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N-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-amine
1-[(3R,4S)-3-amino-4-(propan-2-yl)pyrrolidin-1-yl]-3-(3,4-dimethoxyphenyl)propan-1-one
N-[(5-{[(2-fluorophenyl)methyl]sulfanyl}-4-(2-methylpropyl)-4H-1,2,4-triazol-3-yl)methyl]-3-(2-oxopyrrolidin-1-yl)benzamide
3-chloro-N-[2-(dimethylamino)ethyl]-4-{[1-(4,4,4-trifluorobutyl)piperidin-4-yl]oxy}benzamide
N-[(2,4-dimethoxyphenyl)methyl]-3-{1-[3-(pyridin-3-yl)propanoyl]piperidin-3-yl}propanamide
(4aR,7aS)-1-[(4-methyl-1H-imidazol-5-yl)methyl]-4-(2,2,3,3-tetramethylcyclopropanecarbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-[4-(2,3-dihydro-1H-inden-2-yl)-6-hydroxy-1,4-diazepan-1-yl]-2-methoxyethan-1-one
5-(4-chloro-2-methoxyphenoxymethyl)-N-(2,3-dihydroxypropyl)-1,2-oxazole-3-carboxamide
(2R,3R,6R)-5-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-3-(2-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
3-{1-[(3-cyclohexyl-1H-pyrazol-4-yl)methyl]piperidin-3-yl}-4-ethyl-4,5-dihydro-1H-1,2,4-triazol-5-one
2-amino-N-[(3R,5S)-5-(hydroxymethyl)-1-methylpyrrolidin-3-yl]-4-methyl-1,3-thiazole-5-carboxamide
N-[2-(dimethyl-1,3-thiazol-2-yl)ethyl]-2-methyl-2,8-diazaspiro[4.5]decane-3-carboxamide
2-[5-methyl-4-(4-methylpiperazin-1-yl)thieno[2,3-d]pyrimidine-6-carbonyl]-2-azabicyclo[2.2.1]heptane
3-[1-(1-benzylpyrrolidin-3-yl)piperidin-4-yl]-N-[(4-fluorophenyl)methyl]propanamide
methyl 3-acetamido-5-{[(5-methylthiophen-2-yl)methyl]amino}-1-(oxolan-2-ylmethyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
N-[(3R,4S)-4-cyclopropyl-1-methanesulfonylpyrrolidin-3-yl]-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
9-[(2S)-2-amino-3-(4-methoxyphenyl)propanoyl]-2-methyl-2,9-diazaspiro[5.5]undecan-3-one
(1-{[5-methyl-2-(thiophen-2-yl)-1,3-oxazol-4-yl]methyl}-4-(3-phenylpropyl)piperidin-4-yl)methanol
1-{[4-(hydroxymethyl)oxan-4-yl]methyl}-3-[1-(2-methoxyethyl)-2-methyl-1H-indol-5-yl]-1-methylurea
4-ethyl-3-({1-[(3-methylquinoxalin-2-yl)methyl]piperidin-4-yl}methyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
2-(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)-N-methyl-N-[2-(pyridin-4-yl)ethyl]acetamide
N-(3-ethoxypropyl)-1-ethyl-3-(piperidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
N-(1-benzothiophen-2-ylmethyl)-2-[6-oxo-4-(pyrrolidin-1-yl)-1,6-dihydropyridazin-1-yl]acetamide
(1S,5R)-6-{[2-(furan-2-yl)pyrimidin-5-yl]methyl}-3-[(4-methyl-1H-imidazol-5-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
1-{4-[3-(4-benzylpiperidin-1-yl)-3-oxopropyl]piperidin-1-yl}propane-1,2-dione
N-(2H-1,3-benzodioxol-5-ylmethyl)-6-(morpholin-4-ylmethyl)-2-oxo-1,2-dihydropyridine-3-carboxamide
3-butyl-1-methyl-4-{5-[(methylsulfanyl)methyl]furan-2-carbonyl}piperazin-2-one
1-cyclohexyl-4-[2-(2,5-dimethoxyphenyl)acetyl]-6-(pyridin-3-ylmethoxy)-1,4-diazepan-2-one
1-{3-[(4-fluorophenyl)amino]piperidin-1-yl}-3-methylbut-2-en-1-one
3-ethoxy-1-(4-{4-methyl-5-[(4-methylpiperazin-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)propan-1-one
5-methoxy-1-methyl-2-[2-(1,3-thiazol-2-yl)piperidine-1-carbonyl]-1H-indole
N,N-dimethyl-5-({3-[3-(propan-2-yloxy)benzoyl]piperidin-1-yl}methyl)-1,3-thiazol-2-amine
3-({[3-(1H-imidazol-1-yl)propyl]carbamoyl}methyl)-N,N,4-trimethyl-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
1-(1-cyclopropylpropan-2-yl)-4-[4-(2-methylpropyl)-1H-1,2,3-triazol-1-yl]piperidine
(3R)-1-{[2-(3,4-dimethoxyphenyl)-7-methylquinolin-3-yl]methyl}pyrrolidin-3-ol
N-(3-methoxyphenyl)-3-{1-[2-(2-oxo-1,3-oxazolidin-3-yl)acetyl]piperidin-4-yl}propanamide
4-(4-fluorophenyl)-1-{[5-(2-methoxyethyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}-1,2,3,6-tetrahydropyridine
5-[(1-phenyl-1H-1,2,3-triazol-4-yl)methyl]-4H,5H,6H,7H-[1,3]thiazolo[5,4-c]pyridin-2-amine
1-[3-(dimethyl-1,2-oxazol-4-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-2-(4-fluoro-3-methylphenyl)ethan-1-one
1-methyl-9-[2-(pyridin-3-yloxy)acetyl]-1,4,9-triazaspiro[5.5]undecan-5-one
N-[2-(dimethylsulfamoyl)ethyl]-2-[2-(ethylsulfanyl)-1,3-thiazol-4-yl]acetamide
N-(2,1,3-benzoxadiazol-5-ylmethyl)-N-methyloxane-2-carboxamide
ethyl 4-[1-(5-propylpyrimidin-4-yl)piperidin-4-yl]piperazine-1-carboxylate
1-ethyl-2-oxo-3-[2-(pyridin-2-yl)ethyl]-1H,2H,3H-imidazo[4,5-b]pyridine-6-carboxylic acid
2-{4-[(2-fluorophenyl)methyl]-1-[(2-methylphenyl)methyl]piperazin-2-yl}ethan-1-ol
4-(5-methyl-1,2,4-oxadiazol-3-yl)-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
3-(2-chlorophenyl)-N-[(4-hydroxy-1-methylpiperidin-4-yl)methyl]-3-phenylpropanamide
N-{[5-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N-methyl-1-(propan-2-yl)piperidine-4-carboxamide
2-{1-[(3-benzyl-1,2,4-oxadiazol-5-yl)methyl]piperidin-4-yl}-1,2,3,4-tetrahydroisoquinoline
(7S,9aR)-N-cyclohexyl-7-(hydroxymethyl)-6,9-dioxo-octahydro-1H-pyrazino[1,2-a]piperazine-2-carboxamide