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N-[(3R,5S)-1-(cyclopropylmethyl)-5-(methylcarbamoyl)pyrrolidin-3-yl]-2-methyl-1,3-benzoxazole-6-carboxamide
N,3-dimethyl-N-[(1-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidin-4-yl)methyl]thiophene-2-carboxamide
4-(4-benzyl-1H-1,2,3-triazol-1-yl)-1-(propane-1-sulfonyl)piperidine
1-{5-[4-methoxy-2-(1H-pyrazol-1-yl)phenyl]furan-2-carbonyl}piperidine
5-{[benzyl(methyl)amino]methyl}-N-(2-hydroxyethyl)-1,2-oxazole-3-carboxamide
4-({3-phenyl-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl}methyl)quinoline
(1R,9aR)-1-{[methyl({[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]methyl})amino]methyl}-octahydro-1H-quinolizin-1-ol
1-[(3-methoxyphenyl)methyl]-4-[2-(methylsulfanyl)pyrimidine-5-carbonyl]piperazin-2-one
N-[2-(2-chlorophenyl)ethyl]-1-(4,7-dimethylquinazolin-2-yl)piperidine-4-carboxamide
6-(dimethylamino)-N-[2-(N-methylmethanesulfonamido)ethyl]pyridine-3-carboxamide
N-[(2,6-dimethoxyphenyl)methyl]-5-{1-[(3-fluorophenyl)methyl]-1H-pyrazol-3-yl}-4-methyl-1,3-thiazol-2-amine
5-cyclobutanecarbonyl-1'-(3,6-dimethylpyrazin-2-yl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
2-[5-(2-methoxyacetyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl]pyridine-3-carbonitrile
(isoquinolin-5-ylmethyl)(propyl)(pyridin-3-ylmethyl)amine
(3R,5S)-5-[(4-methylpiperazin-1-yl)methyl]-N-(2-methylpropyl)-1-(pyridin-4-ylmethyl)piperidine-3-carboxamide
1-[2-(cyclohexylsulfanyl)ethyl]-2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazole
2-(methylamino)-1-[4-(3-phenylpropyl)-1,4-diazepan-1-yl]ethan-1-one
1-[(3-fluorophenyl)methyl]-4-(3-hydroxy-4-methylbenzoyl)piperazin-2-one
1-[(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)methyl]-3-phenylpyrrolidin-3-ol
N-[1-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl)ethyl]-1H-pyrazole-4-carboxamide
N-[2-(3-methoxyphenyl)-1-[1-(1,2,5-thiadiazole-3-carbonyl)piperidin-4-yl]ethyl]-N,1-dimethyl-1H-pyrazole-3-carboxamide
3-[2-(naphthalen-2-ylmethyl)-5-oxopyrrolidin-2-yl]-N-{[3-(trifluoromethoxy)phenyl]methyl}propanamide
N-methyl-N-(quinolin-4-ylmethyl)-5-[4-(1H-1,2,4-triazol-1-yl)phenoxymethyl]-1,2-oxazole-3-carboxamide
9-[(3-methoxyphenyl)methyl]-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
N-(dicyclopropylmethyl)-3-{[4-(propan-2-yl)phenyl]methyl}-1,2-oxazole-5-carboxamide
7-fluoro-N-{2-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]ethyl}quinazolin-4-amine
2-ethyl-N-methyl-N-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]-[1,3]oxazolo[5,4-d]pyrimidin-7-amine
2-phenyl-1-{4-[(2,3,6-trifluorophenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}ethan-1-ol
4-[3-(3-methyl-2-oxo-1,2-dihydroquinoxalin-1-yl)propoxy]benzamide
{3-[(3-methoxyphenyl)methyl]-1-(1-methyl-1,2,3,4-tetrahydroquinoline-6-carbonyl)piperidin-3-yl}methanol
1-[(2-methoxyphenyl)methyl]-3-(1-methyl-1H-imidazol-2-yl)piperidine
(2R,3R,6R)-5-(1,3-dimethyl-1H-pyrazole-4-carbonyl)-3-(4-fluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
N-methyl-2-{4-[methyl(2-phenylethyl)amino]-6-oxo-1,6-dihydropyridazin-1-yl}-N-(1,2-oxazol-3-ylmethyl)acetamide
2-[5-(1-oxo-1,2,3,4-tetrahydroisoquinolin-3-yl)-1-(2-phenylethyl)-1H-1,2,4-triazol-3-yl]acetamide
5-({3-[(2,4-difluorophenyl)methyl]-3-(hydroxymethyl)piperidin-1-yl}methyl)-2-methoxyphenol
5-butanoyl-N-[(4-methoxyphenyl)methyl]-1-(pyridin-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
2-(5-acetylthiophen-3-yl)-N-[(3-methoxyphenyl)methyl]acetamide
3-(5-amino-1H-1,2,4-triazol-3-yl)-1-[4-(2-phenoxyethyl)piperazin-1-yl]propan-1-one
2-(5-benzyl-1,2,4-oxadiazol-3-yl)-7,7-dimethyl-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
2,7-dimethyl-4-[(3-methylthiophen-2-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
3-methyl-8-[4-(piperidin-3-ylmethyl)benzoyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-(2-methyl-1,3-benzothiazol-5-yl)-2-(2-methylphenyl)pyrrolidine-1-carboxamide
N-(2-{4-[(2-fluorophenyl)methyl]morpholin-2-yl}ethyl)-1H-1,2,4-triazole-5-carboxamide
methyl({[2-(propan-2-yl)pyrimidin-4-yl]methyl})[1-(thiophen-2-yl)ethyl]amine
1-{6-hydroxy-4-[(1-methyl-1H-imidazol-2-yl)methyl]-1,4-diazepan-1-yl}ethan-1-one
(2R,3R,6R)-5-(1-methyl-1H-indole-3-carbonyl)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecane
N-{[(1r,4r)-4-(methylcarbamoyl)cyclohexyl]methyl}-1H-pyrazole-4-carboxamide
3-(3-methoxypropyl)-1-[4-(piperidin-1-ylmethyl)benzoyl]piperidine
1-(4-fluorophenyl)-4-(4-{1-[methyl(pyridin-4-ylmethyl)amino]-2-phenylethyl}piperidin-1-yl)butane-1,4-dione
N-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}-N-(oxolan-2-ylmethyl)imidazo[1,2-a]pyridine-6-carboxamide