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N-{2-[3-(oxolan-3-yl)-1H-1,2,4-triazol-5-yl]propan-2-yl}thiophene-2-carboxamide
N-[2-(2-amino-1,3-thiazol-4-yl)ethyl]-3,5,7-trimethyl-1H-indole-2-carboxamide
(1R,7S)-6-(4-methyl-1,2,3,6-tetrahydropyridine-1-carbonyl)-3-[2-(4-methylphenyl)ethyl]-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-en-4-one
N-[(3R,4S)-1-acetyl-4-propylpyrrolidin-3-yl]-4-(2-oxopyrrolidin-1-yl)benzamide
2-(furan-2-yl)-5-{1-[(4-methylphenyl)methyl]-1H-1,2,3-triazol-4-yl}pyrimidine
6-chloro-N-[(1-methylpiperidin-4-yl)methyl]-N-(2-phenylethyl)imidazo[1,2-a]pyridine-2-carboxamide
4-{[1-(2-methoxyacetyl)piperidin-4-yl]oxy}-N-[(5-methylpyrazin-2-yl)methyl]benzamide
4-(2-methylpyrrolidine-1-carbonyl)-1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperidine
4-(2-fluorophenyl)-N-(1H-imidazol-2-ylmethyl)benzamide
N-ethyl-N-({1-[2-(3-methoxyphenyl)ethyl]piperidin-3-yl}methyl)pent-4-enamide
5-acetyl-N-{2-[(3-methylpyridin-2-yl)amino]ethyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
4-(4-ethyl-1,2,3-thiadiazole-5-carbonyl)-2-[(4-methoxyphenyl)methyl]morpholine
N-cyclopropyl-N-{[3-(2-methylpropoxy)phenyl]methyl}acetamide
1-{9-[2-(4-methyl-1,3-thiazol-5-yl)ethoxy]-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl}pent-4-en-1-one
3-{3-[2-(2-fluorophenyl)ethyl]piperidine-1-carbonyl}-1,4,6-trimethyl-1,2-dihydropyridin-2-one
N-(5-fluoro-2-methoxyphenyl)-6-hydroxy-1,4-oxazepane-4-carboxamide
1-[4-(2-methyl-1H-imidazol-1-yl)phenyl]-N-[(2R)-3-methylbutan-2-yl]piperidin-4-amine
2-{3-[3-(4-cyclopropanecarbonylphenyl)phenyl]-1H-pyrazol-1-yl}ethan-1-ol
2-(furan-2-yl)-4-({8-methoxy-1H,2H,3H,4H,5H-pyrido[4,3-b]indol-2-yl}methyl)-5-methyl-1,3-oxazole
5-(2-chloro-4-methoxyphenoxymethyl)-N-(2-oxopyrrolidin-3-yl)-1H-pyrazole-3-carboxamide
5-benzyl-5-{1-[(2-methoxyphenyl)methyl]piperidin-4-yl}-3-[2-(pyridin-2-yl)ethyl]imidazolidine-2,4-dione
8-[2-(2-hydroxyphenyl)acetyl]-3-methyl-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
2-[benzyl(methyl)amino]-N-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-2,3-dihydro-1H-indene-2-carboxamide
N-tert-butyl-3-{2-phenyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}propanamide
N-benzyl-1-(cyclohexylmethyl)-6-oxopiperidine-3-carboxamide
1-(4-cyclopentyl-1,4-diazepan-1-yl)-2-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethan-1-one
2-(2-{[(oxolan-2-ylmethyl)(thiophen-3-ylmethyl)amino]methyl}phenoxy)acetamide
5-[(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)methyl]-3-(2-methoxyethyl)-1,2,4-oxadiazole
N-(1-{1-[(3-methoxyphenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-3-phenoxypropanamide
1-[(1S,5R)-3-benzoyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-3-(pyridin-2-yl)propan-1-one
6-(4-methoxyphenyl)-7-methyl-N-[2-(methylamino)ethyl]-8-oxo-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
2-[(4-methoxyphenyl)methyl]-4-(pyridin-4-ylmethyl)morpholine
N-(1-{7-[(4-methoxynaphthalen-1-yl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}-3-methylbutyl)furan-2-carboxamide
2-[1-(furan-2-ylmethyl)-1H,4H-pyrazolo[3,4-d]imidazol-5-yl]-1-(4-methoxyphenyl)-1H-imidazole
6-(3-fluorophenyl)-N-[1-(pyridin-3-yl)propan-2-yl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
5-[(4-benzyl-3-ethyl-5-oxo-1,4-diazepan-1-yl)methyl]-N-methyl-1,2,4-oxadiazole-3-carboxamide
5-methyl-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-3-phenyl-1,2-oxazole-4-carboxamide
5-[1-(1-benzofuran-2-ylmethyl)piperidin-4-yl]-3-(2,3-dihydro-1H-inden-2-yl)-5-methylimidazolidine-2,4-dione
2-(cyclopropylmethyl)-7-[(2-fluorophenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
1-[4-(2H-1,3-benzodioxol-5-ylmethyl)piperazin-1-yl]-2-[(6-{[(4-fluorophenyl)methyl](methyl)amino}pyridazin-3-yl)oxy]ethan-1-one
{[2-(3,4-difluorophenoxy)pyridin-3-yl]methyl}(pentan-2-yl)amine
(3S,4R)-1-[6-(methoxymethyl)pyridine-2-carbonyl]-4-(pyridin-3-yl)pyrrolidine-3-carboxylic acid
1-[(2R,3S,6R)-3-(2H-1,3-benzodioxol-5-yl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]butane-1,2-dione
2-(pyridin-4-yl)-1-{4-[4-(pyrrolidine-1-carbonyl)phenoxy]piperidin-1-yl}ethan-1-one
2-amino-4-[4-methoxy-3-(1H-1,2,4-triazol-1-ylmethyl)phenyl]-5,6,7,8-tetrahydro-1,6-naphthyridine-3-carbonitrile
5-({3-[(1S,9aR)-octahydro-1H-quinolizin-1-yl]propanamido}methyl)-1,2,4-oxadiazole-3-carboxamide
N-(2,3-dihydroxypropyl)-5-(3-fluorophenoxymethyl)-1H-pyrazole-3-carboxamide
4-methyl-2-(pyridin-3-yl)-N-[2-(pyrrolidin-1-yl)ethyl]pyrimidine-5-carboxamide
4-({2-[1-(4-ethyl-2-methyl-1,3-thiazole-5-carbonyl)piperidin-4-yl]-1H-imidazol-1-yl}methyl)pyridine
4-({2-[1-(5-ethyl-1,3-oxazole-4-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}methyl)pyridine