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N-({2-methylimidazo[2,1-b][1,3,4]thiadiazol-6-yl}methyl)-5-(pyrrolidin-2-yl)thiophene-2-carboxamide
9-(5-chloro-2-methylbenzoyl)-2-(oxolan-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
7-(3-chlorophenyl)-4-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
3-{1-[2-(methylsulfanyl)pyridine-3-carbonyl]piperidin-3-yl}-1-(morpholin-4-yl)propan-1-one
2-(2-chlorophenyl)-1-{3-[ethyl(pyridin-4-ylmethyl)amino]piperidin-1-yl}ethan-1-one
N-[(3-chloro-4-fluorophenyl)methyl]-1-(propan-2-yl)-1H-pyrazole-4-carboxamide
6-{4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1,4-diazepane-1-carbonyl}pyridin-3-ol
N-cyclopropyl-2-{4-[(4,6-dimethylpyrimidin-2-yl)amino]piperidin-1-yl}acetamide
N-[(1R,2R)-2-(benzyloxy)cyclopentyl]-3-(trimethyl-1H-pyrazol-4-yl)propanamide
7-(2-aminoethyl)-2-methyl-N-[2-(thiophen-2-yl)ethyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
2-({2-[4-(1H-1,2,3-benzotriazol-1-yl)piperidine-1-carbonyl]phenyl}amino)acetic acid
4-[(2,6-dimethylpyridin-3-yl)oxy]-1-[2-(1,3-thiazol-4-yl)acetyl]piperidine-4-carboxylic acid
[1-(1-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}piperidin-4-yl)piperidin-3-yl]methanol
3-(4-fluorophenyl)-5-[(2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazol-1-yl)methyl]-1,2,4-oxadiazole
5-[(2-chlorophenyl)methyl]-5-[1-(cyclohex-3-ene-1-carbonyl)piperidin-4-yl]-3-(2-methoxyethyl)imidazolidine-2,4-dione
3-{3-cyclopropyl-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-6-yl}-1,5-dimethyl-1H-indazole
1-cyclopentanecarbonyl-N-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]piperidine-4-carboxamide
({1-[2-(4-chlorophenyl)ethyl]piperidin-3-yl}methyl)[(1-ethyl-1H-pyrazol-4-yl)methyl]methylamine
methyl 4-{[4-ethyl-5-oxo-3-(piperidin-4-ylmethyl)-4,5-dihydro-1H-1,2,4-triazol-1-yl]methyl}benzoate
N-({1-[(2-cyanophenyl)methyl]piperidin-3-yl}methyl)but-3-enamide
2-(dimethylamino)-N-({2-[3-(trifluoromethyl)phenoxy]pyridin-3-yl}methyl)butanamide
N-[2-(propan-2-yl)-2H-1,2,3-triazol-4-yl]-2-{4-[6-(1H-pyrazol-1-yl)pyrimidin-4-yl]-1H-pyrazol-1-yl}acetamide
ethyl 3-[(6-hydroxy-1,4-oxazepane-4-carbonyl)amino]-1-benzothiophene-2-carboxylate
2-(1-cyclopentyl-3-oxopiperazin-2-yl)-N-methyl-N-(4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)acetamide
N-{1-[1-(4-chloro-2-fluorobenzoyl)piperidin-4-yl]-1H-pyrazol-5-yl}-3-methylbutanamide
5-[2-(2H-1,3-benzodioxol-5-yl)acetyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxylic acid
6-(piperidin-1-yl)-N-[2-(1H-pyrazol-1-yl)ethyl]-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
3-{1-[4-(1H-imidazol-1-yl)benzoyl]piperidin-4-yl}-N-(3-methoxyphenyl)propanamide
4-{4-[3-(trifluoromethyl)phenoxy]piperidine-1-carbonyl}pyridine
1-[1-(1-tert-butyl-1H-pyrrole-3-carbonyl)piperidin-3-yl]-3-phenylpropan-1-one
2-[2-(1H-imidazol-4-yl)ethyl]-8-(4-methyl-1H-imidazole-2-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
{[4-(3-chlorophenyl)-5-[(pyridin-4-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}(methyl)(thiophen-3-ylmethyl)amine
N-{1-[4-(dimethylamino)phenyl]-3-hydroxypropan-2-yl}-3-propyl-1H-pyrazole-5-carboxamide
3-{2-[(3R,4R)-3-{[ethyl(methyl)amino]methyl}-4-(hydroxymethyl)pyrrolidin-1-yl]-2-oxoethyl}-5,5-dimethylimidazolidine-2,4-dione
2-(2,5-dioxoimidazolidin-1-yl)-N-[1-methyl-4-(morpholin-4-yl)-1H-indazol-3-yl]acetamide
N-methyl-N-[2-(oxan-2-yl)ethyl]pyridine-3-carboxamide
(4aS,8aR)-6-(4-cyclopentylpyrimidin-2-yl)-1-(4-hydroxybutyl)-decahydro-1,6-naphthyridin-2-one
(1R,3S)-7-{6-[ethyl(methyl)amino]pyrimidin-4-yl}-7-azaspiro[3.5]nonane-1,3-diol
4-(6-methyl-2H-1,3-benzodioxol-5-yl)-4H-1,2,4-triazole
[(2,3-difluoro-6-methoxyphenyl)methyl](ethyl)[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]amine
5-{1-[(1R,2S,4R)-bicyclo[2.2.1]hept-5-ene-2-carbonyl]piperidin-4-yl}-5-(pyridin-2-yl)-3-[2-(thiophen-2-yl)ethyl]imidazolidine-2,4-dione
2-(5-{2H,4H,5H,6H-cyclopenta[c]pyrazol-3-yl}-1,2,4-oxadiazol-3-yl)pyridine
1,3-dimethyl-5-[({[6-(pyrrolidine-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl}amino)methyl]-2,3-dihydro-1H-1,3-benzodiazol-2-one
2-methyl-5-(4-{5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl}piperazin-1-yl)-2,3-dihydropyridazin-3-one
7-cyclohexyl-2-[(4-methyl-1H-imidazol-2-yl)methyl]-2,7-diazaspiro[4.5]decan-6-one
N-({5-cyclohexyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)butane-1-sulfonamide
1-[(2,3-dimethoxyphenyl)methyl]-N-(4-fluorophenyl)piperidin-3-amine
2-{3-[3-(1H-1,3-benzodiazol-5-yl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl}acetamide
(5-{2-[5-(1H-pyrazol-3-yl)thiophen-2-yl]-1H-imidazol-1-yl}-1H-1,3-benzodiazol-2-yl)methanol
N-[1-(1-methyl-1H-pyrazol-5-yl)propyl]-1-(5-phenyl-1,3,4-thiadiazol-2-yl)piperidin-4-amine