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4-chloro-2-{2-[2-(morpholin-4-yl)ethyl]piperidine-1-carbonyl}phenol
N-(1-hydroxypropan-2-yl)-N-methyl-4-{[1-(2-phenylethyl)piperidin-4-yl]oxy}benzamide
1-[(5-methylthiophen-2-yl)methyl]-4-(2-phenoxyethyl)-1,4-diazepan-5-one
3-(3-hydroxy-3-methylbutyl)-N-[2-(4-methyl-1,3-thiazol-2-yl)ethyl]benzamide
2-(4-methyl-2-phenylpyrimidine-5-carbonyl)-2,7-diazaspiro[4.5]decane
N-[(4-chloro-1-methyl-1H-indazol-3-yl)methyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
4-[5-cyclobutyl-3-(pyridin-2-yl)-1H-1,2,4-triazol-1-yl]benzene-1-sulfonamide
4-chloro-N-({5-methanesulfonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)benzamide
(3S)-3-[2-(8-chloroquinolin-2-yl)-1H-imidazol-1-yl]azepan-2-one
1-[4-(benzyloxy)piperidin-1-yl]-2-({3-methyl-[1,2,4]triazolo[4,3-b]pyridazin-6-yl}sulfanyl)ethan-1-one
N-{[2-(diethylamino)pyridin-3-yl]methyl}thiophene-2-carboxamide
1-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-4-(pyridin-3-ylmethyl)-1,4-diazepane
N-{[8-(3-phenylpropyl)-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl}pyrazine-2-carboxamide
methyl 5-{[(2,5-dimethylphenyl)methyl]amino}-3-(2-methoxyacetamido)-1-(3-methylbutyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
1-[(4-acetamidophenyl)methyl]-N-[4-(1H-pyrazol-1-yl)phenyl]piperidine-2-carboxamide
7,7-dimethyl-2-[4-(1H-1,2,4-triazol-1-yl)phenyl]-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
1-(azepan-2-ylmethyl)-3-(4-ethenylphenyl)urea
2-{1-cyclopentyl-4-[(3,5-dimethyl-1H-indol-2-yl)methyl]piperazin-2-yl}ethan-1-ol
5-[4-(4-benzyl-1H-pyrazol-5-yl)piperidine-1-carbonyl]-2-cyclopropylpyrimidine
2-{1-[(3,4-difluorophenyl)methyl]-4-(4-ethyl-5-methylpyrimidin-2-yl)piperazin-2-yl}ethan-1-ol
5-(2,6-dimethylphenoxymethyl)-N-{[1-(2-methoxyethyl)-5-oxopyrrolidin-3-yl]methyl}-1,2-oxazole-3-carboxamide
3-(oxolan-2-ylmethyl)-5-propyl-5-[1-(quinoline-6-carbonyl)piperidin-4-yl]imidazolidine-2,4-dione
2-(2-methoxyphenoxy)-2-methyl-1-[3-(1-methyl-1H-imidazol-2-yl)piperidin-1-yl]propan-1-one
methyl 2-{3-[(3,4-difluorophenyl)amino]piperidine-1-carbonyl}benzoate
1-ethyl-4-({[(2-fluoro-5-methoxyphenyl)methyl](methyl)amino}methyl)pyrrolidin-2-one
{[1-(2-fluorophenyl)-3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}[1-(pyridin-4-yl)propyl]amine
2,3-difluoro-N-methyl-N-[(5-propyl-1H-pyrazol-3-yl)methyl]benzamide
1-(4-{4-[4-(2-methylpropyl)-1H-1,2,3-triazol-1-yl]piperidin-1-yl}piperidin-1-yl)ethan-1-one
N5-(2-methoxyethyl)-N3-methyl-1-(3-methylbutyl)-4-oxo-N3-(2-phenylethyl)-1,4-dihydropyridine-3,5-dicarboxamide
2-(1H-1,3-benzodiazol-2-ylmethoxy)-N-methyl-N-(quinolin-5-ylmethyl)acetamide
1-{3-oxo-2,8-diazaspiro[4.5]decan-8-yl}-2-(1,2,3,4-tetrahydroisoquinolin-2-yl)ethane-1,2-dione
ethyl 4-{1-[2-(methylsulfanyl)benzoyl]piperidin-3-yl}piperazine-1-carboxylate
2-[3-(4-chloro-2-methylbenzoyl)piperidine-1-carbonyl]-4H-chromen-4-one
(butan-2-yl)(pyridin-4-ylmethyl)(quinolin-3-ylmethyl)amine
1-[4-(4-benzyl-6-hydroxy-1,4-diazepan-1-yl)piperidin-1-yl]ethan-1-one
5-ethyl-2-methyl-4-{4-[4-(1H-pyrrole-2-carbonyl)piperazin-1-yl]piperidin-1-yl}pyrimidine
N-{1-[1-(2,3-dihydro-1-benzofuran-5-ylmethyl)piperidin-4-yl]-1H-pyrazol-5-yl}-3-phenoxypropanamide
N-(pyridin-3-ylmethyl)-1-[1-(3,3,3-trifluoropropanoyl)piperidin-4-yl]piperidine-3-carboxamide
2-[3-(2H-1,3-benzodioxol-5-yl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-N-phenylacetamide
N,N-dimethyl-4-[4-(3-{[methyl(quinolin-5-ylmethyl)amino]methyl}phenoxy)piperidin-1-yl]-4-oxobutanamide
N-(1-{4-[4-(hydroxydiphenylmethyl)piperidine-1-carbonyl]phenyl}-1H-pyrazol-4-yl)acetamide
(2S)-1-[2-({[(3-methoxyphenyl)methyl](methyl)amino}methyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl]-2-(methylamino)propan-1-one
3-[3-(1-methoxyethyl)phenyl]-5-[(2-methoxyethyl)sulfamoyl]benzoic acid
1-[1-(1-methyl-3-propyl-1H-pyrazole-5-carbonyl)piperidin-3-yl]-4-(2-methylphenyl)piperazine
1-[2-(4-methoxyphenyl)ethyl]-5-{3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}piperidin-2-one
4-(3-fluorophenoxy)-1-[(3-hydroxy-4-methoxyphenyl)methyl]piperidine-4-carboxylic acid
N,N-dimethyl-6-[4-(1,2,3,4-tetrahydroisoquinolin-2-yl)piperidin-1-yl]-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
[(3R,4R)-4-({[2-(dimethylamino)ethyl](methyl)amino}methyl)-1-(3-methyl-1,2-oxazole-5-carbonyl)pyrrolidin-3-yl]methanol
(3aR,6aR)-2-cyclobutanecarbonyl-5-(1,3-thiazol-2-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
(3S)-3-({1-methyl-6-propyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}amino)azepan-2-one