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N-[2-(3-fluorophenyl)ethyl]-3-{5-[methoxy(phenyl)methyl]-1,3,4-oxadiazol-2-yl}propanamide
1-cyclopropyl-5-oxo-N-{2-[(pyridin-3-yl)amino]ethyl}pyrrolidine-3-carboxamide
3-(5-methyl-1H-1,2,4-triazol-3-yl)-1-[4-(3-phenylpropyl)-1,4-diazepan-1-yl]propan-1-one
2-amino-4-[2-(furan-2-yl)pyrimidin-5-yl]-6-(4-hydroxyphenyl)-5-methylpyridine-3-carbonitrile
3-(cyclohex-3-ene-1-carbonyl)-9-methoxy-N-[(3-methoxyphenyl)methyl]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
[(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)methyl](methyl){[3-(1H-pyrazol-1-yl)phenyl]methyl}amine
N-[(2-fluorophenyl)methyl]-4-hydroxy-N-(2-methoxyethyl)-2-(pyridin-3-yl)pyrimidine-5-carboxamide
5-{2-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carbonyl}-N-(1H-1,2,4-triazol-3-ylmethyl)pyridin-2-amine
N-[2-(4-methyl-1H-imidazol-2-yl)ethyl]-2-{3-oxo-1-[(3-phenoxyphenyl)methyl]piperazin-2-yl}acetamide
2-phenoxy-N-{1-[7-(thiophen-2-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]ethyl}acetamide
N-cyclopropyl-1-[2-(4-methoxyphenyl)ethyl]-5-(1,3-thiazole-4-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N-[(1-ethyl-1H-pyrazol-4-yl)methyl]-N-(2-methoxyethyl)-2-methyl-1-benzofuran-5-carboxamide
6-(furan-3-yl)-2-(3-{[methyl(thiophen-2-ylmethyl)amino]methyl}phenyl)-3,4-dihydropyrimidin-4-one
N4-[2-(benzyloxy)ethyl]-5-ethyl-6-methylpyrimidine-2,4-diamine
4-{[1-(2,5-dimethylphenyl)-3-phenyl-1H-pyrazol-4-yl]methyl}-3-ethylpiperazin-2-one
2-[(5-{[3-(3-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]methyl}pyrimidin-2-yl)amino]acetic acid
(1S,5R)-3-[(4-methoxyphenyl)methyl]-6-(2-methylpyrimidine-5-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
N-[(1R,3R)-3-aminocyclopentyl]-1,1-dioxo-1λ6-thiane-4-carboxamide
N-{[2-(4-methylpiperazin-1-yl)pyridin-3-yl]methyl}-5-(oxolan-2-yl)thiophene-2-carboxamide
4-[4-(3-chloro-5-fluoro-4-methoxyphenyl)-1H-1,2,3-triazol-1-yl]piperidine
methyl N-[2-(4-acetyl-4-phenylpiperidin-1-yl)-2-oxoethyl]carbamate
2-{2-[(4-cyclopentyl-1,4-diazepan-1-yl)methyl]phenyl}-6-(difluoromethyl)-3,4-dihydropyrimidin-4-one
1'-[1-methyl-3-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-yl]spiro[indene-1,4'-piperidine]
N-(pyridin-3-ylmethyl)-1-[1-(pyridine-3-carbonyl)piperidin-4-yl]piperidine-3-carboxamide
(2S,4S)-4-amino-1-[2-(2H-1,3-benzodioxol-5-yloxy)acetyl]-N-ethylpyrrolidine-2-carboxamide
(3S,4R)-3-benzyl-4-methyl-1-(pyrazin-2-yl)piperidin-4-ol
3-[3-(furan-2-yl)-1,2,4-oxadiazol-5-yl]-1-{2-[2-(1H-imidazol-1-yl)ethyl]piperidin-1-yl}propan-1-one
1-[1,3-dioxo-2-(oxolan-2-ylmethyl)-2,3-dihydro-1H-isoindol-4-yl]-N,N-diethylpiperidine-3-carboxamide
4-benzyl-1-{[5-(methoxymethyl)-1,2,4-oxadiazol-3-yl]methyl}pyrrolidin-2-one
N-[(1-methylpiperidin-4-yl)methyl]-N-(2-phenylethyl)-2,3-dihydro-1,4-benzodioxine-6-carboxamide
(3S,4R)-4-(2,3-dimethoxyphenyl)-1-(4-hydroxybenzoyl)pyrrolidine-3-carboxylic acid
N-[1-({1-[(3-methylpyridin-2-yl)methyl]-1,2,5,6-tetrahydropyridin-3-yl}methyl)-1H-pyrazol-5-yl]acetamide
1-[4-(3-acetylphenyl)phenyl]-3-(2-hydroxyethyl)-3-propylurea
2-(2,4-dichlorophenoxy)-N-[2-(pyridin-4-yl)ethyl]acetamide
2-(5-chloro-2-methoxypyridin-4-yl)-N-ethylpyridine-4-carboxamide
N-({1-[(2-methylnaphthalen-1-yl)methyl]piperidin-3-yl}methyl)acetamide
8-acetyl-2-[(1-propyl-1H-imidazol-2-yl)methyl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
N-[(2-fluorophenyl)methyl]-N-(2-methoxyethyl)-2-(2-oxopiperidin-1-yl)acetamide
N-{[(2S,4S)-4-fluoro-1-[3-(5-methylfuran-2-yl)-1H-pyrazole-5-carbonyl]pyrrolidin-2-yl]methyl}methanesulfonamide
1-[9-hydroxy-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-3-(1H-1,2,4-triazol-1-yl)propan-1-one
4-[(2R,3R,6R)-3-(2,3-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]pyrimidin-2-amine
9-[4-(propan-2-yl)-1,3-thiazole-2-carbonyl]-1,4,9-triazaspiro[5.5]undecan-5-one
N-[(4-fluorophenyl)methyl]-3-(1-{[2-methyl-4-(1H-pyrazol-1-yl)phenyl]methyl}piperidin-4-yl)propanamide
1-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]-5-(3,5-dimethyl-1H-pyrazol-4-yl)-4-phenyl-1H-imidazole
2-methyl-6-[3-(1H-pyrazol-3-yl)phenyl]-4-(trifluoromethyl)pyridine
(2S,4S)-1-[(2-chlorophenyl)methyl]-4-{[(2,5-difluorophenyl)methyl]amino}-N-ethylpyrrolidine-2-carboxamide
N-(2-chlorophenyl)-7-(cyclopropylmethyl)-6-oxo-2,7-diazaspiro[4.5]decane-2-carboxamide
5-chloro-N-[(2-ethoxyphenyl)methyl]-2-oxo-N-(prop-2-en-1-yl)-1,2-dihydropyridine-3-carboxamide
1-[(3-fluorophenyl)methyl]-4-(prop-2-en-1-yl)-1,4-diazepan-5-one
4-({1-[2-(2-methoxyethoxy)acetyl]pyrrolidin-3-yl}methyl)benzoic acid