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3-{1-[3-(pyridin-4-yl)propanoyl]piperidin-3-yl}-N-[4-(trifluoromethyl)phenyl]propanamide
N-(1,4-dioxan-2-ylmethyl)-1-{1-[(2-methylphenyl)methyl]piperidin-4-yl}piperidine-4-carboxamide
3-fluoro-5-[4-(2-methylphenyl)-3-oxopiperazine-1-carbonyl]benzonitrile
2-[1-(furan-3-ylmethyl)-4-(2-methylpropyl)piperazin-2-yl]ethan-1-ol
5-{4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperidine-1-carbonyl}-2-(pyridin-4-yl)pyrimidine
4-[(2,3-difluoro-4-methylphenyl)methyl]-2-(pyridin-3-yl)morpholine
1-{4-[2-(4-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl]piperidin-1-yl}ethan-1-one
ethyl 4-{3-methoxy-4-[(1-methylpiperidin-4-yl)oxy]benzamido}piperidine-1-carboxylate
2-(morpholin-3-yl)-1-[4-(3-phenylpropyl)-1,4-diazepan-1-yl]ethan-1-one
(1S,5R)-3-[(3-ethyl-1,2-oxazol-5-yl)methyl]-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N,5,7-trimethyl-N-[3-(phenylsulfanyl)propyl]-[1,2,4]triazolo[4,3-a]pyrimidine-3-carboxamide
3-(1-methylpiperidin-2-yl)-N-[2-(1,3-thiazol-2-yl)ethyl]propanamide
1-(3-methoxypiperidin-1-yl)-2-(2,5,7-trimethyl-1H-indol-3-yl)ethan-1-one
N-{[7-chloro-5-(thiophen-3-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-3-[(1,1-dioxo-1λ6-thiolan-3-yl)(methyl)amino]propanamide
3-(2,2-dimethyloxan-4-yl)-3-ethyl-1-(4-fluoro-2-methylphenyl)urea
2-[3-(dimethyl-1,2-oxazol-4-yl)-1H-indazol-1-yl]-N-(2-methyl-2H-1,2,3-triazol-4-yl)acetamide
2-[(4aR,7aS)-4-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]acetic acid
1-methyl-4-({5-[1-(1H-pyrazol-1-yl)propyl]-1,2,4-oxadiazol-3-yl}methyl)piperidine
(2S,4S)-4-amino-N-ethyl-1-(4,5,6,7-tetrahydro-2-benzothiophene-1-carbonyl)pyrrolidine-2-carboxamide
N-methyl-N-({1-[2-(2-methylphenyl)ethyl]piperidin-3-yl}methyl)-1H-indole-2-carboxamide
2-[1-(2,2-dimethylpropyl)-4-[(2-methylphenyl)methyl]piperazin-2-yl]ethan-1-ol
2-(ethanesulfonyl)-N-({1-[2-(3-fluorophenyl)ethyl]piperidin-4-yl}methyl)-N-methylacetamide
5-cyclopropyl-1-[4-(2,5-dimethoxyphenyl)pyrimidin-2-yl]-N-(oxolan-3-yl)-1H-pyrazole-4-carboxamide
3-(6-methoxynaphthalene-2-carbonyl)-1-[2-(1H-pyrazol-4-yl)ethyl]piperidine
2-({[(3R,4R)-4-(hydroxymethyl)-1-(4-methoxy-3,5-dimethylbenzoyl)pyrrolidin-3-yl]methyl}(methyl)amino)ethan-1-ol
6-{3-[4-(4-fluorophenyl)piperazin-1-yl]piperidine-1-carbonyl}-2-methyl-2,3-dihydropyridazin-3-one
(1S,5R)-3-[2-(3-fluorophenoxy)acetyl]-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
(1S,5R)-N-ethyl-N-methyl-7-oxo-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane-3-sulfonamide
3-{1-[4-(1H-pyrazol-3-yl)benzoyl]pyrrolidin-2-yl}pyridine
N-[2-(dimethylamino)-5,6,7,8-tetrahydroquinazolin-5-yl]-2-(2-methyl-1H-indol-3-yl)acetamide
1-[(3-methylpyridin-2-yl)methyl]-4-(5-propyl-1,2-oxazole-4-carbonyl)piperazine
N-[3-(1H-indol-1-yl)propyl]-2-(4-methyl-1,4-diazepan-1-yl)acetamide
3-{[1-(4-fluorophenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}-1H-pyrazole
4-{1-[(1,3-dimethyl-1H-pyrazol-4-yl)sulfonyl]piperidin-3-yl}benzoic acid
1-ethyl-N,N-bis(1,3-oxazol-4-ylmethyl)piperidine-2-carboxamide
N-({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)-N-(2-methoxyethyl)-2-(2-oxo-1,3-oxazolidin-3-yl)acetamide
N-({1-[2-(2-methoxyphenyl)ethyl]piperidin-4-yl}methyl)-N-methyl-2-(5-oxopyrrolidin-2-yl)acetamide
3-{5-[(4-phenylphenyl)methyl]-1,3,4-oxadiazol-2-yl}-1-(thiomorpholin-4-yl)propan-1-one
2-({3-[2-(2,4-difluorophenyl)ethyl]piperidin-1-yl}methyl)-3,5-dimethyl-1,4-dihydropyridin-4-one
(3aR,6aR)-2-acetyl-5-({9-methyl-4-oxo-4H-pyrido[1,2-a]pyrimidin-2-yl}methyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-(4-chlorophenyl)-3-cyclopropyl-5-{5-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-3-yl}-1H-1,2,4-triazole
6-methyl-2-oxo-N-{2-[3-(pyridin-3-yl)-1H-1,2,4-triazol-5-yl]ethyl}-1,2-dihydropyridine-4-carboxamide
2-{[2-(azepan-1-yl)ethyl](methyl)amino}-N-(2,3-dimethylphenyl)acetamide
2-[4-(2,6-dimethoxypyridin-3-yl)-3,5-dimethyl-1H-pyrazol-1-yl]acetamide
N-[1-(4-chlorophenyl)ethyl]-4-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}benzamide
(2S,4R)-4-amino-1-[3-(3-methoxyphenoxy)propyl]-N-methylpyrrolidine-2-carboxamide
N-[1-(cyclohexylmethyl)piperidin-3-yl]-2,6-dimethylpyrimidine-4-carboxamide
(1S,5R)-1,3,3-trimethyl-N-{[1,2,4]triazolo[4,3-a]pyridin-8-yl}-6-azabicyclo[3.2.1]octane-6-carboxamide
1-(2,3-difluoro-4-methoxybenzoyl)-4-phenyl-1,4-diazepane
2-(4-methylpiperazin-1-yl)-N-(2-methylpropyl)-N-(3-phenylprop-2-yn-1-yl)propanamide