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6-[1-(4-fluorophenyl)-2,2-dimethylcyclopropanecarbonyl]-2-(2-hydroxyethyl)-1H,2H,3H,4H,5H,6H,7H-pyrazolo[3,4-c]pyridin-3-one
2-{2-[(3-fluorophenyl)methyl]morpholine-4-carbonyl}-N,N-dimethylaniline
{[2-(benzylsulfanyl)pyrimidin-5-yl]methyl}(methyl)[1-(pyrazin-2-yl)propan-2-yl]amine
{[1-(3-fluorophenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]sulfamoyl}dimethylamine
N-{[4-methoxy-3-(pyrrolidin-1-ylmethyl)phenyl]methyl}-N-methylthian-4-amine
N-{[2-(3,4-difluorophenoxy)pyridin-3-yl]methyl}-4,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
2-(1-{[1-(3,5,5-trimethylhexyl)piperidin-4-yl]methyl}-1H-1,2,3-triazol-4-yl)ethan-1-ol
N-[(3R,4S)-4-cyclopropyl-1-[(2-ethyl-1,3-thiazol-4-yl)methyl]pyrrolidin-3-yl]cyclobutanecarboxamide
2-[methyl(pyridin-3-ylmethyl)amino]-1-[3-(naphthalene-2-carbonyl)piperidin-1-yl]ethan-1-one
1-[9-(but-3-yn-1-yloxy)-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]pent-4-en-1-one
4-[2-(5-methyl-4-{1H,2H,3H,4H,5H-pyrido[4,3-b]indol-2-ylmethyl}-1H-pyrazol-1-yl)ethyl]morpholine
3-[3-fluoro-5-(propan-2-yloxy)phenyl]-N-methylpyrazin-2-amine
N-[(2S)-1-[4-cyclohexyl-3-oxo-6-(pyridin-4-ylmethoxy)-1,4-diazepan-1-yl]-4-(methylsulfanyl)-1-oxobutan-2-yl]acetamide
(4aS,8aR)-1-(3-hydroxypropyl)-6-(piperidin-4-ylmethyl)-decahydro-1,6-naphthyridin-2-one
2-{2-methyl-2,8-diazaspiro[4.5]decane-8-carbonyl}pyridin-4-amine
(3R,4S)-4-cyclopropyl-1-(6,8-difluoro-2-methylquinolin-4-yl)pyrrolidin-3-amine
(3-{2-[1-(4-methoxy-2-methylbenzoyl)piperidin-4-yl]-1H-imidazol-1-yl}propyl)dimethylamine
methyl 1-oxo-2-(2-propoxyethyl)-1,2-dihydroisoquinoline-7-carboxylate
1-(4-{[(2,1,3-benzothiadiazol-5-ylmethyl)amino]methyl}-2-methoxyphenoxy)-3-(diethylamino)propan-2-ol
1-[(3S,4R)-3,4-dihydroxy-4-methylpiperidin-1-yl]-2-[4-(dimethylamino)phenyl]ethan-1-one
(4-{[2-(1-methylpyrrolidin-2-yl)ethyl]amino}quinazolin-2-yl)methanol
N-(1-{4-[(4-cyclopropyl-1H-1,2,3-triazol-1-yl)methyl]piperidin-1-yl}-3-methyl-1-oxobutan-2-yl)acetamide
5-{1-[(4-methoxy-2,5-dimethylphenyl)methyl]piperidin-4-yl}-5-(3-methylbutyl)imidazolidine-2,4-dione
4-(2,2-dimethyl-2,3-dihydro-1-benzofuran-7-yl)-N-methyl-6-oxo-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridine-3-carboxamide
8-[(1-ethyl-1H-pyrazol-4-yl)sulfonyl]-2-(3-methylbut-2-en-1-yl)-2,8-diazaspiro[4.5]decan-3-one
N-cyclopentyl-2-[2-methyl-4-oxo-1-(oxolan-2-ylmethyl)-4,5,6,7-tetrahydro-1H-indol-3-yl]acetamide
2-methoxy-4-{4-[2-(1H-pyrazol-1-yl)ethyl]piperidin-1-yl}pyridine-3-carbonitrile
3-phenyl-6-{[3-(propan-2-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}pyrazolo[1,5-a]pyrimidine
(1S,3R)-3-amino-N-({5-propyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)cyclopentane-1-carboxamide
1-[1-(2-phenylethyl)piperidin-4-yl]piperidine-3-carboxylic acid
1-(4-chloro-1-methyl-1H-pyrrole-2-carbonyl)-4-(furan-3-carbonyl)-1,4-diazepane
4-{[(3R,5S)-3-(pyrrolidine-1-carbonyl)-5-[3-(trifluoromethyl)phenoxymethyl]piperidin-1-yl]methyl}phenol
3-{5-[2-(2-methoxyphenyl)ethyl]-1,3,4-oxadiazol-2-yl}-1-[4-(piperidin-1-ylmethyl)piperidin-1-yl]propan-1-one
(5S,9aS,9bS)-2-[(3-methoxyphenyl)methyl]-5-(5-methylfuran-2-yl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
1-[(3R,4R)-3-(hydroxymethyl)-4-(morpholin-4-ylmethyl)pyrrolidin-1-yl]-2-[4-(methylsulfanyl)phenyl]ethan-1-one
8-[3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)propyl]-2-(propan-2-yl)-2,8-diazaspiro[5.5]undecan-3-one
(2S,4R)-1-[(3-chlorophenyl)methyl]-4-(cycloheptylamino)-N,N-diethylpyrrolidine-2-carboxamide
2-[4-(2H-1,3-benzodioxol-5-yl)-3-butyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-1-yl]-N-(2-hydroxypropyl)acetamide
2-(4-fluorophenyl)-N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]acetamide
1-(2-aminopyrimidin-4-yl)-4-[(2-chlorophenyl)methyl]piperidine-4-carboxylic acid
N-cyclopentyl-2,5-dimethoxy-N-{[4-methoxy-3-(thiophen-2-ylmethoxy)phenyl]methyl}benzamide
2-(4-fluorophenyl)-N-[3-(pyridin-2-yl)propyl]imidazo[1,2-a]pyridine-6-carboxamide
2-[(4-chlorophenyl)methyl]-8-(3-methylpyridin-2-yl)-2,8-diazaspiro[4.5]decan-3-one
1-methyl-N-{[2-(morpholin-4-yl)pyridin-3-yl]methyl}-1H-pyrazole-5-carboxamide
5-{1-azabicyclo[3.2.1]octan-5-yloxy}quinoline
3-[3-(2-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-carbonyl]-1-(propan-2-yl)pyrrolidine
ethyl 2-[4-(3-cyclopropyl-1H-pyrazole-5-carbonyl)morpholin-3-yl]acetate
6-[(3-fluorophenyl)methoxy]-4-(5-methyl-1H-pyrazole-3-carbonyl)-1-(2-methylpropyl)-1,4-diazepan-2-one
(4S,6R)-4-{[1-(2,3-dihydro-1,4-benzodioxin-6-yl)-3-(propan-2-yl)-1H-1,2,4-triazol-5-yl]methyl}-6-methyl-1,3-diazinane-2-thione
N-[2-(4-chlorophenyl)ethyl]-5-methyl-4-[(oxolan-2-ylmethyl)amino]thieno[2,3-d]pyrimidine-6-carboxamide