl)pyrrolidin-1-yl]methyl}thiophen-2-yl)ethan-1-one
1-{1-[(4-hydroxy-3-methoxyphenyl)methyl]piperidin-3-yl}-N-(2-methylpropyl)-1H-1,2,3-triazole-4-carboxamide
2-(4-{[methyl(1-methylpiperidin-4-yl)amino]methyl}phenyl)-6-(trifluoromethyl)-3,4-dihydropyrimidin-4-one
N-{[2-(3,5-dimethyl-1H-pyrazol-1-yl)-5-fluorophenyl]methyl}-3,4-dihydro-2H-1-benzopyran-3-amine
(3aR,6aR)-2-{4H,5H,6H,7H,8H-cyclohepta[b]thiophene-2-carbonyl}-5-methyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
(2R,3R,6R)-5-(2-methoxypyridine-3-carbonyl)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecane
5-hydroxy-N-(1-methylpiperidin-4-yl)-N-(pyridin-3-ylmethyl)pyrazine-2-carboxamide
methyl 3-({4-[hydroxy(1-methyl-1H-imidazol-2-yl)methyl]piperidine-1-carbonyl}amino)benzoate
3-[(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)(propan-2-yl)amino]propanamide
N-({1-[2-(2-fluorophenyl)ethyl]piperidin-4-yl}methyl)-N,6-dimethylpyridine-2-carboxamide
1-(2-cyclooctyl-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl)-N-methyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]piperidine-4-carboxamide
4-methyl-2-{1-[1-(propan-2-yl)-1H-pyrazole-4-carbonyl]piperidin-3-yl}-1H-1,3-benzodiazole
(4aR,7aS)-1-methyl-4-(2-{5H,6H,7H-[1,3]thiazolo[3,2-a]pyrimidin-3-yl}acetyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
8-{1-phenylspiro[2.4]heptane-1-carbonyl}-2,8-diazaspiro[4.5]decan-3-one
N-methyl-2-{3-oxo-1-[5-(phenoxymethyl)-1H-pyrazole-3-carbonyl]piperazin-2-yl}acetamide
N4-methyl-6-(morpholin-4-yl)-N4-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}pyrimidine-2,4-diamine
3-(3,4-diethyl-1-methyl-1H-pyrazol-5-yl)-1-[2-(5-methyl-1,3,4-thiadiazol-2-yl)ethyl]urea
3-{5-[3-(piperidin-1-yl)propanoyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanoic acid
5-(quinolin-3-yl)-2,3-dihydro-1λ6-thiophene-1,1-dione
5-[1-(3,5-dimethylbenzoyl)piperidin-4-yl]-5-(3-methylbutyl)-3-(pyridin-2-ylmethyl)imidazolidine-2,4-dione
4-[1-(7-methanesulfonyl-4-methylquinazolin-2-yl)piperidin-4-yl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
5-acetyl-N-ethyl-N-[2-(morpholin-4-yl)ethyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
methyl 1-[3-(4-{[ethyl(2-methylprop-2-en-1-yl)amino]methyl}phenoxy)-2-hydroxypropyl]piperidine-4-carboxylate
1-{4-[(3-ethoxy-4-methoxyphenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}-2-phenylethan-1-ol
N-[3-(4-methylpiperazin-1-yl)propyl]-2-oxo-6-(propan-2-yl)-1,2-dihydropyridine-3-carboxamide
N-(2-{5-[(2-methoxyethyl)sulfanyl]-4-methyl-4H-1,2,4-triazol-3-yl}ethyl)-2-(2-phenyl-1,3-thiazol-4-yl)acetamide
1-{[4-(difluoromethoxy)phenyl]methyl}-2-[2-(pyrrolidin-1-yl)ethyl]piperidine
7-(1-aminocyclobutanecarbonyl)-N,N-dimethyl-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
(3aR,6aR)-2-[(4-butylphenyl)methyl]-5-methanesulfonyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
3-(4-aminopyridin-2-yl)-N-butylbenzamide
7-(2-methoxyphenyl)-2-(1H-1,2,4-triazol-5-yl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
2-(pyridin-3-yl)-1-[(1S,5R)-3-(pyrimidin-2-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
5-(methoxymethyl)-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]thiophene-2-carboxamide
3-({[(1,5-dimethyl-1H-indazol-3-yl)methyl]amino}methyl)pyrrolidin-3-ol
(3aR,6aR)-2-[(6-hydroxynaphthalen-2-yl)methyl]-5-methanesulfonyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-[1-methyl-5-(pyridin-4-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl]-1,2,3,4-tetrahydroisoquinoline
3-{2-[4-(4-fluorophenyl)piperazin-1-yl]-2-oxoethyl}-3-(2-methoxyphenyl)-1-(3-methoxypropyl)pyrrolidine-2,5-dione
1-(6-methylpyridin-2-yl)-4-{[3-(2,3,4-trimethoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl}piperazine
7-(3,5-difluoro-4-methoxyphenyl)pyrazolo[1,5-a]pyridine
N-[(3S,4R)-1-(3-oxo-3,4-dihydroquinoxaline-2-carbonyl)-4-(propan-2-yl)pyrrolidin-3-yl]methanesulfonamide
(3aS,6aS)-2-(oxan-4-yl)-5-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
4-(1-{6-phenylimidazo[2,1-b][1,3]thiazole-3-carbonyl}piperidin-4-yl)morpholine
2-{[4-(4-fluorophenyl)-1,2,3,6-tetrahydropyridin-1-yl]methyl}-4-phenylphenol