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N,1-dimethyl-3-(2-methylpropyl)-N-(4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)-1H-pyrazole-5-carboxamide
N-[3-(dimethyl-1,2-oxazol-4-yl)propyl]-6-{[(1R,4S,6S)-spiro[bicyclo[2.2.1]heptane-7,1'-cyclopropan]-2-en-6-ylmethyl]amino}pyridine-3-carboxamide
2-amino-4-ethyl-N-[3-(1H-indazol-1-yl)propyl]-1,3-thiazole-5-carboxamide
7-{thieno[3,2-d]pyrimidin-4-yl}-2-oxa-7-azaspiro[4.5]decane
2-methoxy-4-{[5-(4-methyl-1H-imidazol-5-yl)-4-phenyl-1H-imidazol-1-yl]methyl}phenol
ethyl 3-benzyl-1-[(3-ethoxy-3-oxopropyl)carbamoyl]piperidine-3-carboxylate
(1S,5R)-6-propyl-3-(1H-pyrrole-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
(3R,9aR)-3-benzyl-8-[(2-fluorophenyl)methyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
3-[2-(3-fluorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]piperidine
{[3-(3-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl}(methyl)[2-(1-methyl-1H-pyrazol-4-yl)ethyl]amine
N-(furan-3-ylmethyl)-N,2-dimethyl-4-phenylpyrimidine-5-carboxamide
(3S,4S)-1-[4,5-dimethyl-2-(1H-pyrrol-1-yl)thiophene-3-carbonyl]-4-(pyrrolidin-1-yl)pyrrolidin-3-ol
N-[1-(2,2-dimethylpropyl)-5-oxopyrrolidin-3-yl]-4-(1H-indol-3-yl)butanamide
5-(2-methylbutanoyl)-1-(3-phenylpropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
2-pentyl-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
[2-ethoxy-5-({[(1-methylpiperidin-3-yl)methyl](2-phenylethyl)amino}methyl)phenyl]methanol
1-[1-methyl-6-(pyridin-3-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]-3-phenylpyrrolidin-3-ol
4-(4-chlorophenyl)-N-(1H-imidazol-2-ylmethyl)butanamide
N-[3-(dimethyl-1,3-thiazol-2-yl)propyl]-3-(4-methoxyphenyl)-1H-pyrazole-5-carboxamide
N-({8-[(2E)-3-phenylprop-2-en-1-yl]-1-oxa-8-azaspiro[4.5]decan-2-yl}methyl)furan-2-carboxamide
1-[3-(1H-1,3-benzodiazol-2-ylmethyl)piperidin-1-yl]-2-[methyl(pyridin-4-ylmethyl)amino]ethan-1-one
methyl 2-(1-{2-[(3-chlorophenyl)methyl]-1,3-benzoxazol-6-yl}-N-methylformamido)acetate
ethyl 1-benzoyl-3-[(2-fluorophenyl)methyl]piperidine-3-carboxylate
prop-2-en-1-yl 2-(5-methoxy-1H-1,3-benzodiazol-2-yl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carboxylate
2-(8-{[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]methyl}-2,4-dioxo-1-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decan-3-yl)acetamide
2-(2-methoxyethoxy)-1-[2-(1-methyl-1H-1,3-benzodiazol-2-yl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-5-yl]ethan-1-one
4-{[1-(2-phenylethyl)piperidin-4-yl]oxy}-N-(1-propylpiperidin-4-yl)benzamide
N-cyclopentyl-N-{[3-methoxy-4-(oxan-2-ylmethoxy)phenyl]methyl}-4-methylbenzamide
5-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}-1-phenyl-1H-1,2,3,4-tetrazole
5-[1-(2,4-dimethylbenzoyl)piperidin-4-yl]-5-ethyl-3-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]imidazolidine-2,4-dione
2-{1-[(3-methoxyphenyl)methyl]-4-{[5-methyl-2-(thiophen-2-yl)-1,3-oxazol-4-yl]methyl}piperazin-2-yl}ethan-1-ol
N-[1-(2-methoxyethyl)-7-[2-(pyridin-3-yl)piperidine-1-carbonyl]-1H-1,3-benzodiazol-5-yl]cyclohexanecarboxamide
2-methyl-N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]-5-sulfamoylbenzamide
2-[2-({1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}amino)-4-(morpholin-4-yl)pyrimidin-5-yl]-2-methylpropanoic acid
1-[4-({4-[2-(2-fluorophenyl)benzoyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}methyl)piperazin-1-yl]ethan-1-one
5-fluoro-2-[1-(6-methylpyridine-2-carbonyl)piperidin-2-yl]-1H-1,3-benzodiazole
3-(3-fluorophenyl)-5-[(1R,2S,3S,4R,5S)-tricyclo[3.2.1.02,4]octane-3-carbonyl]-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine
1-{1-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]piperidin-4-yl}-N-(2-methylpropyl)-1H-1,2,3-triazole-4-carboxamide
N-methyl-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}-2-[5-(pyrrolidin-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]acetamide
3-(3,5-dimethyl-1H-pyrazol-1-yl)-N-[1-(2,2-dimethylpropyl)-5-oxopyrrolidin-3-yl]propanamide
3-[2-(3-methoxyphenyl)ethyl]-1-(1,3-thiazole-4-carbonyl)piperidine
2-fluoro-N-[1-(pyrimidin-2-yl)piperidin-3-yl]-5-sulfamoylbenzamide
2-methyl-4-(4-{[2-(1H-pyrazol-1-ylmethyl)-1,4-oxazepan-4-yl]methyl}phenyl)butan-2-ol
N-(3-hydroxypropyl)-1-(1-{[4-(trifluoromethyl)phenyl]methyl}piperidin-3-yl)-1H-1,2,3-triazole-4-carboxamide
1-(cyclopropylmethyl)-4-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-2-(propan-2-yl)-1,4-diazepane
2-(1-{5-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl}pyrrolidin-2-yl)-1,3-benzothiazole
(3aS,6aR)-3-[3-(morpholin-4-yl)propyl]-5-(pyridine-2-carbonyl)-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
N-(2-{4-[3-methyl-1-(pyridin-2-yl)-1H-1,2,4-triazol-5-yl]phenoxy}ethyl)acetamide
2-(methylamino)-N-[2-(6-oxo-3-phenyl-1,6-dihydropyridazin-1-yl)ethyl]acetamide
[(3R,5R)-1-(1H-1,2,3-benzotriazole-5-carbonyl)-5-(morpholin-4-ylmethyl)piperidin-3-yl]methanol