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N-[(2R,3R)-1'-(3-chloro-2-fluorobenzoyl)-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]propanamide
4-(1-{[1-(propan-2-yl)-1H-imidazol-2-yl]methyl}piperidine-4-carbonyl)morpholine
4-(4-{[2-(pyrrolidin-1-yl)pyrimidin-5-yl]methyl}piperazin-1-yl)quinazoline
3-({1-[2-(morpholin-2-yl)acetyl]piperidin-4-yl}methyl)-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
1-[3-(hydroxymethyl)-3-(3-methoxypropyl)piperidin-1-yl]-2-(4-methyl-1,4-diazepan-1-yl)ethan-1-one
(3R,9aR)-8-(2-chlorobenzoyl)-3-methyl-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
{[2-(cycloheptanesulfonyl)-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}(methyl)(thiophen-3-ylmethyl)amine
3-{2-[3-(dimethylamino)pyrrolidin-1-yl]ethyl}-8-(1-methyl-1H-pyrazole-4-carbonyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-[2-(dimethyl-1,3-thiazol-2-yl)ethyl]-5-(5-methylfuran-2-yl)-1,2,4-triazin-3-amine
5-(methoxymethyl)-N-[1-methyl-4-(morpholin-4-yl)-1H-indazol-3-yl]furan-2-carboxamide
2,4-dimethoxy-6-(4-{[4-methyl-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}piperidin-1-yl)-1,3,5-triazine
8-cyclopropanecarbonyl-2-(1,3-thiazol-4-ylmethyl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
(1S,5R)-N-(2,4-dimethylphenyl)-3-(pyridin-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane-6-carboxamide
N-{[2-(2,6-dimethylphenoxy)pyridin-3-yl]methyl}-1-ethyl-6-oxopiperidine-3-carboxamide
N-ethyl-5-(methoxymethyl)-N-[(2E)-3-phenylprop-2-en-1-yl]thiophene-2-carboxamide
N-[1-(1H-imidazol-1-yl)-3,3-dimethylbutan-2-yl]-[1,2,4]triazolo[4,3-a]pyridine-7-carboxamide
(2S,4R)-1-(2,3-dihydro-1H-inden-2-yl)-4-{[(4-fluorophenyl)methyl]amino}-N-methylpyrrolidine-2-carboxamide
3-{[(3S,4S)-3,4-bis(hydroxymethyl)pyrrolidin-1-yl]methyl}-2,4-dichlorophenol
N-(2-methylpropyl)-1-[(1s,4s)-4-{[(2,4-dimethoxyphenyl)methyl]amino}cyclohexyl]-1H-1,2,3-triazole-4-carboxamide
N-cyclopropyl-N-ethyl-4-{[1-(2-phenylethyl)piperidin-4-yl]oxy}benzamide
2-benzyl-4-{[5-methyl-2-(thiophen-2-yl)-1,3-oxazol-4-yl]methyl}morpholine
benzyl 4-[3-(4-ethylpiperazin-1-yl)-3-oxopropyl]piperidine-1-carboxylate
1-(4-{4-[3-(benzyloxy)piperidin-1-yl]piperidin-1-yl}benzoyl)-4-ethylpiperazine
N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)piperidin-4-yl]methyl}-2-(1H-pyrazol-1-yl)propanamide
2-{6-chloro-3-[(4-methylpiperazin-1-yl)methyl]imidazo[1,2-a]pyridine-2-carbonyl}-1,2,3,4-tetrahydroisoquinoline
1-cycloheptanecarbonyl-3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidine
3-[1-(3-methylfuran-2-carbonyl)piperidin-3-yl]-N-[4-(trifluoromethyl)phenyl]propanamide
N-[1-(1-{[4-(cyclopentyloxy)phenyl]methyl}piperidin-4-yl)-1H-pyrazol-5-yl]cyclopropanecarboxamide
1-(4-ethyl-5-methylthiophene-3-carbonyl)-4-(1H-pyrazol-1-yl)piperidine-4-carboxylic acid
6-{1-[(2-aminopyridin-3-yl)methyl]piperidin-3-yl}-2-methylpyrimidin-4-ol
methyl 5-[1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylate
1-{1-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]piperidin-4-yl}-3-(pyrrolidine-1-carbonyl)piperidine
[1-(2,3-dihydro-1,4-benzodioxin-6-yl)ethyl](1H-imidazol-4-ylmethyl)methylamine
1-[(2-cyclohexylpyrimidin-5-yl)methyl]azepan-4-amine
4,6-dimethoxy-2-{4-[1-(4-methylpiperazin-1-yl)ethyl]piperidin-1-yl}pyrimidine
1-[3-(2-methylpropyl)-5-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazol-1-yl]butan-2-ol
1-(cyclopropylmethyl)-5-[3-(2-methyl-1H-1,3-benzodiazol-1-yl)propanoyl]-N-(pyridin-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
3-{2-[4-(4-methoxyphenyl)-2-methylpiperazin-1-yl]-2-oxoethyl}-1,3-oxazolidin-2-one
5-tert-butyl-N-{[5-(methoxymethyl)-1,2,4-oxadiazol-3-yl]methyl}-1,3,4-oxadiazol-2-amine
5-(1H-1,3-benzodiazol-1-ylmethyl)-N-[2-(1H-imidazol-4-yl)ethyl]-1H-pyrazole-3-carboxamide
N-{[3-methoxy-4-(oxolan-3-yloxy)phenyl]methyl}-N-(pyridin-3-ylmethyl)-4-(trifluoromethyl)benzamide
N4-[(3S)-1-benzylpyrrolidin-3-yl]-2-(butylsulfanyl)pyrimidine-4,6-diamine
N-[2-(4-chloro-3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-1-cyclopropanecarbonylpiperidine-4-carboxamide
{4-[(2-butyl-5-chloro-1H-imidazol-4-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}methanol
3-(2-{2-azabicyclo[2.2.1]heptan-2-yl}-2-oxoethyl)-3-phenyl-1-(pyridin-4-ylmethyl)pyrrolidine-2,5-dione
4-ethyl-1-methyl-3-[1-(quinolin-8-ylmethyl)piperidin-3-yl]-4,5-dihydro-1H-1,2,4-triazol-5-one
1-[(5-cyclobutyl-1,2,4-oxadiazol-3-yl)methyl]-3-(5-ethyl-1-methyl-1H-1,2,4-triazol-3-yl)urea
1-cyclopentyl-4-(quinolin-4-ylmethyl)piperazin-2-one
4-cyclopropyl-6-{3-[4-(2-methylphenyl)piperazin-1-yl]piperidin-1-yl}pyrimidine
5-{5-[(1-methyl-1H-pyrazol-4-yl)methyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}-3-phenyl-1,2-oxazole