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N-[(3,5-dimethyl-4,5-dihydro-1,2-oxazol-5-yl)methyl]-3-(2-methylpropyl)-1,2-oxazole-5-carboxamide
2-[(2H-1,3-benzodioxol-5-yloxy)methyl]-N-(1-phenylcyclopropyl)-1,3-oxazole-4-carboxamide
1-{2-[2-(trifluoromethyl)phenyl]pyrimidin-4-yl}pyrrolidin-3-ol
(3aR,6aS)-N-[2-(3-methoxyphenyl)phenyl]-octahydropyrrolo[3,4-c]pyrrole-2-carboxamide
N-(2-ethyl-2H-1,2,3-triazol-4-yl)-2-[4-(1,3-thiazol-2-yl)-1H-pyrazol-1-yl]acetamide
(3aR,5S,6S,7aS)-N-(2-chloro-4,6-dimethylphenyl)-5,6-dihydroxy-octahydro-1H-isoindole-2-carboxamide
N-[(1,2-dimethyl-1H-1,3-benzodiazol-5-yl)methyl]-2-(dimethylamino)-2-(3-fluorophenyl)acetamide
N-(2-chlorophenyl)-3-[1-(3-phenylpropyl)piperidin-4-yl]propanamide
4-(1-tert-butyl-1H-pyrrole-3-carbonyl)-2-ethyl-1-(propan-2-yl)piperazine
1-[(3,5-dimethyl-4-oxo-1,4-dihydropyridin-2-yl)methyl]-3-(2-methoxyethyl)piperidine-3-carboxylic acid
4-[1-(propan-2-yl)-1H-pyrazole-4-carbonyl]thiomorpholine
1-[1-(2-chloro-6-fluorophenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]but-2-yn-1-one
(3aS,6aR)-3-cyclopentyl-5-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
2-{4-[(2-fluorophenyl)methyl]morpholin-3-yl}-N-[2-(4-methyl-1H-1,2,3-triazol-1-yl)ethyl]acetamide
3-(2-fluorophenyl)-1-(2-methoxyethyl)-3-{2-[3-(morpholine-4-carbonyl)piperidin-1-yl]-2-oxoethyl}pyrrolidine-2,5-dione
(3R,5R)-N-[2-(benzyloxy)ethyl]-5-(pyrrolidine-1-carbonyl)piperidine-3-carboxamide
1-{[2-(furan-3-yl)-5-methyl-1,3-oxazol-4-yl]methyl}-2-[2-(1H-pyrazol-1-yl)ethyl]piperidine
8-[2-(2,5,7-trimethyl-1H-indol-3-yl)acetyl]-1,3-dioxa-8-azaspiro[4.5]decan-2-one
5-{3-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carbonyl}-1,2-dihydropyridin-2-one
(2R,3R)-1'-(5-cyclopropyl-1,3-oxazole-4-carbonyl)-3-(dimethylamino)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
2-(3-methoxypropyl)-8-(5-propyl-1,2-oxazole-4-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
(3aR,6aR)-2-(cyclobutylmethyl)-5-[(8-methylquinolin-5-yl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-(4-fluorophenyl)-4-[1-(pyridine-2-carbonyl)piperidin-3-yl]piperazine
(2S,4R)-4-(1H-1,3-benzodiazol-2-ylsulfanyl)-1-[(2Z)-2-chloro-3-phenylprop-2-en-1-yl]-N-cyclopropylpyrrolidine-2-carboxamide
1-[2-benzyl-4-(4-methylphenyl)-5-oxopiperazin-1-yl]butane-1,2-dione
3-[2-(3-cyclopropyl-1,2,4-oxadiazol-5-yl)ethyl]-1-[2-(5-methylfuran-2-yl)phenyl]urea
1-methyl-4-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
3-chloro-4-{[1-(1-ethylpiperidin-4-yl)piperidin-4-yl]oxy}-N-(2-methoxyethyl)benzamide
2-(3-hydroxypropyl)-8-[(2E)-3-phenylprop-2-en-1-yl]-2,8-diazaspiro[5.5]undecan-3-one
N-methyl-N-({1-[2-(2-methylphenyl)ethyl]piperidin-3-yl}methyl)-3-phenyl-1,2-oxazole-5-carboxamide
N-{[3-(4-chlorophenyl)-1H-pyrazol-4-yl]methyl}-4-methyl-5-[1-(oxan-2-ylmethyl)-1H-pyrazol-3-yl]-1,3-thiazol-2-amine
3-{3-[3-(4-fluorophenyl)oxolan-3-yl]-1,2,4-oxadiazol-5-yl}-2-methoxypyridine
5-{5-[3-(2-methylpropyl)-1,2-oxazol-5-yl]-1,2,4-oxadiazol-3-yl}-1H-1,3-benzodiazole
3-(3,4-dimethyl-1H-pyrazol-5-yl)-1-{7-[(2-fluoro-5-methoxyphenyl)methyl]-2,7-diazaspiro[4.5]decan-2-yl}propan-1-one
N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-3-[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]propanamide
N-[2-(3,4-dimethoxyphenyl)ethyl]-N-methyl-1-(pyridin-4-ylmethyl)piperidin-3-amine
N-(isoquinolin-5-ylmethyl)-N-methylpyrazolo[1,5-a]pyridine-3-carboxamide
({2-[(2-chlorophenyl)methoxy]-6-methylquinolin-3-yl}methyl)[(1-methyl-1H-pyrazol-4-yl)methyl]amine
1'-(1,7-dimethyl-1H-indole-2-carbonyl)-5-methyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
N-(propan-2-yl)-2-[4-(pyridin-3-ylmethoxy)piperidin-1-yl]pyridine-4-carboxamide
4-methyl-N-[(2,3,5-trimethyl-1H-indol-7-yl)methyl]-1,2,3-thiadiazole-5-carboxamide
4-(6-{3-[1-(2-methoxyethyl)-1H-pyrazol-3-yl]phenyl}pyrazine-2-carbonyl)morpholine
N-[(3S,4R)-1-{2,7-dimethylpyrazolo[1,5-a]pyrimidine-5-carbonyl}-4-(propan-2-yl)pyrrolidin-3-yl]methanesulfonamide
N-[3-(2,3-dihydro-1H-indol-1-yl)propyl]-5-methoxy-1-methyl-1H-indole-2-carboxamide
N-(pyridin-3-ylmethyl)-4-(4-{[2-(thiophen-2-yl)ethyl]amino}piperidin-1-yl)benzamide
3-[4-(3-methylphenyl)piperazin-1-yl]-N-[(5-methylthiophen-2-yl)methyl]propanamide
8-methoxy-2-[2-(methylsulfanyl)pyrimidin-5-yl]quinoline
N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-4-(2-methyl-2H-1,2,3,4-tetrazol-5-yl)benzamide
4-{[1-(2-methoxyacetyl)piperidin-4-yl]oxy}-N-[2,2,2-trifluoro-1-(furan-2-yl)ethyl]benzamide
N6-cyclopropyl-N5-(oxolan-2-ylmethyl)-N5-(pyridin-2-ylmethyl)-[1,2,5]oxadiazolo[3,4-b]pyrazine-5,6-diamine