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2-{1-[(4-methoxy-3-methylphenyl)methyl]-3-oxopiperazin-2-yl}-N-(2-methoxyethyl)acetamide
3-(4-{[3-(thiophen-2-yl)-1,2,4-oxadiazol-5-yl]methyl}piperazin-1-yl)-1λ6-thiolane-1,1-dione
N-({7-[2-(2-methoxyphenyl)acetyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)thiophene-3-sulfonamide
5-(2H-1,3-benzodioxol-5-yl)-3-{[4-(oxolan-3-yl)-1H-1,2,3-triazol-1-yl]methyl}-1,2,4-oxadiazole
5-({[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl](methyl)amino}methyl)-N,N-dimethylpyrimidin-2-amine
N-[1-(2,3-dihydro-1H-inden-2-yl)-5-oxopyrrolidin-3-yl]-2-ethylbenzamide
(2S,4S)-4-(4-cyclohexyl-1H-1,2,3-triazol-1-yl)-N,N-diethylpyrrolidine-2-carboxamide
5-[(1R,5R)-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]-2-phenyl-2,3-dihydro-1H-pyrazol-3-one
2-(1-{[3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}piperidin-3-yl)-1,2,3,4-tetrahydroisoquinoline
4-chloro-N-{[2-(diethylamino)pyridin-3-yl]methyl}-1,3-dimethyl-1H-pyrazole-5-carboxamide
2-[(1H-imidazol-2-ylmethyl)(methyl)amino]-2-{4-[(morpholine-4-carbonyl)amino]phenyl}acetic acid
N-(3-chloro-4-propanamidophenyl)-2-(2-oxopyrrolidin-1-yl)propanamide
N-({8-[(2E)-3-[4-(dimethylamino)phenyl]prop-2-en-1-yl]-1-oxa-8-azaspiro[4.5]decan-2-yl}methyl)furan-2-carboxamide
2-({4-[1-(3-methylphenyl)-1H-pyrazol-4-yl]pyrimidin-2-yl}amino)ethan-1-ol
(2S)-2-{[2-(ethylamino)pyrimidin-5-yl]formamido}-2-phenylacetamide
2,6-dimethyl-3-{1-methyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazine-2-carbonyl}imidazo[1,2-a]pyridine
4-[3-(pyridin-2-yl)azetidine-1-carbonyl]-1-oxaspiro[4.4]nonan-2-one
2-[(1-cyclopentylpiperidin-4-yl)oxy]-5-methoxy-N-[3-(1H-pyrazol-1-yl)propyl]benzamide
1-({2-methylpyrido[2,3-d]pyrimidin-4-yl}amino)cyclopentane-1-carboxamide
(3S,5S)-1-(2,3-dihydro-1H-inden-2-yl)-5-(6,7-dimethoxy-1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-N-(2-methylpropyl)pyrrolidin-3-amine
[(3R,4R)-4-(piperidin-1-ylmethyl)-1-[4-(propan-2-yloxy)benzoyl]pyrrolidin-3-yl]methanol
5-methyl-N-[(1S,2R)-2-{[1-(pyridine-4-carbonyl)piperidin-4-yl]amino}cyclobutyl]thiophene-3-carboxamide
N-(naphthalen-1-ylmethyl)-2-{[4-(pyrimidin-2-yl)piperazin-1-yl]methyl}-1,3-oxazole-4-carboxamide
1-[(3R,4S)-3-amino-4-propylpyrrolidin-1-yl]-3-(2-methyl-1H-imidazol-1-yl)propan-1-one
methyl 3-{[(2-methyl-1,3-thiazol-4-yl)formamido]methyl}-5-[3-(trifluoromethyl)benzamido]benzoate
2-methoxy-5-({[1-(1-methyl-1H-pyrazol-5-yl)propyl]carbamoyl}amino)benzamide
(3aS,6aS)-2-pentyl-5-[2-(1,3-thiazol-5-yl)acetyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
5-(3-{4-[(3-methoxyphenyl)methyl]-3-oxopiperazin-1-yl}-3-oxopropyl)imidazolidine-2,4-dione
N-(2,1,3-benzoxadiazol-5-ylmethyl)-N-methyl-5-[(5,6,7,8-tetrahydronaphthalen-2-yloxy)methyl]-1,2-oxazole-3-carboxamide
(2E)-N-[1-(5-{[2-(4-fluorophenoxy)ethyl]sulfanyl}-4-methyl-4H-1,2,4-triazol-3-yl)ethyl]-3-(4-methoxyphenyl)prop-2-enamide
1-(dimethyl-1,3-oxazole-5-carbonyl)-4-(4-methoxybenzoyl)piperazine
N-butyl-2-fluoro-N-(pyridin-4-ylmethyl)-5-sulfamoylbenzamide
methyl 1-ethoxy-2-oxo-8-(3-oxo-2,3-dihydro-1H-indene-1-carbonyl)-1,8-diazaspiro[4.5]decane-4-carboxylate
2-(2-{4-[(4-fluorophenyl)methyl]piperazin-1-yl}-2-oxoethyl)-2,3-dihydro-1H-indazol-3-one
1-ethyl-8-[(8-methoxy-2H-chromen-3-yl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-(2-{5-cyclopropanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-2-oxoethyl)-1,2-dihydropyrimidin-2-one
N-{2-[(furan-2-ylmethyl)(prop-2-en-1-yl)carbamoyl]phenyl}-N-methylthiophene-2-carboxamide
2-(2-aminopyrimidin-5-yl)-N-ethyl-7-fluoro-N-(pyridin-2-ylmethyl)quinoline-4-carboxamide
9-[(2,3-dichlorophenyl)methyl]-2-(2-methoxyethyl)-2,9-diazaspiro[5.5]undecan-3-one
4-[1-(pyrrolidin-1-yl)ethyl]-1-(1H-1,2,4-triazole-5-carbonyl)piperidine
4-(8-methoxyquinolin-2-yl)-N-methyl-1H-pyrrolo[2,3-b]pyridin-6-amine
1-[(3-chloro-1-benzothiophen-2-yl)methyl]-4-(hydroxymethyl)azepan-4-ol
N-{2-[(4-ethyl-5-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}-2-methyl-1,3-benzothiazole-5-carboxamide
1-cyclopentyl-5-[4-(pyrimidin-2-yl)piperazine-1-carbonyl]piperidin-2-one
4-({5-methyl-2-[3-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)thiomorpholine
1-cyclopentyl-N-methyl-5-oxo-N-{[2-(1H-pyrazol-1-yl)phenyl]methyl}pyrrolidine-3-carboxamide
3-[1-(carbamoylmethyl)-1H-imidazol-2-yl]-N-(4-methoxyphenyl)piperidine-1-carboxamide
1-[1-(1-{5-methylthieno[2,3-d]pyrimidin-4-yl}piperidin-4-yl)-1H-1,2,3-triazol-4-yl]ethan-1-ol
2-ethyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-N-propylpyrimidine-5-carboxamide
methyl({[2-(methylsulfanyl)phenyl]methyl}){[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]methyl}amine