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N-(2,4-dichloro-3-methylphenyl)-4-(dimethylamino)azepane-1-carboxamide
1-[2-(4-chlorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]-2-[(2-methoxyethyl)(methyl)amino]ethan-1-one
(3aS,6aS)-5-(2-cyclopentylacetyl)-1-oxo-2-(prop-2-en-1-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
5-{3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-2-phenylpyrimidine
5-{2-[4-(cyclohexylmethyl)-3-(2-hydroxyethyl)piperazin-1-yl]-2-oxoethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
6-ethyl-4-[2-(3-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl]-1,2-dihydropyridin-2-one
3-[1-(cyclohex-1-ene-1-carbonyl)piperidin-4-yl]-N-{[3-(trifluoromethyl)phenyl]methyl}propanamide
{[5-(1,5-dimethyl-1H-pyrrol-2-yl)-1,3,4-oxadiazol-2-yl]methyl}[2-methoxy-1-(1-methyl-1H-pyrazol-5-yl)ethyl]amine
1-{7-[(4-acetylpiperazin-1-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl}-3-(furan-2-yl)-3-phenylpropan-1-one
5-ethyl-1'-(quinoline-2-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
5-{1-[4-(dimethylamino)benzoyl]piperidin-4-yl}-5-ethyl-3-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]imidazolidine-2,4-dione
2-{5-[2-(2-methoxyethyl)pyrimidin-5-yl]-4-phenyl-1H-imidazol-1-yl}acetic acid
N-(1-methyl-1H-1,3-benzodiazol-5-yl)-4-(2-methylphenoxy)piperidine-1-carboxamide
1-({3-[1-(4-methylphenyl)cyclopentyl]-1,2,4-oxadiazol-5-yl}methyl)-4-(pyrimidin-2-yl)-1,4-diazepane
N-{1-[1-(2,4-difluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}-3-(2-ethyl-1H-imidazol-1-yl)propanamide
(3R,5R)-N-[2-(5-chloro-4-methyl-1,3-thiazol-2-yl)ethyl]-5-(morpholine-4-carbonyl)piperidine-3-carboxamide
1-(adamantan-1-yl)-4-(4-methyl-1,3-thiazole-5-carbonyl)piperazine
6-(azepan-1-yl)-N-ethyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]pyridine-3-carboxamide
1-{[4-(difluoromethoxy)phenyl]methyl}-3-(1-methyl-1H-imidazol-2-yl)piperidine
N-[2-(2,3-dihydro-1H-indol-1-yl)ethyl]-2-methyl-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
(3R,4R)-3-methyl-4-(oxan-4-yl)-1-[(5-propylfuran-2-yl)methyl]piperidin-4-ol
4-(1-{[3-(2,4-difluorophenyl)-1H-pyrazol-4-yl]methyl}piperidin-4-yl)pyridine
1-[3-(4-methoxy-2-methylphenyl)-1-methyl-1H-1,2,4-triazol-5-yl]piperidine
2-methyl-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-5-sulfamoylbenzamide
(3aR,6aS)-5-(2,3-dihydro-1-benzofuran-5-carbonyl)-1-oxo-2-propyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
5-(2-chloro-4-methoxyphenoxymethyl)-N-[(3-fluorophenyl)methyl]-1,2-oxazole-3-carboxamide
1-(cyclohexylmethyl)-N3-({5-methylimidazo[1,2-a]pyridin-2-yl}methyl)-4-oxo-N5-(propan-2-yl)-1,4-dihydropyridine-3,5-dicarboxamide
N-(1-butyl-4-methyl-1H-pyrazol-5-yl)-2-(4-oxo-3,4-dihydro-1,2,3-benzotriazin-3-yl)acetamide
N4-{[1-(3-methoxypropyl)pyrrolidin-3-yl]methyl}-6-methylpyrimidine-2,4-diamine
4-[1-(1,5-dimethyl-1H-pyrazole-3-carbonyl)pyrrolidin-3-yl]-1-(2-phenylethyl)piperidine
1-(4-methoxyphenyl)-3-methyl-4-{[2-(1H-pyrazol-1-yl)phenyl]methyl}piperazin-2-one
3-(butan-2-yl)-1-(2,3,4,9-tetrahydro-1H-carbazol-6-ylmethyl)urea
methyl 2-{[5-(4-fluorophenyl)-4-[1-(2-oxo-2-phenylacetyl)piperidin-3-yl]pyrimidin-2-yl]sulfanyl}acetate
(3S,4S)-4-cyclopropyl-1-(6-methylpyridazin-3-yl)pyrrolidine-3-carboxylic acid
N-benzyl-N-ethyl-2-{[4-(pyrimidin-2-yl)piperazin-1-yl]methyl}-1,3-oxazole-4-carboxamide
4-[(1R,3S)-1-hydroxy-3-(2-hydroxyethoxy)-7-azaspiro[3.5]nonan-7-yl]pyridine-2-carboxylic acid
N-[2-(2-ethoxyphenoxy)ethyl]-1-ethyl-N,4,6-trimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
N-[(2R,3R)-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2,5-dimethylfuran-3-carboxamide
1-{2-[(4S)-2-oxo-4-phenyl-1,3-oxazolidin-3-yl]acetyl}piperidine-4-carbonitrile
2,7-dimethyl-N-{[2-(pyrazin-2-yl)-1,3-thiazol-4-yl]methyl}-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
methyl (2S)-1-(4-{[(2,3-dimethoxyphenyl)methyl]amino}-5-methylthieno[2,3-d]pyrimidine-6-carbonyl)pyrrolidine-2-carboxylate
4-[4-(2-methanesulfonylethyl)piperazine-1-carbonyl]-2,6-dimethylquinoline
2-({[1-butyl-2-(4-methylpentanesulfonyl)-1H-imidazol-5-yl]methyl}(methyl)amino)ethan-1-ol
3-({1-[(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}oxy)pyridine
4-(3-fluorophenyl)-N-(oxolan-2-ylmethyl)-N-{[4-(pyridin-3-ylmethoxy)phenyl]methyl}benzamide
(1R,5R)-3-(4-chloro-1,3-dimethyl-1H-pyrazole-5-carbonyl)-6-(cyclobutylmethyl)-3,6-diazabicyclo[3.2.2]nonane
5-(3,4-dihydro-2H-1-benzopyran-3-carbonyl)-3-(2-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine
(2S,4R)-N-ethyl-1-(pyridine-4-carbonyl)-4-(3,3,3-trifluoropropanamido)pyrrolidine-2-carboxamide
{[1-(2-fluorophenyl)-3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}(methyl)[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]amine
2-[9-(3-methoxypyrazin-2-yl)-3-oxo-2,9-diazaspiro[5.5]undecan-2-yl]propanoic acid