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9-{[5-fluoro-2-(1H-pyrazol-1-yl)phenyl]methyl}-1-methyl-1,4,9-triazaspiro[5.5]undecan-5-one
1-[5-(2-methoxyacetyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl]-2-phenylpropan-1-one
N-(furan-2-ylmethyl)-N-[2-(morpholin-4-yl)ethyl]oxolane-2-carboxamide
2-[3-(3,4-difluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]acetamide
1-{3-[4-(2-methoxyphenyl)piperazin-1-yl]piperidin-1-yl}-3-phenylpropan-1-one
2-(dimethylamino)-2-(2-methylphenyl)-N-{[4-(methylsulfanyl)phenyl]methyl}acetamide
4-[(5-fluoro-3-methyl-1H-indol-2-yl)methyl]-N-(pyridin-2-ylmethyl)piperazine-2-carboxamide
3-(1H-imidazol-2-yl)-1-[1-(2-methoxyphenyl)-1H-pyrazole-4-carbonyl]piperidine
N-{[7-(5-ethyl-1,2-oxazole-3-carbonyl)-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}-2-(phenylsulfanyl)acetamide
1-[(4-fluorophenyl)methyl]-3-(2-hydroxy-2-methylpropyl)-2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carboxylic acid
[(2S,6S)-11-methoxy-4-(pyrazine-2-carbonyl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(9),10,12-trien-6-yl]methanol
N-cycloheptyl-5-cyclohexaneamido-1-(2-methoxyethyl)-1H-1,3-benzodiazole-7-carboxamide
1-(diphenylmethyl)-N-[3-(4-methyl-1,3-thiazol-5-yl)propyl]-1H-1,2,3-triazole-4-carboxamide
{[3-(2H-1,3-benzodioxol-5-yl)-1,2,4-oxadiazol-5-yl]methyl}(methyl){[1-(morpholin-4-yl)cyclohexyl]methyl}amine
1-(4-{[(2R,3R,6R)-3-(3-hydroxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]methyl}thiophen-2-yl)ethan-1-one
N-[3-hydroxy-2-(thiophen-3-ylmethyl)propyl]-1-methyl-1H-indole-6-carboxamide
5-cyclopropyl-N-[2-(dimethylamino)ethyl]-N-({1-[(2-methoxyphenyl)methyl]piperidin-3-yl}methyl)-1,2-oxazole-3-carboxamide
2-methyl-N-(oxolan-2-ylmethyl)-N-(thiophen-3-ylmethyl)propanamide
N-{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N-methyl-3-(trimethyl-1H-pyrazol-4-yl)propanamide
N-[(4-chloro-1-methyl-1H-indazol-3-yl)methyl]-1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carboxamide
5-(2-{[(2-fluorophenyl)methyl]amino}ethyl)-1-{[3-(trifluoromethyl)phenyl]methyl}pyrrolidin-2-one
1-[1'-(1H-pyrrole-3-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]propan-1-one
3-[(dimethylamino)methyl]-1-{4H-thieno[3,2-b]pyrrole-5-carbonyl}pyrrolidin-3-ol
5-[(dimethylamino)methyl]-N-[(2E)-3,7-dimethylocta-2,6-dien-1-yl]furan-2-carboxamide
methyl[(4-methyl-1H-imidazol-2-yl)methyl](2-phenoxypropyl)amine
3-[3-(3-fluoro-4-methoxybenzoyl)piperidine-1-carbonyl]-2H-chromen-2-one
N,N-dimethyl-1-[(5-propylfuran-2-yl)methyl]azepan-4-amine
N-[(1,3-dimethylpyrrolidin-3-yl)methyl]-5-[(quinolin-8-yloxy)methyl]-1,2-oxazole-3-carboxamide
3-{[4-ethyl-5-oxo-3-(piperidin-3-yl)-4,5-dihydro-1H-1,2,4-triazol-1-yl]methyl}-N,N-dimethyl-1,2,4-oxadiazole-5-carboxamide
N-ethyl-4-oxo-N-[(5-propyl-1,2,4-oxadiazol-3-yl)methyl]-1,4-dihydroquinoline-2-carboxamide
N-{[2-(1H-imidazol-1-yl)pyridin-3-yl]methyl}-2-(morpholin-4-yl)-2-(pyridin-3-yl)acetamide
4-(2-cyclopropylacetyl)-1-(propan-2-yl)-6-{[4-(trifluoromethoxy)phenyl]methoxy}-1,4-diazepan-2-one
3-[3-(5-cyclopropyl-1H-pyrazol-1-yl)propyl]-1-(3-methoxy-4-methylphenyl)urea
1-(2-cyclohexylethyl)-N-[2-(1H-indol-1-yl)ethyl]-N-methyl-1H-1,2,3-triazole-4-carboxamide
[1-(1-methyl-1H-indole-3-carbonyl)-3-(3-phenylpropyl)piperidin-3-yl]methanol
[4-(3-chloro-5-methoxybenzoyl)-1,4-oxazepan-6-yl]methanol
2-[1-(4-ethylphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl]pyridine
1-(3,5-dimethyl-2-{1-propyl-1H,4H-pyrazolo[3,4-d]imidazol-5-yl}phenyl)-1H-pyrazole
4-methyl-7-({4-[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]piperazin-1-yl}methyl)-2H-chromen-2-one
2-(3-{[4-(propan-2-yl)phenyl]amino}piperidin-1-yl)ethan-1-ol
2-(3-{[4-(dimethylamino)azepan-1-yl]methyl}phenoxy)acetamide
(3S,4S)-4-(morpholin-4-yl)-1-(5-phenyl-1,2-oxazole-3-carbonyl)pyrrolidin-3-ol
1-(4-fluorophenyl)-4-[9-methoxy-7-(2-methoxyphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]butane-1,4-dione
2-(4-{[4-(1-methyl-1H-indole-2-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl]methyl}piperazin-1-yl)ethan-1-ol
N-{[5-(dimethylcarbamoyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}-1H-indole-6-carboxamide
3-methyl-1-[4-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)phenyl]-3-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]urea
8-[(3-methylphenyl)methanesulfonyl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
2-[(5-methylpyrazin-2-yl)methyl]-8-(2-propoxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
1-{3-[4-(3-chlorophenyl)piperazin-1-yl]piperidin-1-yl}-2-(3-methyl-1H-pyrazol-1-yl)ethan-1-one
1-(3-methoxyphenoxy)-3-({8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2,4,6-tetraen-3-yl}amino)propan-2-ol